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Published in Proceedings of the National Academy of Sciences - PNAS (20.12.2005)
Published in Proceedings of the National Academy of Sciences - PNAS (20.12.2005)
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An endocannabinoid mechanism for stress-induced analgesia
Piomelli, Daniele, Tarzia, Giorgio, Hohmann, Andrea G, Mangieri, Regina, Duranti, Andrea, Tontini, Andrea, Krey, Jocelyn F, Neely, Mark H, Crystal, Jonathon D, Suplita, Richard L, Mor, Marco, Bolton, Nathan M, Fegley, Darren, Holmes, Philip V, Michael Walker, J
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Published in Nature (23.06.2005)
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2-N-Acylaminoalkylindoles: Design and Quantitative Structure−Activity Relationship Studies Leading to MT2-Selective Melatonin Antagonists
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Published in Journal of medicinal chemistry (30.08.2001)
Published in Journal of medicinal chemistry (30.08.2001)
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Mimosine induces apoptosis in the HL60 human tumor cell line
Renò, F, Tontini, A, Burattini, S, Papa, S, Falcieri, E, Tarzia, G
Published in Apoptosis (London) (01.12.1999)
Published in Apoptosis (London) (01.12.1999)
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Oleylethanolamide regulates feeding and body weight through activation of the nuclear receptor PPAR-α
Piomelli, Daniele, Fu, Jin, Gaetani, Silvana, Oveisi, Fariba, Lo Verme, Jesse, Serrano, Antonia, Rodríguez de Fonseca, Fernando, Rosengarth, Anja, Luecke, Hartmut, Di Giacomo, Barbara, Tarzia, Giorgio
Published in Nature (04.09.2003)
Published in Nature (04.09.2003)
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Characterization of the fatty acid amide hydrolase inhibitor cyclohexyl carbamic acid 3'-carbamoyl-biphenyl-3-yl ester (URB597): effects on anandamide and oleoylethanolamide deactivation
Fegley, Darren, Gaetani, Silvana, Duranti, Andrea, Tontini, Andrea, Mor, Marco, Tarzia, Giorgio, Piomelli, Daniele
Published in The Journal of pharmacology and experimental therapeutics (01.04.2005)
Published in The Journal of pharmacology and experimental therapeutics (01.04.2005)
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5-(2-Ethyl-phenyl)-3-(3-methoxy-phenyl)-1H-[1,2,4]triazole (DL-111-IT) and related compounds induce apoptotic patterns in cultures of human tumor cell lines
Burattini, S, Luchetti, F, Battistelli, M, Della Felice, M, Papa, S, Piersanti, G, Tarzia, G, Falcieri, E
Published in Journal of biological regulators and homeostatic agents (01.10.2003)
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Published in Journal of biological regulators and homeostatic agents (01.10.2003)
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Modulation of anxiety through blockade of anandamide hydrolysis
Piomelli, Daniele, Kathuria, Satish, Gaetani, Silvana, Fegley, Darren, Valiño, Fernando, Duranti, Andrea, Tontini, Andrea, Mor, Marco, Tarzia, Giorgio, Rana, Giovanna La, Calignano, Antonio, Giustino, Arcangela, Tattoli, Maria, Palmery, Maura, Cuomo, Vincenzo
Published in Nature medicine (01.01.2003)
Published in Nature medicine (01.01.2003)
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Cyclohexylcarbamic Acid 3‘- or 4‘-Substituted Biphenyl-3-yl Esters as Fatty Acid Amide Hydrolase Inhibitors: Synthesis, Quantitative Structure−Activity Relationships, and Molecular Modeling Studies
Mor, Marco, Rivara, Silvia, Lodola, Alessio, Plazzi, Pier Vincenzo, Tarzia, Giorgio, Duranti, Andrea, Tontini, Andrea, Piersanti, Giovanni, Kathuria, Satish, Piomelli, Daniele
Published in Journal of medicinal chemistry (07.10.2004)
Published in Journal of medicinal chemistry (07.10.2004)
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Synthesis and biological evaluation of pyrido[2,3-b]pyrazine and pyrido[2,3-b]pyrazine-n-oxide as selective glycine antagonists
Cugola, Alfredo, Donati, Daniele, Guarneri, M., Micheli, Fabrizio, Missio, Andrea, Pecunioso, Angelo, Reggiani, Angelo, Tarzia, G., Zanirato, V.
