Identification of a novel series of potent and selective CCR6 inhibitors as biological probes
Tawaraishi, Taisuke, Sakauchi, Nobuki, Hidaka, Kousuke, Yoshikawa, Kyoko, Okui, Toshitake, Kuno, Haruhiko, Chisaki, Ikumi, Aso, Kazuyoshi
Published in Bioorganic & medicinal chemistry letters (01.10.2018)
Published in Bioorganic & medicinal chemistry letters (01.10.2018)
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Collaborative Virtual Screening Identifies a 2‑Aryl-4-aminoquinazoline Series with Efficacy in an In Vivo Model of Trypanosoma cruzi Infection
Tawaraishi, Taisuke, Ochida, Atsuko, Akao, Yuichiro, Itono, Sachiko, Kamaura, Masahiro, Akther, Thamina, Shimada, Mitsuyuki, Canan, Stacie, Chowdhury, Sanjoy, Cao, Yafeng, Condroski, Kevin, Engkvist, Ola, Francisco, Amanda, Ghosh, Sunil, Kaki, Rina, Kelly, John M., Kimura, Chiaki, Kogej, Thierry, Nagaoka, Kazuya, Naito, Akira, Pairaudeau, Garry, Radu, Constantin, Roberts, Ieuan, Shum, David, Watanabe, Nao-aki, Xie, Huanxu, Yonezawa, Shuji, Yoshida, Osamu, Yoshida, Ryu, Mowbray, Charles, Perry, Benjamin
Published in Journal of medicinal chemistry (26.01.2023)
Published in Journal of medicinal chemistry (26.01.2023)
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헤테로시클릭 NMDA 길항제
AIDA JUMPEI, NAKAMURA MINORU, YUKAWA TAKAFUMI, OGURO YUYA, YAMAGUCHI FUMIE, TAWARAISHI TAISUKE, IKEDA SHUHEI, KAMATA MAKOTO, IWANAGA KOUICHI, MURAKAMI MASATAKA, OCHIDA ATSUKO, OYABU NORIO, WAKABAYASHI TAKESHI, YAMAMOTO SATOSHI
Year of Publication 20.07.2022
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Year of Publication 20.07.2022
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HETEROCYCLIC COMPOUNDS AND USES THEREOF
NAKAMURA MINORU, OGURO YUYA, YAMAGUCHI FUMIE, TAWARAISHI TAISUKE, IKEDA SHUHEI, WAKABAYASHI KENJI, OCHITA ATSUKO, AIDA JUNPEI, YAMAMOTO TETSUSHI, KAMATA MAKOTO, IWANAGA KOICHI, MURAKAMI MASATAKA, OYABU NORIO, YUKAWA TAKESHI
Year of Publication 27.05.2021
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Year of Publication 27.05.2021
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Structure–activity relationships and key structural feature of pyridyloxybenzene-acylsulfonamides as new, potent, and selective peroxisome proliferator-activated receptor (PPAR) γ Agonists
Rikimaru, Kentaro, Wakabayashi, Takeshi, Abe, Hidenori, Tawaraishi, Taisuke, Imoto, Hiroshi, Yonemori, Jinichi, Hirose, Hideki, Murase, Katsuhito, Matsuo, Takanori, Matsumoto, Mitsuharu, Nomura, Chisako, Tsuge, Hiroko, Arimura, Naoto, Kawakami, Kazutoshi, Sakamoto, Junichi, Funami, Miyuki, Mol, Clifford D., Snell, Gyorgy P., Bragstad, Kenneth A., Sang, Bi-Ching, Dougan, Douglas R., Tanaka, Toshimasa, Katayama, Nozomi, Horiguchi, Yoshiaki, Momose, Yu
Published in Bioorganic & medicinal chemistry (15.05.2012)
Published in Bioorganic & medicinal chemistry (15.05.2012)
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헤테로사이클릭 화합물 및 이의 용도
AIDA JUMPEI, NAKAMURA MINORU, TAKAMI KAZUAKI, MORIMOTO SHINJI, OGURO YUYA, ITO MITSUHIRO, TAWARAISHI TAISUKE, MIKAMI SATOSHI, TAKASHIMA SACHIE, MATSUMOTO SHIGEMITSU, WADA YASUFUMI, KAMATA MAKOTO, DAINI MASAKI, KAKEI HIROYUKI, KAMEI TAKU, MURAKAMI MASATAKA, IWANAGA KOUICHI, WAKABAYASHI TAKESHI, NAKAMURA SHINJI, TOKUNAGA NORIHITO, SETO MASAKI, YAMAMOTO SATOSHI
