A Synthetically Simple, Click-Generated Cyclam-Based Zinc(II) Sensor
Tamanini, Emiliano, Katewa, Arna, Sedger, Lisa M, Todd, Matthew H, Watkinson, Michael
Published in Inorganic chemistry (05.01.2009)
Published in Inorganic chemistry (05.01.2009)
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Journal Article
Structure of the Epigenetic Oncogene MMSET and Inhibition by N‑Alkyl Sinefungin Derivatives
Tisi, Dominic, Chiarparin, Elisabetta, Tamanini, Emiliano, Pathuri, Puja, Coyle, Joseph E, Hold, Adam, Holding, Finn P, Amin, Nader, Martin, Agnes C. L, Rich, Sharna J, Berdini, Valerio, Yon, Jeff, Acklam, Paul, Burke, Rosemary, Drouin, Ludovic, Harmer, Jenny E, Jeganathan, Fiona, van Montfort, Rob L. M, Newbatt, Yvette, Tortorici, Marcello, Westlake, Maura, Wood, Amy, Hoelder, Swen, Heightman, Tom D
Published in ACS chemical biology (18.11.2016)
Published in ACS chemical biology (18.11.2016)
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Journal Article
Fragment-Based Discovery of a Novel, Brain Penetrant, Orally Active HDAC2 Inhibitor
Tamanini, Emiliano, Miyamura, Shin, Buck, Ildiko M., Cons, Benjamin D., Dawson, Lee, East, Charlotte, Futamura, Takashi, Goto, Shintaro, Griffiths-Jones, Charlotte, Hashimoto, Tetsuya, Heightman, Tom D., Ishikawa, Shunpei, Ito, Hideki, Kaneko, Yosuke, Kawato, Tatsuya, Kondo, Kazumi, Kurihara, Naoki, McCarthy, James M., Mori, Yukiko, Nagase, Tsuyoshi, Nakaishi, Yuichiro, Reeks, Judith, Sato, Akimasa, Schöpf, Patrick, Tai, Kuninori, Tamai, Taichi, Tisi, Dominic, Woolford, Alison J.-A.
Published in ACS medicinal chemistry letters (13.10.2022)
Published in ACS medicinal chemistry letters (13.10.2022)
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Journal Article
Effective Methods for the Biotinylation of Azamacrocycles
Krivickas, Sara J, Tamanini, Emiliano, Todd, Matthew H, Watkinson, Michael
Published in Journal of organic chemistry (26.10.2007)
Published in Journal of organic chemistry (26.10.2007)
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Journal Article
Proton-Driven Switching Between Receptors for C60 and C70
Stefankiewicz, Artur R., Tamanini, Emiliano, Pantoş, G. Dan, Sanders, Jeremy K. M.
Published in Angewandte Chemie International Edition (14.06.2011)
Published in Angewandte Chemie International Edition (14.06.2011)
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Journal Article
Proton-Driven Switching Between Receptors for C60 and C70
Stefankiewicz, Artur R., Tamanini, Emiliano, Pantoş, G. Dan, Sanders, Jeremy K. M.
Published in Angewandte Chemie (14.06.2011)
Published in Angewandte Chemie (14.06.2011)
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Journal Article
Discovery of a Potent Nonpeptidomimetic, Small-Molecule Antagonist of Cellular Inhibitor of Apoptosis Protein 1 (cIAP1) and X‑Linked Inhibitor of Apoptosis Protein (XIAP)
Tamanini, Emiliano, Buck, Ildiko M, Chessari, Gianni, Chiarparin, Elisabetta, Day, James E. H, Frederickson, Martyn, Griffiths-Jones, Charlotte M, Hearn, Keisha, Heightman, Tom D, Iqbal, Aman, Johnson, Christopher N, Lewis, Edward J, Martins, Vanessa, Peakman, Torren, Reader, Michael, Rich, Sharna J, Ward, George A, Williams, Pamela A, Wilsher, Nicola E
Published in Journal of medicinal chemistry (08.06.2017)
Published in Journal of medicinal chemistry (08.06.2017)
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Journal Article
Structure-Based Design of Potent and Orally Active Isoindolinone Inhibitors of MDM2-p53 Protein–Protein Interaction
Chessari, Gianni, Hardcastle, Ian R, Ahn, Jong Sook, Anil, Burcu, Anscombe, Elizabeth, Bawn, Ruth H, Bevan, Luke D, Blackburn, Timothy J, Buck, Ildiko, Cano, Celine, Carbain, Benoit, Castro, Juan, Cons, Ben, Cully, Sarah J, Endicott, Jane A, Fazal, Lynsey, Golding, Bernard T, Griffin, Roger J, Haggerty, Karen, Harnor, Suzannah J, Hearn, Keisha, Hobson, Stephen, Holvey, Rhian S, Howard, Steven, Jennings, Claire E, Johnson, Christopher N, Lunec, John, Miller, Duncan C, Newell, David R, Noble, Martin E. M, Reeks, Judith, Revill, Charlotte H, Riedinger, Christiane, St. Denis, Jeffrey D, Tamanini, Emiliano, Thomas, Huw, Thompson, Neil T, Vinković, Mladen, Wedge, Stephen R, Williams, Pamela A, Wilsher, Nicola E, Zhang, Bian, Zhao, Yan
Published in Journal of medicinal chemistry (08.04.2021)
Published in Journal of medicinal chemistry (08.04.2021)
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Journal Article
Proton‐Driven Switching Between Receptors for C 60 and C 70
Stefankiewicz, Artur R., Tamanini, Emiliano, Pantoş, G. Dan, Sanders, Jeremy K. M.
