Cutting Edge: Piezo1 Mechanosensors Optimize Human T Cell Activation
Liu, Chinky Shiu Chen, Raychaudhuri, Deblina, Paul, Barnali, Chakrabarty, Yogaditya, Ghosh, Amrit Raj, Rahaman, Oindrila, Talukdar, Arindam, Ganguly, Dipyaman
Published in The Journal of immunology (1950) (15.02.2018)
Published in The Journal of immunology (1950) (15.02.2018)
Get full text
Journal Article
Ligand-based Pharmacophore Modeling, Virtual Screening and Molecular Docking Studies for Discovery of Potential Topoisomerase I Inhibitors
Pal, Sourav, Kumar, Vinay, Kundu, Biswajit, Bhattacharya, Debomita, Preethy, Nagothy, Reddy, Mamindla Prashanth, Talukdar, Arindam
Published in Computational and structural biotechnology journal (01.01.2019)
Published in Computational and structural biotechnology journal (01.01.2019)
Get full text
Journal Article
Semisynthetic Quercetin Derivatives with Potent Antitumor Activity in Colon Carcinoma
Mukherjee, Ayan, Mishra, Snehasis, Kotla, Naveen Kumar, Manna, Krishnendu, Roy, Swarnali, Kundu, Biswajit, Bhattacharya, Debomita, Das Saha, Krishna, Talukdar, Arindam
Published in ACS omega (30.04.2019)
Published in ACS omega (30.04.2019)
Get full text
Journal Article
Topoisomerase I inhibitors: Challenges, progress and the road ahead
Talukdar, Arindam, Kundu, Biswajit, Sarkar, Dipayan, Goon, Sunny, Mondal, Mohabul Alam
Published in European journal of medicinal chemistry (05.06.2022)
Published in European journal of medicinal chemistry (05.06.2022)
Get full text
Journal Article
Understanding the riboflavin biosynthesis pathway for the development of antimicrobial agents
Kundu, Biswajit, Sarkar, Dipayan, Ray, Namrata, Talukdar, Arindam
Published in Medicinal research reviews (01.07.2019)
Published in Medicinal research reviews (01.07.2019)
Get full text
Journal Article
Discovery and Development of Quinazolinones and Quinazolinediones for Ameliorating Nonalcoholic Fatty Liver Disease (NAFLD) by Modulating COP1-ATGL Axis
Sarkar, Dipayan, Chowdhury, Saheli, Goon, Sunny, Sen, Abhishek, Dastidar, Uddipta Ghosh, Mondal, Mohabul Alam, Chakrabarti, Partha, Talukdar, Arindam
Published in Journal of medicinal chemistry (28.12.2023)
Published in Journal of medicinal chemistry (28.12.2023)
Get full text
Journal Article
Development, Optimization, and In Vivo Validation of New Imidazopyridine Chemotypes as Dual TLR7/TLR9 Antagonists through Activity-Directed Sequential Incorporation of Relevant Structural Subunits
Das, Nirmal, Bandopadhyay, Purbita, Roy, Swarnali, Sinha, Bishnu Prasad, Dastidar, Uddipta Ghosh, Rahaman, Oindrila, Pal, Sourav, Ganguly, Dipyaman, Talukdar, Arindam
Published in Journal of medicinal chemistry (08.09.2022)
Published in Journal of medicinal chemistry (08.09.2022)
Get full text
Journal Article
A Chemical Switch for Transforming a Purine Agonist for Toll-like Receptor 7 to a Clinically Relevant Antagonist
Mukherjee, Ayan, Raychaudhuri, Deblina, Sinha, Bishnu Prasad, Kundu, Biswajit, Mitra, Mousumi, Paul, Barnali, Bandopadhyay, Purbita, Ganguly, Dipyaman, Talukdar, Arindam
Published in Journal of medicinal chemistry (14.05.2020)
Published in Journal of medicinal chemistry (14.05.2020)
Get full text
Journal Article
Discovery and Mechanistic Study of Tailor-Made Quinoline Derivatives as Topoisomerase 1 Poison with Potent Anticancer Activity
Kundu, Biswajit, Das, Subhendu K, Paul Chowdhuri, Srijita, Pal, Sourav, Sarkar, Dipayan, Ghosh, Arijit, Mukherjee, Ayan, Bhattacharya, Debomita, Das, Benu Brata, Talukdar, Arindam