Year of Publication 08.12.2020
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Year of Publication 08.12.2020
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CYCLIC DINUCLEOTIDE AS STING (STIMULATOR OF INTERFERON GENES) AGONIST
SAITO MORIHISA, SHIOKAWA ZENYU, MURATA SHUMPEI, SEDO MASAKI, YOSHIKAWA MASATO, PAUL D GREENSPAN, YOSHITOMI YAYOI, TAWARAISHI TAISUKE, ODA TSUNEO, NAKADA YOSHIHISA, OKANIWA MASANORI, OKABE ATSUTOSHI, WADA YASUFUMI, MOCHIZUKI MICHIYO, KATO TAISUKE, SASAKI YUSUKE, HIDAKA KOSUKE, TOMINARI YUSUKE, SHIBUYA AKITO, SEKI MICHIHIRO, NAKAGAWA YASUO, BRIAN SCOTT FREEZE
Year of Publication 09.04.2020
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Year of Publication 09.04.2020
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STING 작용제로서의 환식 다이뉴클레오타이드
GREENSPAN PAUL D, SHIOKAWA ZENYU, MURATA SHUMPEI, SEKI TOMOHIRO, YOSHIKAWA MASATO, YOSHITOMI YAYOI, TAWARAISHI TAISUKE, ODA TSUNEO, NAKADA YOSHIHISA, OKANIWA MASANORI, OKABE ATSUTOSHI, WADA YASUFUMI, MOCHIZUKI MICHIYO, KATO TAISUKE, SASAKI YUSUKE, HIDAKA KOSUKE, SAITOH MORIHISA, TOMINARI YUSUKE, SHIBUYA AKITO, FREEZE BRIAN SCOTT, SETO MASAKI, NAKAGAWA YASUO
Year of Publication 08.10.2019
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Year of Publication 08.10.2019
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HETEROCYCLIC NMDA ANTAGONISTS
OCHIDA, Atsuko, AIDA, Jumpei, IWANAGA, Kouichi, YAMAMOTO, Satoshi, YAMAGUCHI, Fumie, NAKAMURA, Minoru, KAMATA, Makoto, TAWARAISHI, Taisuke, WAKABAYASHI, Takeshi, MURAKAMI, Masataka, OYABU, Norio, OGURO, Yuya, YUKAWA, Takafumi, IKEDA, Shuhei
Year of Publication 18.05.2023
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Year of Publication 18.05.2023
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HETEROCYCLIC NMDA ANTAGONISTS
OCHIDA, Atsuko, AIDA, Jumpei, IWANAGA, Kouichi, YAMAMOTO, Satoshi, YAMAGUCHI, Fumie, NAKAMURA, Minoru, KAMATA, Makoto, TAWARAISHI, Taisuke, WAKABAYASHI, Takeshi, MURAKAMI, Masataka, OYABU, Norio, OGURO, Yuya, YUKAWA, Takafumi, IKEDA, Shuhei
Year of Publication 04.05.2023
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Year of Publication 04.05.2023
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HETEROCYCLIC NMDA ANTAGONISTS
OCHIDA, Atsuko, AIDA, Jumpei, IWANAGA, Kouichi, YAMAMOTO, Satoshi, YAMAGUCHI, Fumie, NAKAMURA, Minoru, KAMATA, Makoto, TAWARAISHI, Taisuke, WAKABAYASHI, Takeshi, MURAKAMI, Masataka, OYABU, Norio, OGURO, Yuya, YUKAWA, Takafumi, IKEDA, Shuhei
Year of Publication 05.01.2023
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Year of Publication 05.01.2023
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HETEROCYCLIC NMDA ANTAGONISTS
OCHIDA, Atsuko, AIDA, Jumpei, IWANAGA, Kouichi, YAMAMOTO, Satoshi, YAMAGUCHI, Fumie, NAKAMURA, Minoru, KAMATA, Makoto, TAWARAISHI, Taisuke, WAKABAYASHI, Takeshi, MURAKAMI, Masataka, OYABU, Norio, OGURO, Yuya, YUKAWA, Takafumi, IKEDA, Shuhei
Year of Publication 21.09.2022
