Targeting Cavity-Creating p53 Cancer Mutations with Small-Molecule Stabilizers: the Y220X Paradigm
Bauer, Matthias R, Krämer, Andreas, Settanni, Giovanni, Jones, Rhiannon N, Ni, Xiaomin, Khan Tareque, Raysa, Fersht, Alan R, Spencer, John, Joerger, Andreas C
Published in ACS chemical biology (20.03.2020)
Published in ACS chemical biology (20.03.2020)
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Solvent‐Free Synthesis of Core‐Functionalised Naphthalene Diimides by Using a Vibratory Ball Mill: Suzuki, Sonogashira and Buchwald–Hartwig Reactions
Panther, Lydia A., Guest, Daniel P., McGown, Andrew, Emerit, Hugo, Tareque, Raysa Khan, Jose, Arathy, Dadswell, Chris M., Coles, Simon J., Tizzard, Graham J., González‐Méndez, Ramón, Goodall, Charles A. I., Bagley, Mark C., Spencer, John, Greenland, Barnaby W.
Published in Chemistry : a European journal (01.09.2022)
Published in Chemistry : a European journal (01.09.2022)
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Journal Article
Genotoxicity and Epigenotoxicity of Carbazole-Derived Molecules on MCF-7 Breast Cancer Cells
Luparello, Claudio, Cruciata, Ilenia, Joerger, Andreas C, Ocasio, Cory A, Jones, Rhiannon, Tareque, Raysa Khan, Bagley, Mark C, Spencer, John, Walker, Martin, Austin, Carol, Ferrara, Tiziana, D Oca, Pietro, Bellina, Rossella, Branni, Rossella, Caradonna, Fabio
Published in International journal of molecular sciences (26.03.2021)
Published in International journal of molecular sciences (26.03.2021)
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Deliberately Losing Control of C−H Activation Processes in the Design of Small‐Molecule‐Fragment Arrays Targeting Peroxisomal Metabolism
Khan Tareque, Raysa, Hassell‐Hart, Storm, Krojer, Tobias, Bradley, Anthony, Velupillai, Srikannathasan, Talon, Romain, Fairhead, Michael, Day, Iain J., Bala, Kamlesh, Felix, Robert, Kemmitt, Paul D., Brennan, Paul, Delft, Frank, Díaz Sáez, Laura, Huber, Kilian, Spencer, John
Published in ChemMedChem (15.12.2020)
Published in ChemMedChem (15.12.2020)
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Synthesis and biological evaluation of benzodiazepines containing a pentafluorosulfanyl group
Jose, Arathy, Tareque, Raysa Khan, Mortensen, Martin, Legay, Remi, Coles, Simon J., Tizzard, Graham J., Greenland, Barnaby W., Smart, Trevor G., Bagley, Mark C., Spencer, John
Published in Tetrahedron (09.04.2021)
Published in Tetrahedron (09.04.2021)
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