PRELIMINARY CLINICAL DATA FROM A PHASE 1B STUDY OF MAVORIXAFOR AND IBRUTINIB IN PATIENTS WITH WALDENSTRöM MACROGLOBULINEMIA WITH MYD88 AND CXCR4 MUTATIONS
Treon, S., Buske, C., Thomas, S., Branagan, A., Dimopoulos, M., Castillo, J. J., Garzon, F., Tang, W., Ronan, R., Seyffert, S., Garg, V., Ali, S., Taveras, A., Badarau, A., Zmajkovicova, K., Maier, S., Maierhofer, B., Matous, J.
Published in Hematological oncology (01.06.2021)
Published in Hematological oncology (01.06.2021)
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P792: CRISPR/CAS9‐BASED MODEL OF HETEROZYGOUS CXCR4 WT/R334X MUTATION TO STUDY CELLULAR PHENOTYPES IN WHIM SYNDROME
Zmajkovicova, K., Pawar, S., Maier‐Munsa, S., Badarau, A., Taveras, A. G.
Published in HemaSphere (23.06.2022)
Published in HemaSphere (23.06.2022)
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P793: SCREENING OF NATURALLY OCCURRING CXCR4 VARIANTS FOR IDENTIFICATION OF NOVEL PATHOGENIC MUTATIONS FOR WHIM SYNDROME
Pawar, S., Wiest, I., Maier-Munsa, S., Maierhofer, B., Sondheimer, N., Taveras, A. G., Badarau, A., Zmajkovicova, K.
Published in HemaSphere (23.06.2022)
Published in HemaSphere (23.06.2022)
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P1253: MAVORIXAFOR DISRUPTS THE CROSS TALK BETWEEN WALDENSTRÖM'S MACROGLOBULINEMIA CELLS AND THE BONE MARROW MICROENVIRONMENT RESULTING IN ENHANCED SENSITIVITY TO B‐CELL TARGETED THERAPIES
Monticelli, H., Kruitwagen, T., Tardelli, M., Rebelo, T., Maierhofer, B., Maier‐Munsa, S., Zmajkovicova, K., Taveras, A. G., Nguyen, C.
Published in HemaSphere (23.06.2022)
Published in HemaSphere (23.06.2022)
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The farnesyl transferase inhibitor SCH 66336 induces a G(2) --> M or G(1) pause in sensitive human tumor cell lines
Ashar, H R, James, L, Gray, K, Carr, D, McGuirk, M, Maxwell, E, Black, S, Armstrong, L, Doll, R J, Taveras, A G, Bishop, W R, Kirschmeier, P
Published in Experimental cell research (01.01.2001)
Published in Experimental cell research (01.01.2001)
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Ras oncoprotein inhibitors: The discovery of potent, ras nucleotide exchange inhibitors and the structural determination of a drug-protein complex
Taveras, A.G., Remiszewski, S.W., Doll, R.J., Cesarz, D., Huang, E.C., Kirschmeier, P., Pramanik, B.N., Snow, M.E., Wang, Y.-S., del Rosario, J.D., Vibulbhan, B., Bauer, B.B., Brown, J.E., Carr, D., Catino, J., Evans, C.A., Girijavallabhan, V., Heimark, L., James, L., Liberles, S., Nash, C., Perkins, L., Senior, M.M., Tsarbopoulos, A., Ganguly, A.K., Aust, R., Brown, E., Delisle, D., Fuhrman, S., Hendrickson, T., Kissinger, C., Love, R., Sisson, W., Villafranca, E., Webber, S.E.
Published in Bioorganic & medicinal chemistry (01.01.1997)
Published in Bioorganic & medicinal chemistry (01.01.1997)
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Surface finish mechanics explain different clinical survivorship of cemented femoral stems for total hip arthroplasty
Beksac, Burak, Taveras, Nicole A, Valle, Alejandro Gonzalez Della, Salvati, Eduardo A
Published in Journal of long-term effects of medical implants (2006)
Published in Journal of long-term effects of medical implants (2006)
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Antitumor 8-chlorobenzocycloheptapyridines: a new class of selective, nonpeptidic, nonsulfhydryl inhibitors of ras farnesylation
Mallams, A.K., Njoroge, F.G., Doll, R.J., Snow, M.E., Kaminski, J.J., Rossman, R.R., Vibulbhan, B., Bishop, W.R., Kirschmeier, P., Liu, M., Bryant, M.S., Alvarez, C., Carr, D., James, L., King, I., Li, Z., Lin, C.-C., Nardo, C., Petrin, J., Remiszewski, S.W., Taveras, A.G., Wang, S., Wong, J., Catino, J., Girijavallabhan, V., Ganguly, A.K.
