Synthesis and Biological Evaluation of 1-Methyl-1H-indole-Pyrazoline Hybrids as Potential Tubulin Polymerization Inhibitors
Zhang, Ya-Liang, Qin, Ya-Juan, Tang, Dan-Jie, Yang, Meng-Ru, Li, Bo-Yan, Wang, Yan-Ting, Cai, Hong-Yu, Wang, Bao-Zhong, Zhu, Hai-Liang
Published in ChemMedChem (05.07.2016)
Published in ChemMedChem (05.07.2016)
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Metronidazole containing pyrazole derivatives potently inhibit tyrosyl-tRNA synthetase: design, synthesis, and biological evaluation
Chen, Long-Wang, Wang, Peng-Fei, Tang, Dan-Jie, Tao, Xiang-Xiang, Man, Ruo-Jun, Qiu, Han-Yue, Wang, Zhong-Chang, Xu, Chen, Zhu, Hai-Liang
Published in Chemical biology & drug design (01.10.2016)
Published in Chemical biology & drug design (01.10.2016)
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Synthesis and biological evaluation of novel indole derivatives containing sulfonamide scaffold as potential tubulin inhibitor
Man, Ruo-Jun, Tang, Dan-Jie, Lu, Xiao-Yuan, Duan, Yong-Tao, Tao, Xiang-Xiang, Yang, Meng-Ru, Wang, Le-Le, Wang, Bao-Zhong, Xu, Chen, Zhu, Hai-Liang
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Published in MedChemComm (01.01.2016)
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Design, synthesis and biological evaluation of pyrazolyl-nitroimidazole derivatives as potential EGFR/HER-2 kinase inhibitors
Tao, Xiang-Xiang, Duan, Yong-Tao, Chen, Long-Wang, Tang, Dan-Jie, Yang, Meng-Ru, Wang, Peng-Fei, Xu, Chen, Zhu, Hai-Liang
Published in Bioorganic & medicinal chemistry letters (15.01.2016)
Published in Bioorganic & medicinal chemistry letters (15.01.2016)
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Design, Synthesis and Antitumor Activity of Novel link-bridge and B-Ring Modified Combretastatin A-4 (CA-4) Analogues as Potent Antitubulin Agents
Duan, Yong-Tao, Man, Ruo-Jun, Tang, Dan-Jie, Yao, Yong-Fang, Tao, Xiang-Xiang, Yu, Chen, Liang, Xin-Yi, Makawana, Jigar A, Zou, Mei-Juan, Wang, Zhong-Chang, Zhu, Hai-Liang
Published in Scientific reports (03.05.2016)
Published in Scientific reports (03.05.2016)
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Discovery and molecular modeling of novel 1-indolyl acetate – 5-Nitroimidazole targeting tubulin polymerization as antiproliferative agents
Duan, Yong-Tao, Sang, Ya-Li, Makawana, Jigar A., Teraiya, Shashikant B., Yao, Yong-Fang, Tang, Dan-Jie, Tao, Xiang-Xiang, Zhu, Hai-Liang
Published in European journal of medicinal chemistry (06.10.2014)
Published in European journal of medicinal chemistry (06.10.2014)
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Synthesis, biological evaluation, and molecular docking studies of novel 2-styryl-5-nitroimidazole derivatives containing 1,4-benzodioxan moiety as FAK inhibitors with anticancer activity
Duan, Yong-Tao, Yao, Yong-Fang, Huang, Wei, Makawana, Jigar A., Teraiya, Shashikant B., Thumar, Nilesh j., Tang, Dan-Jie, Tao, Xiang-Xiang, Wang, Zhong-Chang, Jiang, Ai-Qin, Zhu, Hai-Liang
Published in Bioorganic & medicinal chemistry (01.06.2014)
Published in Bioorganic & medicinal chemistry (01.06.2014)
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Synthesis and biological evaluation of quinoline–imidazole hybrids as potent telomerase inhibitors: a promising class of antitumor agents
Duan, Yong-Tao, Yao, Yong-Fang, Tang, Dan-Jie, Thumar, Nilesh j., Teraiya, Shashikant B., Makawana, Jigar A., Sang, Ya-Li, Wang, Zhong-Chang, Tao, Xiang-Xiang, Jiang, Ai-Qin, Zhu, Hai-Liang
Published in RSC advances (2014)
Published in RSC advances (2014)
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Modification, Biological Evaluation and 3D QSAR Studies of Novel 2
Yang, Yu-Shun, Zhang, Fei, Tang, Dan-Jie, Yang, Yong-Hua, Zhu, Hai-Liang
Published in PloS one (14.05.2014)
Published in PloS one (14.05.2014)
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Journal Article
Synthesis and Biological Evaluation of 1‐Methyl‐1 H ‐indole–Pyrazoline Hybrids as Potential Tubulin Polymerization Inhibitors
Zhang, Ya‐Liang, Qin, Ya‐Juan, Tang, Dan‐Jie, Yang, Meng‐Ru, Li, Bo‐Yan, Wang, Yan‐Ting, Cai, Hong‐Yu, Wang, Bao‐Zhong, Zhu, Hai‐Liang
Published in ChemMedChem (05.07.2016)
Published in ChemMedChem (05.07.2016)
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Journal Article
Synthesis and biological evaluation of novel indole derivatives containing sulfonamide scaffold as potential tubulin inhibitorThe authors declare no competing interests.Electronic supplementary information (ESI) available. CCDC 1412186. For ESI and crystallographic data in CIF or other electronic format see DOI: 10.1039/c6md00255b
Man, Ruo-Jun, Tang, Dan-Jie, Lu, Xiao-Yuan, Duan, Yong-Tao, Tao, Xiang-Xiang, Yang, Meng-Ru, Wang, Le-Le, Wang, Bao-Zhong, Xu, Chen, Zhu, Hai-Liang
Year of Publication 14.09.2016
Year of Publication 14.09.2016
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