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Fraser, Bryan J., Beldar, Serap, Seitova, Almagul, Hutchinson, Ashley, Mannar, Dhiraj, Li, Yanjun, Kwon, Daniel, Tan, Ruiyan, Wilson, Ryan P., Leopold, Karoline, Subramaniam, Sriram, Halabelian, Levon, Arrowsmith, Cheryl H., Bénard, François
Published in Nature chemical biology (01.09.2022)
Published in Nature chemical biology (01.09.2022)
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68Ga-Labeled [Leu13ψThz14]Bombesin(7–14) Derivatives: Promising GRPR-Targeting PET Tracers with Low Pancreas Uptake
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Published in Molecules (Basel, Switzerland) (11.06.2022)
Published in Molecules (Basel, Switzerland) (11.06.2022)
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Journal Article
68Ga-Labeled [Thz14]Bombesin(7–14) Analogs: Promising GRPR-Targeting Agonist PET Tracers with Low Pancreas Uptake
Wang, Lei, Bratanovic, Ivica Jerolim, Zhang, Zhengxing, Kuo, Hsiou-Ting, Merkens, Helen, Zeisler, Jutta, Zhang, Chengcheng, Tan, Ruiyan, Bénard, François, Lin, Kuo-Shyan
Published in Molecules (Basel, Switzerland) (20.02.2023)
Published in Molecules (Basel, Switzerland) (20.02.2023)
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Targeting Refractory Mantle Cell Lymphoma for Imaging and Therapy Using C-X-C Chemokine Receptor Type 4 Radioligands
Kwon, Daniel, Takata, Katsuyoshi, Zhang, Zhengxing, Chong, Lauren, Fraser, Bryan, Zeisler, Jutta, Miyata-Takata, Tomoko, Merkens, Helen, Rousseau, Julie, Aoki, Tomohiro, Kuo, Hsiou-Ting, Tan, Ruiyan, Zhang, Chengcheng, Lau, Joseph, Villa, Diego, Uribe, Carlos F, Lin, Kuo-Shyan, Steidl, Christian, Benard, Francois
Published in Clinical cancer research (14.04.2022)
Published in Clinical cancer research (14.04.2022)
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Evaluation of lysine modifications in the PSMA-targeting pharmacophore using positron emission tomography imaging in a preclinical model of human prostate cancer
Zhang, Chengcheng, Zhang, Zhengxing, Merkens, Helen, Colpo, Nadine, Tan, Ruiyan, Lin, Kuo-Shyan, Benard, Francois
Published in Nuclear medicine and biology (01.11.2023)
Published in Nuclear medicine and biology (01.11.2023)
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Journal Article
Structure, activity and inhibition of human TMPRSS2, a protease implicated in SARS-CoV-2 activation
Fraser, Bryan J, Beldar, Serap, Seitova, Almagul, Hutchinson, Ashley, Mannar, Dhiraj, Li, Yanjun, Kwon, Daniel, Tan, Ruiyan, Wilson, Ryan P, Leopold, Karoline, Subramaniam, Sriram, Halabelian, Levon, Arrowsmith, Cheryl H, Benard, Francois
Published in bioRxiv (24.06.2021)
Published in bioRxiv (24.06.2021)
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Paper
Stabilization of 68Ga-labeled [Thz14]Bombesin(7–14) analogue for imaging gastrin-releasing peptide receptor expression with positron emission tomography
Wang, Lei, Kuo, Hsiou-Ting, Zhang, Zhengxing, Zhang, Chengcheng, Merkens, Helen, Colpo, Nadine, Wilson, Ryan, Zeisler, Jutta, Tan, Ruiyan, Benard, Francois, Lin, Kuo-Shyan
Published in Nuclear medicine and biology (01.11.2023)
Published in Nuclear medicine and biology (01.11.2023)
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Journal Article
Synthesis and evaluation of 68Ga-labeled [Leu13ψThz14] Bombesin(7-14) analogues for imaging gastrin-releasing peptide receptor expression with positron emission tomography
Wang, Lei, Zhang, Zhengxing, Merkens, Helen, Colpo, Nadine, Zeisler, Jutta, Zhang, Chengcheng, Roxin, Aron, Tan, Ruiyan, Benard, Francois, Lin, Kuo-Shyan
Published in Nuclear medicine and biology (01.05.2022)
Published in Nuclear medicine and biology (01.05.2022)
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Journal Article
P-311 - Synthesis and evaluation of 68Ga-labeled [Leu13ψThz14] Bombesin(7-14) analogues for imaging gastrin-releasing peptide receptor expression with positron emission tomography
Wang, Lei, Zhang, Zhengxing, Merkens, Helen, Colpo, Nadine, Zeisler, Jutta, Zhang, Chengcheng, Roxin, Aron, Tan, Ruiyan, Benard, Francois, Lin, Kuo-Shyan
Published in Nuclear medicine and biology (01.05.2022)
Published in Nuclear medicine and biology (01.05.2022)
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Journal Article
Ga-Labeled [Thz[sup.14]]Bombesin Analogs: Promising GRPR-Targeting Agonist PET Tracers with Low Pancreas Uptake
Wang, Lei, Bratanovic, Ivica Jerolim, Zhang, Zhengxing, Kuo, Hsiou-Ting, Merkens, Helen, Zeisler, Jutta, Zhang, Chengcheng, Tan, Ruiyan, Bénard, François, Lin, Kuo-Shyan
Published in Molecules (Basel, Switzerland) (01.02.2023)
Published in Molecules (Basel, Switzerland) (01.02.2023)
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Journal Article
What a difference a methylene makes: replacing Glu with Asp or Aad in the Lys-urea-Glu pharmacophore of PSMA-targeting radioligands to reduce kidney and salivary gland uptake
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Published in Theranostics (01.01.2022)
Published in Theranostics (01.01.2022)
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Lys-urea-Aad, Lys-urea-Cmc and Lys-urea-Cms as potential pharmacophores for the design of PSMA-targeted radioligands to reduce off-target uptake in kidneys and salivary glands
Kuo, Hsiou-Ting, Zhang, Zhengxing, Zhang, Chengcheng, Merkens, Helen, Tan, Ruiyan, Wong, Antonio A. W. L., Uribe, Carlos F., Bénard, François, Lin, Kuo-Shyan
Published in Theranostics (01.01.2023)
Published in Theranostics (01.01.2023)
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Journal Article
68 Ga-Labeled [Thz 14 ]Bombesin(7-14) Analogs: Promising GRPR-Targeting Agonist PET Tracers with Low Pancreas Uptake
Wang, Lei, Bratanovic, Ivica Jerolim, Zhang, Zhengxing, Kuo, Hsiou-Ting, Merkens, Helen, Zeisler, Jutta, Zhang, Chengcheng, Tan, Ruiyan, Bénard, François, Lin, Kuo-Shyan
Published in Molecules (Basel, Switzerland) (20.02.2023)
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Published in Molecules (Basel, Switzerland) (20.02.2023)
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