Identification of Breast Cancer Inhibitors Specific for G Protein‐Coupled Estrogen Receptor (GPER)‐Expressing Cells
Aiello, Francesca, Carullo, Gabriele, Giordano, Francesca, Spina, Elena, Nigro, Alessandra, Garofalo, Antonio, Tassini, Sabrina, Costantino, Gabriele, Vincetti, Paolo, Bruno, Agostino, Radi, Marco
Published in ChemMedChem (22.08.2017)
Published in ChemMedChem (22.08.2017)
Get full text
Journal Article
From High-Throughput Screening to Target Validation: Benzo[d]isothiazoles as Potent and Selective Agonists of Human Transient Receptor Potential Cation Channel Subfamily M Member 5 Possessing In Vivo Gastrointestinal Prokinetic Activity in Rodents
Barilli, Alessio, Aldegheri, Laura, Bianchi, Federica, Brault, Laurent, Brodbeck, Daniela, Castelletti, Laura, Feriani, Aldo, Lingard, Iain, Myers, Richard, Nola, Selena, Piccoli, Laura, Pompilio, Daniela, Raveglia, Luca F, Salvagno, Cristian, Tassini, Sabrina, Virginio, Caterina, Sabat, Mark
Published in Journal of medicinal chemistry (13.05.2021)
Published in Journal of medicinal chemistry (13.05.2021)
Get full text
Journal Article
Multitarget CFTR Modulators Endowed with Multiple Beneficial Side Effects for Cystic Fibrosis Patients: Toward a Simplified Therapeutic Approach
Tassini, Sabrina, Langron, Emily, Delang, Leen, Mirabelli, Carmen, Lanko, Kristina, Crespan, Emmanuele, Kissova, Miroslava, Tagliavini, Giulia, Fontò, Greta, Bertoni, Simona, Palese, Simone, Giorgio, Carmine, Ravanetti, Francesca, Ragionieri, Luisa, Zamperini, Claudio, Mancini, Arianna, Dreassi, Elena, Maga, Giovanni, Vergani, Paola, Neyts, Johan, Radi, Marco
Published in Journal of medicinal chemistry (12.12.2019)
Published in Journal of medicinal chemistry (12.12.2019)
Get full text
Journal Article
Discovery of Multitarget Agents Active as Broad-Spectrum Antivirals and Correctors of Cystic Fibrosis Transmembrane Conductance Regulator for Associated Pulmonary Diseases
Tassini, Sabrina, Sun, Liang, Lanko, Kristina, Crespan, Emmanuele, Langron, Emily, Falchi, Federico, Kissova, Miroslava, Armijos-Rivera, Jorge I, Delang, Leen, Mirabelli, Carmen, Neyts, Johan, Pieroni, Marco, Cavalli, Andrea, Costantino, Gabriele, Maga, Giovanni, Vergani, Paola, Leyssen, Pieter, Radi, Marco
Published in Journal of medicinal chemistry (23.02.2017)
Published in Journal of medicinal chemistry (23.02.2017)
Get full text
Journal Article
A combined ligand- and structure-based approach for the identification of rilmenidine-derived compounds which synergize the antitumor effects of doxorubicin
Vucicevic, Jelica, Srdic-Rajic, Tatjana, Pieroni, Marco, Laurila, Jonne M.M., Perovic, Vladimir, Tassini, Sabrina, Azzali, Elisa, Costantino, Gabriele, Glisic, Sanja, Agbaba, Danica, Scheinin, Mika, Nikolic, Katarina, Radi, Marco, Veljkovic, Nevena
Published in Bioorganic & medicinal chemistry (15.07.2016)
Published in Bioorganic & medicinal chemistry (15.07.2016)
Get full text
Journal Article
Identification of Breast Cancer Inhibitors Specific for GProtein-Coupled Estrogen Receptor (GPER)-Expressing Cells
Aiello, Francesca, Carullo, Gabriele, Giordano, Francesca, Spina, Elena, Nigro, Alessandra, Garofalo, Antonio, Tassini, Sabrina, Costantino, Gabriele, Vincetti, Paolo, Bruno, Agostino, Radi, Marco
Published in ChemMedChem (01.08.2017)
Published in ChemMedChem (01.08.2017)
Get full text
Journal Article
A multicomponent pharmacophore fragment-decoration approach to identify selective LRRK2-targeting probes
