Evaluation of a New Molecular Entity as a Victim of Metabolic Drug-Drug Interactions-an Industry Perspective
Bohnert, Tonika, Patel, Aarti, Templeton, Ian, Chen, Yuan, Lu, Chuang, Lai, George, Leung, Louis, Tse, Susanna, Einolf, Heidi J, Wang, Ying-Hong, Sinz, Michael, Stearns, Ralph, Walsky, Robert, Geng, Wanping, Sudsakorn, Sirimas, Moore, David, He, Ling, Wahlstrom, Jan, Keirns, Jim, Narayanan, Rangaraj, Lang, Dieter, Yang, Xiaoqing
Published in Drug metabolism and disposition (01.08.2016)
Published in Drug metabolism and disposition (01.08.2016)
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Journal Article
Contribution of itraconazole metabolites to inhibition of CYP3A4 in vivo
Templeton, I E, Thummel, K E, Kharasch, E D, Kunze, K L, Hoffer, C, Nelson, W L, Isoherranen, N
Published in Clinical pharmacology and therapeutics (01.01.2008)
Published in Clinical pharmacology and therapeutics (01.01.2008)
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Journal Article
Evaluation of 6β-hydroxycortisol, 6β-hydroxycortisone, and a combination of the two as endogenous probes for inhibition of CYP3A4 in vivo
Peng, C-C, Templeton, I, Thummel, K E, Davis, C, Kunze, K L, Isoherranen, N
Published in Clinical pharmacology and therapeutics (01.06.2011)
Published in Clinical pharmacology and therapeutics (01.06.2011)
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Journal Article
Quantitative Prediction of Drug–Drug Interactions Involving Inhibitory Metabolites in Drug Development: How Can Physiologically Based Pharmacokinetic Modeling Help?
Templeton, IE, Chen, Y, Mao, J, Lin, J, Yu, H, Peters, S, Shebley, M, Varma, MV
Published in CPT: pharmacometrics and systems pharmacology (01.10.2016)
Published in CPT: pharmacometrics and systems pharmacology (01.10.2016)
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Journal Article
Response to “Quantitative Prediction of Drug‐Drug Interactions Involving Inhibitory Metabolites by Physiologically Based Pharmacokinetic Models: Is It Worth?”
Templeton, IE, Chen, Y, Mao, J, Lin, J, Yu, H, Peters, S, Shebley, M, Varma, MV
Published in CPT: pharmacometrics and systems pharmacology (01.04.2017)
Published in CPT: pharmacometrics and systems pharmacology (01.04.2017)
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Journal Article
Compendium of gene expression profiles comprising a baseline model of the human liver drug metabolism transcriptome
Slatter, J. G., Templeton, I. E., Castle, J. C., Kulkarni, A., Rushmore, T. H., Richards, K., He, Y., Dai, X., Cheng, O. J., Caguyong, M., Ulrich, R. G.
Published in Xenobiotica (01.10.2006)
Published in Xenobiotica (01.10.2006)
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Journal Article
Evaluation of the pharmacokinetic (PK) profile of vismodegib (VISMO) in patients (pts) with multiple basal cell carcinomas (BCCs) across two intermittent treatment regimens in the MIKIE study
Schadendorf, D., Hauschild, A., Fosko, S., Zloty, D., Labeille, B., Grob, J.J., Puig, S., Makrutzki, M., Templeton, I., Rogers, G., Dreno, B., Kunstfeld, R.
Published in Annals of oncology (01.10.2016)
Published in Annals of oncology (01.10.2016)
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Journal Article
Grating demultiplexer integrated with MSM detector array in InGaAs/AlGaAs/GaAs for WDM
FALLAHI, M, MCGREER, K. A, DELAGE, A, TEMPLETON, I. M, CHATENOUD, F, BARBER, R
Published in IEEE photonics technology letters (01.07.1993)
Published in IEEE photonics technology letters (01.07.1993)
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Journal Article
Exposure of advanced positive and negative e-beam resists with focused ion beams
MATTIUSSI, G. A, SCANLON, P. J, TEMPLETON, I. M
Published in Journal of the Electrochemical Society (01.08.1993)
Published in Journal of the Electrochemical Society (01.08.1993)
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Journal Article
Electrically pumped circular-grating distributed-Bragg-reflector lasers
Wu, C.M., Svilans, M., Fallahi, M., Templeton, I., Makino, T., Glinski, J., Maciejko, R., Najafi, S.I., Blaauw, C., Maritan, C., Knight, D.G.
Published in IEEE photonics technology letters (01.09.1992)
Published in IEEE photonics technology letters (01.09.1992)
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Journal Article
Ridge waveguide quantum-well wavelength division demultiplexing detector with four channels
Moss, D., Ye, F., Landheer, D., Jessop, P.E., Simmons, J.G., Champion, H.G., Templeton, I., Chatenoud, F.
Published in IEEE photonics technology letters (01.07.1992)
Published in IEEE photonics technology letters (01.07.1992)
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Journal Article