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Year of Publication 21.09.2022
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Heterocyclic NMDA antagonists
OCHIDA, Atsuko, AIDA, Jumpei, IWANAGA, Kouichi, YAMAMOTO, Satoshi, YAMAGUCHI, Fumie, NAKAMURA, Minoru, KAMATA, Makoto, TAWARAISHI, Taisuke, WAKABAYASHI, Takeshi, MURAKAMI, Masataka, OYABU, Norio, OGURO, Yuya, YUKAWA, Takafumi, IKEDA, Shuhei
Year of Publication 30.06.2022
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Year of Publication 30.06.2022
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RECEPTOR AGONISTS
KANZAKI, NAOYUKI, MIKI, TAKASHI, HINUMA, SHUJI, KAWAMATA, YUJI, HIROHASHI, MARIKO, OI, SATORU, ISHICHI, YUJI, TAWARAISHI, TAISUKE, ITOH, FUMIO
Year of Publication 12.08.2004
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Year of Publication 12.08.2004
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HETEROCYCLIC NMDA ANTAGONISTS
OCHIDA, Atsuko, AIDA, Jumpei, IWANAGA, Kouichi, YAMAMOTO, Satoshi, YAMAGUCHI, Fumie, NAKAMURA, Minoru, KAMATA, Makoto, TAWARAISHI, Taisuke, WAKABAYASHI, Takeshi, MURAKAMI, Masataka, OYABU, Norio, OGURO, Yuya, YUKAWA, Takafumi, IKEDA, Shuhei
Year of Publication 02.06.2022
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Year of Publication 02.06.2022
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ANTIBODY-DRUG CONJUGATES COMPRISING A CYCLIC DINUCLEOTIDE
SEKI, TOMOHIRO, SHIOKAWA, ZENYU, TOMINARI, YUSUKE, SHIBUYA, AKITO, MOCHIZUKI, MICHIYO, NAKAGAWA, YASUO, MURATA, SHUMPEI, NAKAYAMA, YAYOI, OKABE, ATSUTOSHI, SASAKI, YUSUKE, FREEZE, BRIAN SCOTT, GREENSPAN, PAUL D, KATO, TAISUKE, HIDAKA, KOSUKE, NAKADA, YOSHIHISA, SAITOH, MORIHISA, OKANIWA, MASANORI, SETO, MASAKI, YOSHIKAWA, MASATO, ODA, TSUNEO, TAWARAISHI, TAISUKE, WADA, YASUFUMI
Year of Publication 29.02.2024
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Year of Publication 29.02.2024
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Heterocyclic compound and use thereof
Tokunaga, Norihito, Seto, Masaki, Ito, Mitsuhiro, Daini, Masaki, Iwanaga, Kouichi, Kamata, Makoto, Takami, Kazuaki, Wakabayashi, Takeshi, Morimoto, Shinji, Matsumoto, Shigemitsu, Kamei, Taku, Murakami, Masataka, Mikami, Satoshi, Takashima, Sachie, Tawaraishi, Taisuke, Nakamura, Shinji, Yamamoto, Satoshi, Wada, Yasufumi, Kakei, Hiroyuki, Oguro, Yuya, Aida, Jumpei, Nakamura, Minoru
Year of Publication 18.07.2023
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Year of Publication 18.07.2023
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Antibody-drug conjugates comprising a cyclic dinucleotide
Seto, Masaki, Shiokawa, Zenyu, Kato, Taisuke, Saitoh, Morihisa, Hidaka, Kosuke, Freeze, Brian Scott, Tominari, Yusuke, Oda, Tsuneo, Mochizuki, Michiyo, Nakayama, Yayoi, Nakagawa, Yasuo, Murata, Shumpei, Okaniwa, Masanori, Yoshikawa, Masato, Tawaraishi, Taisuke, Wada, Yasufumi, Seki, Tomohiro, Nakada, Yoshihisa, Okabe, Atsutoshi, Shibuya, Akito, Sasaki, Yusuke, Greenspan, Paul D
Year of Publication 06.06.2023
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Year of Publication 06.06.2023
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