Published in Bioorganic & medicinal chemistry (01.01.1997)
Published in Bioorganic & medicinal chemistry (01.01.1997)
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Biological Effects and Mechanism of Action of Farnesyl Transferase Inhibitors
Ashar, Hena R, Armstrong, Lydia, James, Linda J, Carr, Donna M, Gray, Kimberley, Taveras, Arthur, Doll, Ronald J, Bishop, W. Robert, Kirschmeier, Paul T
Published in Chemical research in toxicology (16.10.2000)
Published in Chemical research in toxicology (16.10.2000)
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Detection and structural characterization of ras oncoprotein-inhibitors complexes by electrospray mass spectrometry
Ganguly, A.K., Pramanik, B.N., Huang, E.C., Liberles, S., Heimark, L., Liu, Y.H., Tsarbopoulos, A., Doll, R.J., Taveras, A.G., Remiszewski, S., Snow, M.E., Wang, Y.S., Vibulbhan, B., Cesarz, D., Brown, J.E., del Rosario, J., James, L., Kirschmeier, P., Girijavallabhan, V.
Published in Bioorganic & medicinal chemistry (01.05.1997)
Published in Bioorganic & medicinal chemistry (01.05.1997)
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P793: SCREENING OF NATURALLY OCCURRING CXCR4 VARIANTS FOR IDENTIFICATION OF NOVEL PATHOGENIC MUTATIONS FOR WHIM SYNDROME
Pawar, S., Wiest, I., Maier‐Munsa, S., Maierhofer, B., Sondheimer, N., Taveras, A. G., Badarau, A., Zmajkovicova, K.
Published in HemaSphere (01.06.2022)
Published in HemaSphere (01.06.2022)
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Antitumor activity of SCH 66336, an orally bioavailable tricyclic inhibitor of farnesyl protein transferase, in human tumor xenograft models and Wap-ras transgenic mice
MING LIU, BRYANT, M. S, DELL, J, SINHA, D, SYED, J, KORFMACHER, W. A, NOMEIR, A. A, LIN, C.-C, WANG, L, TAVERAS, A. G, DOLL, R. J, NJOROGE, F. G, JIANPING CHEN, MALLAMS, A. K, REMISZEWSKI, S, CATINO, J. J, GIRIJAVALLABHAN, V. M, KIRSCHMEIER, P, BISHOP, W. R, SUINING LEE, YAREMKO, B, LIPARI, P, MALKOWSKI, M, FERRARI, E, NIELSEN, L, PRIOLI, N
Published in Cancer research (Chicago, Ill.) (01.11.1998)
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Published in Cancer research (Chicago, Ill.) (01.11.1998)
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Solid-state photochemistry. Remarkable effects of the packing of molecules in crystals on the diastereoselectivity of the intramolecular 2 + 2 photocycloaddition of a 4-(3'-butenyl)-2,5-cyclohexadien-1-one
Schultz, Arthur G, Taveras, Arthur G, Taylor, Richard E, Tham, Fook S, Kullnig, Rudolph K
Published in Journal of the American Chemical Society (01.10.1992)
Published in Journal of the American Chemical Society (01.10.1992)
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P60 DISCOVERY OF POTENT MMP-13 SPECIFIC INHIBITOR WITHOUT MUSCULOSKELETAL SIDE EFFECTS
Piecha, D., Baragi, V., Jaworski, A., Korniski, B., Nix, D., Powers, T., Steeneck, C., Taveras, A., VanVelduizen, J., Weik, J., Hofmann, M.
Published in Osteoarthritis and cartilage (2006)
Published in Osteoarthritis and cartilage (2006)
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Tricyclic Farnesyl Protein Transferase Inhibitors: Crystallographic and Calorimetric Studies of Structure−Activity Relationships
Strickland, Corey L, Weber, Patricia C, Windsor, William T, Wu, Zhen, Le, Hung V, Albanese, Margaret M, Alvarez, Carmen S, Cesarz, David, del Rosario, Joycelyn, Deskus, Jeffrey, Mallams, Alan K, Njoroge, F. George, Piwinski, John J, Remiszewski, Stacy, Rossman, Randall R, Taveras, Arthur G, Vibulbhan, Bancha, Doll, Ronald J, Girijavallabhan, Viyyoor M, Ganguly, Ashit K
Published in Journal of medicinal chemistry (17.06.1999)
Published in Journal of medicinal chemistry (17.06.1999)
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