WaterMap‐Guided Structure‐Based Virtual Screening for Acetylcholinesterase Inhibitors
Targowska‐Duda, Katarzyna M., Maj, Maciej, Drączkowski, Piotr, Budzyńska, Barbara, Boguszewska‐Czubara, Anna, Wróbel, Tomasz M., Laitinen, Tuomo, Kaczmar, Patrycja, Poso, Antti, Kaczor, Agnieszka A.
Published in ChemMedChem (20.04.2022)
Published in ChemMedChem (20.04.2022)
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Multitarget Derivatives of D2AAK1 as Potential Antipsychotics: The Effect of Substitution in the Indole Moiety
Kondej, Magda, Wróbel, Tomasz M., Targowska‐Duda, Katarzyna M., Leandro Martínez, Antón, Koszła, Oliwia, Stępnicki, Piotr, Zięba, Agata, Paz, Alba, Wronikowska‐Denysiuk, Olga, Loza, Maria I., Castro, Marián, Kaczor, Agnieszka A.
Published in ChemMedChem (03.08.2022)
Published in ChemMedChem (03.08.2022)
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6-Gingerol, a Major Constituent of Zingiber officinale Rhizoma, Exerts Anticonvulsant Activity in the Pentylenetetrazole-Induced Seizure Model in Larval Zebrafish
Gawel, Kinga, Kukula-Koch, Wirginia, Banono, Nancy Saana, Nieoczym, Dorota, Targowska-Duda, Katarzyna M, Czernicka, Lidia, Parada-Turska, Jolanta, Esguerra, Camila V
Published in International journal of molecular sciences (20.07.2021)
Published in International journal of molecular sciences (20.07.2021)
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Efficacy of Dabrafenib and Trametinib in a Patient with Squamous-Cell Carcinoma, with Mutation p.D594G in BRAF and p.R461 in NF1 Genes-A Case Report with Literature Review
Grenda, Anna, Krawczyk, Pawel, Targowska-Duda, Katarzyna M, Kieszko, Robert, Paśnik, Iwona, Milanowski, Janusz
Published in International journal of molecular sciences (07.01.2023)
Published in International journal of molecular sciences (07.01.2023)
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Angiotensin II Type 1 Receptor Blockers Inhibit KAT II Activity in the Brain—Its Possible Clinical Applications
Zakrocka, Izabela, Targowska-Duda, Katarzyna M., Wnorowski, Artur, Kocki, Tomasz, Jóźwiak, Krzysztof, Turski, Waldemar A.
Published in Neurotoxicity research (01.11.2017)
Published in Neurotoxicity research (01.11.2017)
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Funnel metadynamics and behavioral studies reveal complex effect of D2AAK1 ligand on anxiety-like processes
Bartuzi, Damian, Kędzierska, Ewa, Targowska-Duda, Katarzyna M., Koszła, Oliwia, Wróbel, Tomasz M., Jademyr, Simon, Karcz, Tadeusz, Szczepańska, Katarzyna, Stępnicki, Piotr, Wronikowska-Denysiuk, Olga, Biała, Grażyna, Handzlik, Jadwiga, Kristensen, Jesper L., Poso, Antti, Kaczor, Agnieszka A.
Published in Scientific reports (07.12.2022)
Published in Scientific reports (07.12.2022)
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Novel multi-target ligands of dopamine and serotonin receptors for the treatment of schizophrenia based on indazole and piperazine scaffolds-synthesis, biological activity, and structural evaluation
Stępnicki, Piotr, Wronikowska-Denysiuk, Olga, Zięba, Agata, Targowska-Duda, Katarzyna M., Bartyzel, Agata, Wróbel, Martyna Z., Wróbel, Tomasz M., Szałaj, Klaudia, Chodkowski, Andrzej, Mirecka, Karolina, Budzyńska, Barbara, Fornal, Emilia, Turło, Jadwiga, Castro, Marián, Kaczor, Agnieszka A.
