Grapevine Botryosphaeria dieback fungi have specific aggressiveness factor repertory involved in wood decay and stilbene metabolization
Stempien, Elodie, Goddard, Mary-Lorène, Wilhelm, Kim, Tarnus, Céline, Bertsch, Christophe, Chong, Julie
Published in PloS one (20.12.2017)
Published in PloS one (20.12.2017)
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Journal Article
Selective inhibition of PfA-M1, over PfA-M17, by an amino-benzosuberone derivative blocks malaria parasites development in vitro and in vivo
Bounaadja, Lotfi, Schmitt, Marjorie, Albrecht, Sébastien, Mouray, Elisabeth, Tarnus, Céline, Florent, Isabelle
Published in Malaria journal (21.09.2017)
Published in Malaria journal (21.09.2017)
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Journal Article
Iminosugar-Cyclopeptoid Conjugates Raise Multivalent Effect in Glycosidase Inhibition at Unprecedented High Levels
Lepage, Mathieu L., Schneider, Jérémy P., Bodlenner, Anne, Meli, Alessandra, De Riccardis, Francesco, Schmitt, Marjorie, Tarnus, Céline, Nguyen-Huynh, Nha-Thi, Francois, Yannis-Nicolas, Leize-Wagner, Emmanuelle, Birck, Catherine, Cousido-Siah, Alexandra, Podjarny, Alberto, Izzo, Irene, Compain, Philippe
Published in Chemistry : a European journal (04.04.2016)
Published in Chemistry : a European journal (04.04.2016)
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Journal Article
Aminobenzosuberone Scaffold as a Modular Chemical Tool for the Inhibition of Therapeutically Relevant M1 Aminopeptidases
Salomon, Emmanuel, Schmitt, Marjorie, Marapaka, Anil Kumar, Stamogiannos, Athanasios, Revelant, Germain, Schmitt, Céline, Alavi, Sarah, Florent, Isabelle, Addlagatta, Anthony, Stratikos, Efstratios, Tarnus, Céline, Albrecht, Sébastien
Published in Molecules (Basel, Switzerland) (11.10.2018)
Published in Molecules (Basel, Switzerland) (11.10.2018)
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Journal Article
Synthesis and Glycosidase Inhibition Properties of Calix[8]arene-Based Iminosugar Click Clusters
Schneider, Jérémy P., Tommasone, Stefano, Della Sala, Paolo, Gaeta, Carmine, Talotta, Carmen, Tarnus, Céline, Neri, Placido, Bodlenner, Anne, Compain, Philippe
Published in Pharmaceuticals (Basel, Switzerland) (01.11.2020)
Published in Pharmaceuticals (Basel, Switzerland) (01.11.2020)
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Journal Article
Wood Metabolomic Responses of Wild and Cultivated Grapevine to Infection with Neofusicoccum parvum, a Trunk Disease Pathogen
Labois, Clément, Wilhelm, Kim, Laloue, Hélène, Tarnus, Céline, Bertsch, Christophe, Goddard, Mary-Lorène, Chong, Julie
Published in Metabolites (04.06.2020)
Published in Metabolites (04.06.2020)
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Journal Article
A Convergent Strategy for the Synthesis of Second-Generation Iminosugar Clusters Using "Clickable" Trivalent Dendrons
Joosten, Antoine, Schneider, Jérémy P., Lepage, Mathieu L., Tarnus, Céline, Bodlenner, Anne, Compain, Philippe
Published in European journal of organic chemistry (01.03.2014)
Published in European journal of organic chemistry (01.03.2014)
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Journal Article
Aminobenzosuberone derivatives as PfA-M1 inhibitors: Molecular recognition and antiplasmodial evaluation
Salomon, Emmanuel, Schmitt, Marjorie, Mouray, Elisabeth, McEwen, Alastair G., Bounaadja, Lotfi, Torchy, Morgan, Poussin-Courmontagne, Pierre, Alavi, Sarah, Tarnus, Céline, Cavarelli, Jean, Florent, Isabelle, Albrecht, Sébastien
