C‑6α- vs C‑7α-Substituted Steroidal Aromatase Inhibitors: Which Is Better? Synthesis, Biochemical Evaluation, Docking Studies, and Structure–Activity Relationships
Roleira, Fernanda M. F, Varela, Carla, Amaral, Cristina, Costa, Saul C, Correia-da-Silva, Georgina, Moraca, Federica, Costa, Giosuè, Alcaro, Stefano, Teixeira, Natércia A. A, Tavares da Silva, Elisiário J
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Published in Journal of medicinal chemistry (11.04.2019)
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Synthetic cannabinoids JWH-018, JWH-122, UR-144 and the phytocannabinoid THC activate apoptosis in placental cells
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Published in Toxicology letters (01.02.2020)
Published in Toxicology letters (01.02.2020)
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Synthetic cannabinoids and endometrial stromal cell fate: Dissimilar effects of JWH-122, UR-144 and WIN55,212-2
Fonseca, Bruno M., Fernandes, Renata, Almada, Marta, Santos, Márcia, Carvalho, Félix, Teixeira, Natércia A., Correia-da-Silva, Georgina
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New Structure–Activity Relationships of A- and D-Ring Modified Steroidal Aromatase Inhibitors: Design, Synthesis, and Biochemical Evaluation
Varela, Carla, Tavares da Silva, Elisiário J, Amaral, Cristina, Correia da Silva, Georgina, Baptista, Teresa, Alcaro, Stefano, Costa, Giosuè, Carvalho, Rui A, Teixeira, Natércia A. A, Roleira, Fernanda M. F
Published in Journal of medicinal chemistry (26.04.2012)
Published in Journal of medicinal chemistry (26.04.2012)
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Spatio-temporal expression patterns of anandamide-binding receptors in rat implantation sites: evidence for a role of the endocannabinoid system during the period of placental development
Fonseca, Bruno M, Correia-da-Silva, Georgina, Taylor, Anthony H, Konje, Justin C, Bell, Stephen C, Teixeira, Natércia A
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Published in Reproductive biology and endocrinology (27.10.2009)
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Design, synthesis and biochemical studies of new 7α-allylandrostanes as aromatase inhibitors
Varela, Carla L., Amaral, Cristina, Correia-da-Silva, Georgina, Carvalho, Rui A., Teixeira, Natércia A., Costa, Saul C., Roleira, Fernanda M.F., Tavares-da-Silva, Elisiário J.
Published in Steroids (01.07.2013)
Published in Steroids (01.07.2013)
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Characterisation of the endocannabinoid system in rat haemochorial placenta
Fonseca, Bruno M., Correia-da-Silva, Georgina, Taylor, Anthony H., Lam, Patricia M.W., Marczylo, Timothy H., Konje, Justin C., Teixeira, Natércia A.
Published in Reproductive toxicology (Elmsford, N.Y.) (01.11.2012)
Published in Reproductive toxicology (Elmsford, N.Y.) (01.11.2012)
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Structure−Activity Relationships of New A,D-Ring Modified Steroids as Aromatase Inhibitors: Design, Synthesis, and Biological Activity Evaluation
Cepa, Margarida M. D. S, Tavares da Silva, Elisiário J, Correia-da-Silva, Georgina, Roleira, Fernanda M. F, Teixeira, Natércia A. A
Published in Journal of medicinal chemistry (06.10.2005)
Published in Journal of medicinal chemistry (06.10.2005)
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Insights into the Synthesis of Steroidal A-Ring Olefins
Varela, Carla L., Roleira, Fernanda M. F., Costa, Saul C. P., Pinto, Alexandra S. C. T., Martins, Ana I. O. S., Carvalho, Rui A., Teixeira, Natércia A., Correia-da-Silva, Georgina, Tavares-da-Silva, Elisiário
Published in Helvetica chimica acta (01.01.2014)
Published in Helvetica chimica acta (01.01.2014)
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Molecular mechanisms of aromatase inhibition by new A, D-ring modified steroids
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Published in Biological chemistry (01.09.2008)
Published in Biological chemistry (01.09.2008)
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Exploring new chemical functionalities to improve aromatase inhibition of steroids
Varela, Carla L., Amaral, Cristina, Correia-da-Silva, Georgina, Costa, Saul C., Carvalho, Rui A., Costa, Giosuè, Alcaro, Stefano, Teixeira, Natércia A.A., Tavares-da-Silva, Elisiário J., Roleira, Fernanda M.F.
Published in Bioorganic & medicinal chemistry (15.06.2016)
Published in Bioorganic & medicinal chemistry (15.06.2016)
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Erythrocyte membrane band 3 profile imposed by cellular aging, by activated neutrophils and by neutrophilic elastase
Santos-Silva, Alice, Castro, Elisabeth M.B, Teixeira, Natércia A, Guerra, Francisco Carvalho, Quintanilha, Alexandre
Published in Clinica chimica acta (28.07.1998)
Published in Clinica chimica acta (28.07.1998)
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Synthesis and biochemical studies of 17-substituted androst-3-enes and 3,4-epoxyandrostanes as aromatase inhibitors
Cepa, Margarida M.D.S., Tavares da Silva, Elisiário J., Correia-da-Silva, Georgina, Roleira, Fernanda M.F., Teixeira, Natércia A.A.
Published in Steroids (22.12.2008)
Published in Steroids (22.12.2008)
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Lipidomic approach towards deciphering anandamide effects in rat decidual cell: ANANDAMIDE'S EFFECT ON DECIDUAL PHOSPHOLIPIDOME
Almada, Marta, Domingues, M. Rosário, Dória, M. Luísa, Fonseca, Bruno M., Teixeira, Natércia A., Correia-da-Silva, Georgina
Published in Journal of cellular physiology (01.07.2015)
Published in Journal of cellular physiology (01.07.2015)
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New steroidal aromatase inhibitors: suppression of estrogen-dependent breast cancer cell proliferation and induction of cell death
Cepa, Margarida, Correia-da-Silva, Georgina, da Silva, Elisiário J Tavares, Roleira, Fernanda M F, Borges, Margarida, Teixeira, Natércia A
Published in BMC cell biology (24.07.2008)
Published in BMC cell biology (24.07.2008)
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Metabolic fate of AMP, IMP, GMP and XMP in the cytosol of rat brain: an experimental and theoretical analysis
Torrecilla, Amparo, Marques, Agostinho F. P., Buscalioni, Rafael D., Oliveira, Jorge M. A., Teixeira, Natercia A., Atencia, Eva Ana, Günther Sillero, María A., Sillero, Antonio
Published in Journal of neurochemistry (01.03.2001)
Published in Journal of neurochemistry (01.03.2001)
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Patterns of expression of Bax, Bcl-2 and Bcl-xL in the implantation site in rat during pregnancy
CORREIA-DA-SILVA, G, BELL, S. C, PRINGLE, J. H, TEIXEIRA, N. A
Published in Placenta (Eastbourne) (01.11.2005)
Published in Placenta (Eastbourne) (01.11.2005)
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