Tassini, Sabrina, Castagnolo, Daniele, Scalacci, Nicolo, Kissova, Miroslava, Armijos-Rivera, Jorge I., Giagnorio, Federica, Maga, Giovanni, Costantino, Gabriele, Crespan, Emmanuele, Radi, Marco
Published in MedChemComm (16.03.2016)
Published in MedChemComm (16.03.2016)
Get full text
Journal Article
A multicomponent pharmacophore fragment-decoration approach to identify selective LRRK2-targeting probesThe authors declare no competing interest.Electronic supplementary information (ESI) available: Experimental procedures and analytical data for compounds 9 and 10, in vitro LRRK2 inhibition assays, inhibition mechanism and kinase panel data. See DOI: 10.1039/c5md00462d
Tassini, Sabrina, Castagnolo, Daniele, Scalacci, Nicolò, Kissova, Miroslava, Armijos-Rivera, Jorge I, Giagnorio, Federica, Maga, Giovanni, Costantino, Gabriele, Crespan, Emmanuele, Radi, Marco
Year of Publication 16.03.2016
Year of Publication 16.03.2016
Get full text
Journal Article
HETEROCYCLIC COMPOUNDS AS DELTA-5 DESATURASE INHIBITORS AND METHODS OF USE
SIEGMUND, Aaron C, AMEGADZIE, Albert, POZZAN, Alfonso, REEVES, Corey, BOURBEAU, Matthew P, MINATTI, Ana E, TASSINI, Sabrina, ALLEN, Jennifer R, TONELLI, Federica, MA, Vu Van, LATTANZI, Giulia, WALTON, Mary, GOODMAN, Clifford, LINGARD, Iain, CHEN, Ning, LIU, Qingyian, LOW, Jonathan D
Year of Publication 05.10.2022
Get full text
Year of Publication 05.10.2022
Patent
Heterocyclic compounds as Delta-5 Desaturase inhibitors and methods of use
SIEGMUND, Aaron C, AMEGADZIE, Albert, POZZAN, Alfonso, REEVES, Corey, BOURBEAU, Matthew P, MINATTI, Ana E, TASSINI, Sabrina, ALLEN, Jennifer R, TONELLI, Federica, MA, Vu Van, LATTANZI, Giulia, WALTON, Mary, GOODMAN, Clifford, LINGARD, Iain, CHEN, Ning, LIU, Qingyian, LOW, Jonathan D
Year of Publication 09.06.2022
Get full text
Year of Publication 09.06.2022
Patent
HETEROCYCLIC COMPOUNDS AS DELTA-5 DESATURASE INHIBITORS AND METHODS OF USE
SIEGMUND, Aaron C, AMEGADZIE, Albert, POZZAN, Alfonso, REEVES, Corey, BOURBEAU, Matthew P, MINATTI, Ana E, TASSINI, Sabrina, ALLEN, Jennifer R, TONELLI, Federica, MA, Vu Van, LATTANZI, Giulia, WALTON, Mary, GOODMAN, Clifford, LINGARD, Iain, CHEN, Ning, LIU, Qingyian, LOW, Jonathan D
Year of Publication 10.06.2021
Get full text
Year of Publication 10.06.2021
Patent
HETEROCYCLIC COMPOUNDS AS DELTA-5 DESATURASE INHIBITORS AND METHODS OF USE
TONELLI, FEDERICA, CHEN, NING, LIU, QINGYIAN, ALLEN, JENNIFER R, LOW, JONATHAN D, MA, VU VAN, POZZAN, ALFONSO, WALTON, MARY, GOODMAN, CLIFFORD, LINGARD, IAIN, LATTANZI, GIULIA, MINATTI, ANA E, BOURBEAU, MATTHEW P, SIEGMUND, AARON C, AMEGADZIE, ALBERT, REEVES, COREY, TASSINI, SABRINA
Year of Publication 03.06.2021
Get full text
Year of Publication 03.06.2021
Patent
HETEROCYCLIC COMPOUNDS AS DELTA-5 DESATURASE INHIBITORS AND METHODS OF USE
SIEGMUND, Aaron C, AMEGADZIE, Albert, POZZAN, Alfonso, REEVES, Corey, BOURBEAU, Matthew P, MINATTI, Ana E, TASSINI, Sabrina, ALLEN, Jennifer R, TONELLI, Federica, MA, Vu Van, LATTANZI, Giulia, WALTON, Mary, GOODMAN, Clifford, LINGARD, Iain, CHEN, Ning, LIU, Qingyian, LOW, Jonathan D
Year of Publication 03.06.2021
Get full text
Year of Publication 03.06.2021
Patent
Heterocyclic compounds as Delta-5 Desaturase inhibitors and methods of use
TONELLI, FEDERICA, MINATTI, ANA ELENA, CHEN, NING, LIU, QINGYIAN, LOW, JONATHAN D, ALLEN, JENNIFER REBECCA, MA, VU VAN, POZZAN, ALFONSO, WALTON, MARY, GOODMAN, CLIFFORD, LINGARD, IAIN, LATTANZI, GIULIA, SIEGMUND, AARON C, BOURBEAU, MATTHEW PAUL, AMEGADZIE, ALBERT, REEVES, COREY, TASSINI, SABRINA
Year of Publication 01.09.2021
Get full text
Year of Publication 01.09.2021
Patent