Published in Angewandte Chemie International Edition (14.06.2011)
Published in Angewandte Chemie International Edition (14.06.2011)
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Journal Article
Fragment-Based Drug Discovery Targeting Inhibitor of Apoptosis Proteins: Discovery of a Non-Alanine Lead Series with Dual Activity Against cIAP1 and XIAP
Chessari, Gianni, Buck, Ildiko M, Day, James E. H, Day, Philip J, Iqbal, Aman, Johnson, Christopher N, Lewis, Edward J, Martins, Vanessa, Miller, Darcey, Reader, Michael, Rees, David C, Rich, Sharna J, Tamanini, Emiliano, Vitorino, Marc, Ward, George A, Williams, Pamela A, Williams, Glyn, Wilsher, Nicola E, Woolford, Alison J.-A
Published in Journal of medicinal chemistry (27.08.2015)
Published in Journal of medicinal chemistry (27.08.2015)
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Journal Article
Abstract 5902: Targeting MAPK-driven tumors via inhibition of MAP2K4
Wade, Mark, Tamanini, Emiliano, Unbekandt, Mathieu, Wallis, Nicola, Lyons, John, Munck, Joanne, Woodhead, Andrew, Schopf, Patrick, Stow, Jessie, East, Charlotte, Clark, Mellissa, Denis, Jeffrey St, Pathuri, Puja
Published in Cancer research (Chicago, Ill.) (22.03.2024)
Published in Cancer research (Chicago, Ill.) (22.03.2024)
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Journal Article
Abstract 1652: Development of a potent class of small molecule inhibitors of the MDM2-p53 protein-protein interaction
Fazal, Lynsey, Ahn, Maria, Bevan, Luke, Buck, Ildiko, Castro, Juan, Chessari, Gianni, Cons, Ben, Hearn, Keisha, Howard, Steven, Johnson, Chris, Reeks, Judith, Tamanini, Emiliano, Thompson, Neil, Walton, Hugh, Williams, Pamela, Bawn, Ruth H., Blackburn, Tim J., Cano, Celine, Cully, Sarah J., Golding, Bernard, Griffin, Roger, Haggerty, Karen, Hardcastle, Ian, Newell, Herbie, Noble, Martin, Thomas, Huw, Willmore, Elaine, Zhao, Yan, Wedge, Steve
Published in Cancer research (Chicago, Ill.) (01.07.2018)
Published in Cancer research (Chicago, Ill.) (01.07.2018)
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Journal Article
Ion Pairs and C 60 : Simultaneous Guests in Supramolecular Nanotubes
Tamanini, Emiliano, Pantoş, G. Dan, Sanders, Jeremy K. M.
Published in Chemistry : a European journal (04.01.2010)
Published in Chemistry : a European journal (04.01.2010)
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Journal Article
Ion Pairs and C sub(60): Simultaneous Guests in Supramolecular Nanotubes
Tamanini, Emiliano, Pantos, GDan, Sanders, JeremyKM
Published in Chemistry : a European journal (01.01.2010)
Published in Chemistry : a European journal (01.01.2010)
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Journal Article
Abstract 6588: Discovery of ASTX295, a potent, next-generation small molecule antagonist of MDM2 with differentiated pharmacokinetic profile
Ahn, Maria, Bevan, Luke, Buck, Ildiko, Cano, Celine, Castro, Juan, Cons, Ben, Endicott, Jane, Fazal, Lynsey, Ferrari, Nicola, Hardcastle, Ian, Hearn, Keisha, Holvey, Rhian, Howard, Steven, Johnson, Chris, Jennings, Claire, Kucia-Tran, Justyna, Kyle, Suzanne, Lunec, John, Lyons, John, Miller, Duncan, Rees, David, Noble, Martin, Newell, David R., Reeks, Judith, Saini, Harpreet, St. Denis, Jeffrey, Tamanini, Emiliano, Thomas, Huw, Thompson, Neil, Vinkovic, Mladen, Ward, George, Wallis, Nicola, Walton, Hugh, Wedge, Stephen, Williams, Pamela, Willmore, Elaine, Wilshire, Nicola, Zhao, Yan, Chessari, Gianni
Published in Cancer research (Chicago, Ill.) (22.03.2024)
Published in Cancer research (Chicago, Ill.) (22.03.2024)
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