Published in Bioorganic & medicinal chemistry letters (19.11.1996)
Published in Bioorganic & medicinal chemistry letters (19.11.1996)
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Selective inhibition of 2-AG hydrolysis enhances endocannabinoid signaling in hippocampus
Freund, Tamás F, Piomelli, Daniele, Makara, Judit K, Mor, Marco, Fegley, Darren, Szabó, Szilárd I, Kathuria, Satish, Astarita, Giuseppe, Duranti, Andrea, Tontini, Andrea, Tarzia, Giorgio, Rivara, Silvia
Published in Nature neuroscience (01.09.2005)
Published in Nature neuroscience (01.09.2005)
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AN IMPROVED ROUTE TO CYCLOALKA[b]PYRROLE 2-CARBOXYLATES
Balsamini, C., Bedini, A., Tarzia, G., Tontini, A.
Published in Organic preparations and procedures international (01.08.1997)
Published in Organic preparations and procedures international (01.08.1997)
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Synthesis and biological evaluation of 6-bromo-6-substituted penicillanic acid derivatives as β-lactamase inhibitors
Bedini, A, Balsamini, C, Di Giacomo, B, Tontini, A, Citterio, B, Giorgi, L, Di Modugno, E, Tarzia, G
Published in Farmaco (Società chimica italiana : 1989) (01.08.2002)
Published in Farmaco (Società chimica italiana : 1989) (01.08.2002)
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Rapid and transient stimulation of intracellular reactive oxygen species by melatonin in normal and tumor leukocytes
Radogna, Flavia, Paternoster, Laura, De Nicola, Milena, Cerella, Claudia, Ammendola, Sergio, Bedini, Annalida, Tarzia, Giorgio, Aquilano, Katia, Ciriolo, Maria, Ghibelli, Lina
Published in Toxicology and applied pharmacology (15.08.2009)
Published in Toxicology and applied pharmacology (15.08.2009)
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2-n-Butyl-9-methyl-8-[1,2,3]triazol-2-yl-9H-purin-6-ylamine and analogues as A(2A) adenosine receptor antagonists. Design, synthesis, and pharmacological characterization
Minetti, P, Tinti, MO, Carminati, P, Castorina, M, Di Cesare, MA, Di Serio, S, Gallo, G, Ghirardi, O, Giorgi, F, Giorgi, L, Piersanti, G, Bartoccini, F, Tarzia, G
Published in Journal of medicinal chemistry (03.11.2005)
Published in Journal of medicinal chemistry (03.11.2005)
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Design, Synthesis, and Structure−Activity Relationships of Alkylcarbamic Acid Aryl Esters, a New Class of Fatty Acid Amide Hydrolase Inhibitors
Tarzia, Giorgio, Duranti, Andrea, Tontini, Andrea, Piersanti, Giovanni, Mor, Marco, Rivara, Silvia, Plazzi, Pier Vincenzo, Park, Chris, Kathuria, Satish, Piomelli, Daniele
Published in Journal of medicinal chemistry (05.06.2003)
Published in Journal of medicinal chemistry (05.06.2003)
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Synthesis of new C-6 alkyliden penicillin derivatives as β-lactamase inhibitors
Di Giacomo, B, Tarzia, G, Bedini, A, Gatti, G, Bartoccini, F, Balsamini, C, Tontini, A, Baffone, W, Di Modugno, E, Felici, A
Published in Farmaco (Società chimica italiana : 1989) (01.04.2002)
Published in Farmaco (Società chimica italiana : 1989) (01.04.2002)
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Synthesis of Novel 6-α and 6-β-Alkylcarbonylmethyl Substituted Penems
PENTASSUGLIA, G., TARZIA, G., ANDREOTTI, D., BISMARA, C., CARLESSO, R., DONATI, D., GAVIRAGHI, G., PERBONI, A., PEZZOLI, A., ROSSI, T., TAMBURINI, B., URSINI, A.
Published in Journal of antibiotics (1995)
Published in Journal of antibiotics (1995)
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QM/MM modelling of oleamide hydrolysis in fatty acid amide hydrolase (FAAH) reveals a new mechanism of nucleophile activation
Lodola, Alessio, Mor, Marco, Hermann, Johannes C, Tarzia, Giorgio, Piomelli, Daniele, Mulholland, Adrian J
Published in Chemical communications (Cambridge, England) (21.09.2005)
Published in Chemical communications (Cambridge, England) (21.09.2005)
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