Published in Journal of enzyme inhibition and medicinal chemistry (01.12.2023)
Published in Journal of enzyme inhibition and medicinal chemistry (01.12.2023)
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3-Furan-2-yl-N-p-tolyl-acrylamide, a highly selective positive allosteric modulator of α7 nicotinic receptors, produces anxiolytic-like activity in mice
Targowska-Duda, Katarzyna M, Budzynska, Barbara, Michalak, Agnieszka, Jozwiak, Krzysztof, Biala, Grazyna, Arias, Hugo R
Published in Journal of psychopharmacology (Oxford) (01.05.2019)
Published in Journal of psychopharmacology (Oxford) (01.05.2019)
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N -(2-Hydroxyphenyl)-1-[3-(2-oxo-2,3-dihydro-1 H - benzimidazol-1-yl)propyl]piperidine-4-Carboxamide (D2AAK4), a Multi-Target Ligand of Aminergic GPCRs, as a Potential Antipsychotic
Kaczor, Agnieszka A, Targowska-Duda, Katarzyna M, Silva, Andrea G, Kondej, Magda, Biała, Grażyna, Castro, Marián
Published in Biomolecules (Basel, Switzerland) (24.02.2020)
Published in Biomolecules (Basel, Switzerland) (24.02.2020)
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Preclinical effects of cannabidiol in an experimental model of migraine
Sturaro, Chiara, Fakhoury, Bianca, Targowska-Duda, Katarzyna M, Zribi, Gilles, Schoch, Jennifer, Ruzza, Chiara, Calò, Girolamo, Toll, Lawrence, Cippitelli, Andrea
Published in Pain (Amsterdam) (01.11.2023)
Published in Pain (Amsterdam) (01.11.2023)
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Loop diuretics inhibit kynurenic acid production and kynurenine aminotransferases activity in rat kidneys
Zakrocka, Izabela, Targowska-Duda, Katarzyna M, Kocki, Tomasz, Turski, Waldemar, Urbańska, Ewa M, Załuska, Wojciech
Published in Pharmacological reports (11.09.2024)
Published in Pharmacological reports (11.09.2024)
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NOP receptor agonist attenuates nitroglycerin-induced migraine-like symptoms in mice
Targowska-Duda, Katarzyna M., Ozawa, Akihiko, Bertels, Zachariah, Cippitelli, Andrea, Marcus, Jason L., Mielke-Maday, Hanna K., Zribi, Gilles, Rainey, Amanda N., Kieffer, Brigitte L., Pradhan, Amynah A., Toll, Lawrence
Published in Neuropharmacology (15.06.2020)
Published in Neuropharmacology (15.06.2020)
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N-(3-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}propyl)-1H-indazole-3-carboxamide (D2AAK3) as a potential antipsychotic: In vitro, in silico and in vivo evaluation of a multi-target ligand
Kaczor, Agnieszka A., Targowska-Duda, Katarzyna M., Stępnicki, Piotr, Silva, Andrea G., Koszła, Oliwia, Kędzierska, Ewa, Grudzińska, Angelika, Kruk-Słomka, Marta, Biała, Grażyna, Castro, Marián
Published in Neurochemistry international (01.06.2021)
Published in Neurochemistry international (01.06.2021)
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Coronaridine congeners inhibit human α3β4 nicotinic acetylcholine receptors by interacting with luminal and non-luminal sites
Arias, Hugo R., Targowska-Duda, Katarzyna M., Feuerbach, Dominik, Jozwiak, Krzysztof
Published in The international journal of biochemistry & cell biology (01.08.2015)
Published in The international journal of biochemistry & cell biology (01.08.2015)
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Type I and type II positive allosteric modulators of α7 nicotinic acetylcholine receptors induce antidepressant-like activity in mice by a mechanism involving receptor potentiation but not neurotransmitter reuptake inhibition. Correlation with mTOR intracellular pathway activation
Targowska-Duda, Katarzyna M., Budzynska, Barbara, Michalak, Agnieszka, Wnorowski, Artur, Loland, Claus J., Maj, Maciej, Manetti, Dina, Romanelli, Maria Novella, Jozwiak, Krzysztof, Biala, Grazyna, Arias, Hugo R.
Published in European neuropsychopharmacology (01.11.2021)
Published in European neuropsychopharmacology (01.11.2021)
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Angiotensin II type 1 receptor blockers decrease kynurenic acid production in rat kidney in vitro
Zakrocka, Izabela, Targowska-Duda, Katarzyna M., Wnorowski, Artur, Kocki, Tomasz, Jóźwiak, Krzysztof, Turski, Waldemar A.
Published in Naunyn-Schmiedeberg's archives of pharmacology (01.02.2019)
Published in Naunyn-Schmiedeberg's archives of pharmacology (01.02.2019)
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