Discovery of MK-8719, a Potent O‑GlcNAcase Inhibitor as a Potential Treatment for Tauopathies
Selnick, Harold G, Hess, J. Fred, Tang, Cuyue, Liu, Kun, Schachter, Joel B, Ballard, Jeanine E, Marcus, Jacob, Klein, Daniel J, Wang, Xiaohai, Pearson, Michelle, Savage, Mary J, Kaul, Ramesh, Li, Tong-Shuang, Vocadlo, David J, Zhou, Yuanxi, Zhu, Yongbao, Mu, Changwei, Wang, Yaode, Wei, Zhongyong, Bai, Chang, Duffy, Joseph L, McEachern, Ernest J
Published in Journal of medicinal chemistry (27.11.2019)
Published in Journal of medicinal chemistry (27.11.2019)
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Journal Article
Effects of Fibrates on Metabolism of Statins in Human Hepatocytes
PRUEKSARITANONT, Thomayant, CUYUE TANG, YUE QIU, MU, Lillian, SUBRAMANIAN, Raju, LIN, Jiunn H
Published in Drug metabolism and disposition (01.11.2002)
Published in Drug metabolism and disposition (01.11.2002)
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Journal Article
Mechanistic Studies on Metabolic Interactions between Gemfibrozil and Statins
Prueksaritanont, Thomayant, Zhao, Jamie J, Ma, Bennett, Roadcap, Brad A, Tang, Cuyue, Qiu, Yue, Liu, Lida, Lin, Jiunn H, Pearson, Paul G, Baillie, Thomas A
Published in The Journal of pharmacology and experimental therapeutics (01.06.2002)
Published in The Journal of pharmacology and experimental therapeutics (01.06.2002)
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Journal Article
Discovery of 2,5-diarylnicotinamides as selective orexin-2 receptor antagonists (2-SORAs)
Mercer, Swati P., Roecker, Anthony J., Garson, Susan, Reiss, Duane R., Meacham Harrell, C., Murphy, Kathy L., Bruno, Joseph G., Bednar, Rodney A., Lemaire, Wei, Cui, Donghui, Cabalu, Tamara D., Tang, Cuyue, Prueksaritanont, Thomayant, Hartman, George D., Young, Steven D., Winrow, Christopher J., Renger, John J., Coleman, Paul J.
Published in Bioorganic & medicinal chemistry letters (15.12.2013)
Published in Bioorganic & medicinal chemistry letters (15.12.2013)
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Journal Article
METABOLISM-BASED DRUG-DRUG INTERACTIONS: WHAT DETERMINES INDIVIDUAL VARIABILITY IN CYTOCHROME P450 INDUCTION?
Tang, Cuyue, Lin, Jiunn H, Lu, Anthony Y H
Published in Drug metabolism and disposition (01.05.2005)
Published in Drug metabolism and disposition (01.05.2005)
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Journal Article
3-Aryl-5-phenoxymethyl-1,3-oxazolidin-2-ones as positive allosteric modulators of mGluR2 for the treatment of schizophrenia: Hit-to-lead efforts
Brnardic, Edward J., Fraley, Mark E., Garbaccio, Robert M., Layton, Mark E., Sanders, John M., Culberson, Chris, Jacobson, Marlene A., Magliaro, Brian C., Hutson, Pete H., O’Brien, Julie A., Huszar, Sarah L., Uslaner, Jason M., Fillgrove, Kerry L., Tang, Cuyue, Kuo, Yuhsin, Sur, Sylvie M., Hartman, George D.
Published in Bioorganic & medicinal chemistry letters (15.05.2010)
Published in Bioorganic & medicinal chemistry letters (15.05.2010)
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Journal Article
Substrate Inhibition Kinetics for Cytochrome P450-Catalyzed Reactions
Lin, Y, Lu, P, Tang, C, Mei, Q, Sandig, G, Rodrigues, A D, Rushmore, T H, Shou, M
Published in Drug metabolism and disposition (01.04.2001)
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Published in Drug metabolism and disposition (01.04.2001)
Journal Article
Pyridyl amides as potent inhibitors of T-type calcium channels
Reger, Thomas S., Yang, Zhi-Qiang, Schlegel, Kelly-Ann S., Shu, Youheng, Mattern, Christa, Cube, Rowena, Rittle, Kenneth E., McGaughey, Georgia B., Hartman, George D., Tang, Cuyue, Ballard, Jeanine, Kuo, Yuhsin, Prueksaritanont, Thomayant, Nuss, Cindy E., Doran, Scott M., Fox, Steven V., Garson, Susan L., Li, Yuxing, Kraus, Richard L., Uebele, Victor N., Renger, John J., Barrow, James C.