Published in Journal of medicinal chemistry (11.04.2019)
Published in Journal of medicinal chemistry (11.04.2019)
Get full text
Journal Article
Systematic Optimization of Potent and Orally Bioavailable Purine Scaffold as a Dual Inhibitor of Toll-Like Receptors 7 and 9
Kundu, Biswajit, Raychaudhuri, Deblina, Mukherjee, Ayan, Sinha, Bishnu Prasad, Sarkar, Dipika, Bandopadhyay, Purbita, Pal, Sourav, Das, Nirmal, Dey, Debdeep, Ramarao, Kantubhukta, Nagireddy, Kasireddy, Ganguly, Dipyaman, Talukdar, Arindam
Published in Journal of medicinal chemistry (08.07.2021)
Published in Journal of medicinal chemistry (08.07.2021)
Get full text
Journal Article
Exploring the Structural Attributes of Yoda1 for the Development of New-Generation Piezo1 Agonist Yaddle1 as a Vaccine Adjuvant Targeting Optimal T Cell Activation
Goon, Sunny, Shiu Chen Liu, Chinky, Ghosh Dastidar, Uddipta, Paul, Barnali, Mukherjee, Suravi, Sarkar, Himadri Sekhar, Desai, Milie, Jana, Rituparna, Pal, Sourav, Sreedevi, Namala Venkata, Ganguly, Dipyaman, Talukdar, Arindam
Published in Journal of medicinal chemistry (23.05.2024)
Published in Journal of medicinal chemistry (23.05.2024)
Get full text
Journal Article
Synthesis and characterization of new potent TLR7 antagonists based on analysis of the binding mode using biomolecular simulations
Pal, Sourav, Paul, Barnali, Bandopadhyay, Purbita, Preethy, Nagothy, Sarkar, Dipika, Rahaman, Oindrila, Goon, Sunny, Roy, Swarnali, Ganguly, Dipyaman, Talukdar, Arindam
Published in European journal of medicinal chemistry (15.01.2021)
Published in European journal of medicinal chemistry (15.01.2021)
Get full text
Journal Article
Development of a metabolically stable topoisomerase I poison as anticancer agent
Kundu, Biswajit, Sarkar, Dipayan, Chowdhuri, Srijita Paul, Pal, Sourav, Das, Subhendu K., Das, Benu Brata, Talukdar, Arindam
Published in European journal of medicinal chemistry (15.09.2020)
Published in European journal of medicinal chemistry (15.09.2020)
Get full text
Journal Article
Development of selective class I protein arginine methyltransferase inhibitors through fragment-based drug design approach
Bhattacharya, Debomita, Shi Ming Li, Alice, Paul, Barnali, Ghosh Dastidar, Uddipta, Santhakumar, Vijayaratnam, Sarkar, Dipika, Chau, Irene, Li, Fengling, Ghosh, Trisha, Vedadi, Masoud, Talukdar, Arindam
Published in European journal of medicinal chemistry (15.11.2023)
Published in European journal of medicinal chemistry (15.11.2023)
Get full text
Journal Article
Hit-to-lead optimization of 2-aminoquinazolines as anti-microbial agents against Leishmania donovani
Das, Nirmal, Roy, Jayasree, Patra, Binita, Saunders, Eleanor, Sarkar, Dipika, Goon, Sunny, Sinha, Bishnu Prasad, Roy, Shreya, Roy, Swarnali, Sarif, Jafar, Bandopadhyay, Purbita, Barik, Subhasis, Mukherjee, Suravi, McNamara, Nicole, Varghese, Swapna, Simpson, Kaylene, Baell, Jonathan, McConville, Malcolm, Ganguly, Dipyaman, Talukdar, Arindam
Published in European journal of medicinal chemistry (05.04.2024)
Published in European journal of medicinal chemistry (05.04.2024)
Get full text
Journal Article
Mitigating hERG Liability of Toll‐Like Receptor 9 and 7 Antagonists through Structure‐Based Design
Das, Nirmal, Bhattacharya, Debomita, Bandopadhyay, Purbita, Dastidar, Uddipta Ghosh, Paul, Barnali, Rahaman, Oindrila, Hoque, Israful, Patra, Binita, Ganguly, Dipyaman, Talukdar, Arindam
Published in ChemMedChem (15.06.2023)
Published in ChemMedChem (15.06.2023)
Get full text
Journal Article