Published in Bioorganic chemistry (01.05.2020)
Published in Bioorganic chemistry (01.05.2020)
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Journal Article
Rapid and efficient synthesis of a novel series of substituted aminobenzosuberone derivatives as potent, selective, non-peptidic neutral aminopeptidase inhibitors
Albrecht, Sébastien, Salomon, Emmanuel, Defoin, Albert, Tarnus, Céline
Published in Bioorganic & medicinal chemistry (15.08.2012)
Published in Bioorganic & medicinal chemistry (15.08.2012)
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Journal Article
Synthesis of the first examples of iminosugar clusters based on cyclopeptoid cores
Lepage, Mathieu L, Meli, Alessandra, Bodlenner, Anne, Tarnus, Céline, De Riccardis, Francesco, Izzo, Irene, Compain, Philippe
Published in Beilstein journal of organic chemistry (23.06.2014)
Published in Beilstein journal of organic chemistry (23.06.2014)
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Journal Article
Selective aminopeptidase-N (CD13) inhibitors with relevance to cancer chemotherapy
Schmitt, Céline, Voegelin, Manon, Marin, Aurélie, Schmitt, Marjorie, Schegg, Fabienne, Hénon, Philippe, Guenot, Dominique, Tarnus, Céline
Published in Bioorganic & medicinal chemistry (01.04.2013)
Published in Bioorganic & medicinal chemistry (01.04.2013)
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Journal Article
Synthesis of 4-amino-4,5-dideoxy- l-lyxofuranose derivatives and their evaluation as fucosidase inhibitors
Chevrier, Carine, Le Nouën, Didier, Defoin, Albert, Tarnus, Céline
Published in Carbohydrate research (15.07.2011)
Published in Carbohydrate research (15.07.2011)
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Journal Article
Exploring S1 plasticity and probing S1′ subsite of mammalian aminopeptidase N/CD13 with highly potent and selective aminobenzosuberone inhibitors
Revelant, Germain, Al-Lakkis-Wehbe, Mira, Schmitt, Marjorie, Alavi, Sarah, Schmitt, Céline, Roux, Lionel, Al-Masri, Mounir, Schifano-Faux, Nadège, Maiereanu, Carmen, Tarnus, Céline, Albrecht, Sébastien
Published in Bioorganic & medicinal chemistry (01.07.2015)
Published in Bioorganic & medicinal chemistry (01.07.2015)
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Journal Article
Synthesis of amino-hydroxy-benzocycloheptenones as potent, selective, non-peptidic dinuclear zinc metalloaminopeptidase inhibitors
Al-Lakkis-Wehbe, Mira, Chaillou, Bérénice, Defoin, Albert, Albrecht, Sébastien, Tarnus, Céline
Published in Bioorganic & medicinal chemistry (01.11.2013)
Published in Bioorganic & medicinal chemistry (01.11.2013)
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Journal Article
An innovative strategy for the synthesis of a new series of potent aminopeptidase (APN or CD13) inhibitors derived from the oxepin-4-one family
Roux, Lionel, Charrier, Cédric, Salomon, Emmanuel, Ilhan, Meral, Bisseret, Philippe, Tarnus, Céline
Published in Tetrahedron letters (18.05.2011)
Published in Tetrahedron letters (18.05.2011)
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Journal Article
Amino-benzosuberone: A novel warhead for selective inhibition of human aminopeptidase-N/CD13
Albrecht, Sébastien, Al-Lakkis-Wehbe, Mira, Orsini, Alban, Defoin, Albert, Pale, Patrick, Salomon, Emmanuel, Tarnus, Céline, Weibel, Jean-Marc
Published in Bioorganic & medicinal chemistry (15.02.2011)
Published in Bioorganic & medicinal chemistry (15.02.2011)
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Journal Article