Published in Bioorganic & medicinal chemistry letters (15.03.2011)
Published in Bioorganic & medicinal chemistry letters (15.03.2011)
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Journal Article
Major Role of Human Liver Microsomal Cytochrome P450 2C9 (CYP2C9) in the Oxidative Metabolism of Celecoxib, a Novel Cyclooxygenase-II Inhibitor
Tang, C, Shou, M, Mei, Q, Rushmore, T H, Rodrigues, A D
Published in The Journal of pharmacology and experimental therapeutics (01.05.2000)
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Published in The Journal of pharmacology and experimental therapeutics (01.05.2000)
Journal Article
Effect of P-glycoprotein-mediated efflux on cerebrospinal fluid concentrations in rhesus monkeys
Tang, Cuyue, Kuo, Yuhsin, Pudvah, Nicole T., Ellis, Joan D., Michener, Maria S., Egbertson, Melissa, Graham, Samuel L., Cook, Jacquelynn J., Hochman, Jerome H., Prueksaritanont, Thomayant
Published in Biochemical pharmacology (15.09.2009)
Published in Biochemical pharmacology (15.09.2009)
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Journal Article
Indazole derivatives as novel bradykinin B1 receptor antagonists
BODMER-NARKEVITCH, Vera, ANTHONY, Neville J, BOCK, Mark G, KUDUK, Scott D, COFRE, Victoria, JOLLY, Samson M, MURPHY, Kathy L, RANSOM, Richard W, REISS, Duane R, CUYUE TANG, PRUEKSARITANONT, Thomayant, PETTIBONE, Douglas J
Published in Bioorganic & medicinal chemistry letters (01.12.2010)
Published in Bioorganic & medicinal chemistry letters (01.12.2010)
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Journal Article
In Vitro and in Vivo CYP3A64 Induction and Inhibition Studies in Rhesus Monkeys: A Preclinical Approach for CYP3A-Mediated Drug Interaction Studies
PRUEKSARITANONT, Thomayant, KUO, Yuhsin, CUYUE TANG, CHUNZE LI, YUE QIU, BING LU, STRONG-BASALYGA, Kristie, RICHARDS, Karen, CARR, Brian, LIN, Jiunn H
Published in Drug metabolism and disposition (01.09.2006)
Published in Drug metabolism and disposition (01.09.2006)
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Journal Article
2-Aminobenzophenones as a Novel Class of Bradykinin B1 Receptor Antagonists
Su, Dai-Shi, Lim, John L, Tinney, Elizabeth, Wan, Bang-Lin, Murphy, Kathy L, Reiss, Duane R, Harrell, C. Meacham, O’Malley, Stacy S, Ransom, Rick W, Chang, Raymond S. L, Pettibone, Douglas J, Yu, Jian, Tang, Cuyue, Prueksaritanont, Thomayant, Freidinger, Roger M, Bock, Mark G, Anthony, Neville J
Published in Journal of medicinal chemistry (10.07.2008)
Published in Journal of medicinal chemistry (10.07.2008)
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Journal Article
Rifampin Induces the in Vitro Oxidative Metabolism, but Not the in Vivo Clearance of Diclofenac in Rhesus Monkeys
PRUEKSARITANONT, Thomayant, CHUNZE LI, CUYUE TANG, KUO, Yuhsin, STRONG-BASALYGA, Kristie, CARR, Brian
Published in Drug metabolism and disposition (01.11.2006)
Published in Drug metabolism and disposition (01.11.2006)
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Journal Article
A new class of bradykinin B1 receptor antagonists with high oral bioavailability and minimal PXR activity
FENG, Dong-Mei, DIPARDO, Robert M, PETTIBONE, Douglas J, BOCK, Mark G, KUDUK, Scott D, WAI, Jenny M, CHANG, Ronald K, DI MARCO, Christina N, MURPHY, Kathy L, RANSOM, Richard W, REISS, Duane R, CUYUE TANG, PRUEKSARITANONT, Thomayant
Published in Bioorganic & medicinal chemistry letters (15.01.2008)
Published in Bioorganic & medicinal chemistry letters (15.01.2008)
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