Structural development of non-secosteroidal vitamin D receptor (VDR) ligands without any asymmetric carbon
Misawa, Takashi, Tsuji, Genichiro, Takahashi, Takeo, Ochiai, Eiji, Takagi, Ken-ichiro, Horie, Kyohei, Kakuda, Shinji, Takimoto-Kamimura, Midori, Kurihara, Masaaki, Demizu, Yosuke
Published in Bioorganic & medicinal chemistry (15.12.2018)
Published in Bioorganic & medicinal chemistry (15.12.2018)
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Design, synthesis and X-ray crystallographic study of new nonsecosteroidal vitamin D receptor ligands
Demizu, Yosuke, Takahashi, Takeo, Kaneko, Fumiya, Sato, Yukiko, Okuda, Haruhiro, Ochiai, Eiji, Horie, Kyohei, Takagi, Ken-ichiro, Kakuda, Shinji, Takimoto-Kamimura, Midori, Kurihara, Masaaki
Published in Bioorganic & medicinal chemistry letters (15.10.2011)
Published in Bioorganic & medicinal chemistry letters (15.10.2011)
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Synthesis and Biological Activities of 1α,4α,25- and 1α,4β,25-Trihydroxyvitamin D3 and Their Metabolism by Human CYP24A1 and UDP-Glucuronosyltransferase
Sawada, Daisuke, Tsukuda, Yuya, Yasuda, Kaori, Sakaki, Toshiyuki, Saito, Hiroshi, Takagi, Ken-ichiro, Takenouchi, Kazuya, Chen, Tai C., Reddy, G. Satyanarayana, Kittaka, Atsushi
Published in Chemical & pharmaceutical bulletin (01.10.2012)
Published in Chemical & pharmaceutical bulletin (01.10.2012)
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Synthesis and Biological Evaluation of 4-Substituted Vitamin D and 14-Epi-Previtamin D Analogs
Sawada, Daisuke, Tsukuda, Yuya, Saito, Hiroshi, Takagi, Ken-ichiro, Horie, Kyouhei, Ochiai, Eiji, Takenouchi, Kazuya, Kittaka, Atsushi
Published in Chemical & Pharmaceutical Bulletin (01.12.2009)
Published in Chemical & Pharmaceutical Bulletin (01.12.2009)
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Cloning and Characterization of the cDNA for Human Airway Trypsin-like Protease
Yamaoka, K, Masuda, K, Ogawa, H, Takagi, K, Umemoto, N, Yasuoka, S
Published in The Journal of biological chemistry (08.05.1998)
Published in The Journal of biological chemistry (08.05.1998)
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Journal Article
Synthesis and Biological Activities of 1α,4α,25- and 1α,4β,25-Trihydroxyvitamin D3 and Their Metabolism by Human CYP24A1 and UDP-Glucuronosyltransferase
Daisuke Sawadaa, Yuya Tsukudaa, Kaori Yasudab, Toshiyuki Sakakib, Hiroshi Saitoc, Ken-ichiro Takagic, Kazuya Takenouchic, Tai C.Chend, G.Satyanarayana Reddye, f, Atsushi Kittakaa
Published in Chemical and Pharmaceutical Bulletin (01.10.2012)
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Published in Chemical and Pharmaceutical Bulletin (01.10.2012)
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Synthesis and metabolic studies of 1α,2α,25-, 1α,4α,25- and 1α,4β,25-trihydroxyvitamin D3
Takano, Masashi, Sawada, Daisuke, Yasuda, Kaori, Nishikawa, Miyu, Takeuchi, Akiko, Takagi, Ken-ichiro, Horie, Kyohei, Reddy, G. Satyanarayana, Chen, Tai C., Sakaki, Toshiyuki, Kittaka, Atsushi
Published in The Journal of steroid biochemistry and molecular biology (01.04.2015)
Published in The Journal of steroid biochemistry and molecular biology (01.04.2015)
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Journal Article
Synthesis of 2α-Heteroarylalkyl Active Vitamin D3 with Therapeutic Effect on Enhancing Bone Mineral Density in Vivo
Matsuo, Miki, Hasegawa, Asami, Takano, Masashi, Saito, Hiroshi, Kakuda, Shinji, Chida, Takayuki, Takagi, Ken-ichiro, Ochiai, Eiji, Horie, Kyohei, Harada, Yoshifumi, Takimoto-Kamimura, Midori, Takenouchi, Kazuya, Sawada, Daisuke, Kittaka, Atsushi
Published in ACS medicinal chemistry letters (11.07.2013)
Published in ACS medicinal chemistry letters (11.07.2013)
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Journal Article
Synthesis of 2α- and 2β-substituted-14- epi-previtamin D 3 and their genomic activity
Sawada, Daisuke, Katayama, Tomoyuki, Tsukuda, Yuya, Saito, Nozomi, Saito, Hiroshi, Takagi, Ken-ichiro, Ochiai, Eiji, Ishizuka, Seiichi, Takenouchi, Kazuya, Kittaka, Atsushi
Published in Tetrahedron (17.07.2010)
Published in Tetrahedron (17.07.2010)
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New C15-Substituted Active Vitamin D3
Shindo, Kanako, Kumagai, Go, Takano, Masashi, Sawada, Daisuke, Saito, Nozomi, Saito, Hiroshi, Kakuda, Shinji, Takagi, Ken-ichiro, Ochiai, Eiji, Horie, Kyohei, Takimoto-Kamimura, Midori, Ishizuka, Seiichi, Takenouchi, Kazuya, Kittaka, Atsushi
Published in Organic letters (03.06.2011)
Published in Organic letters (03.06.2011)
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Journal Article
Synthesis of 2β-substituted-14-epi-previtamin D3 and testing of its genomic activity
SAWADA, Daisuke, TSUKUDA, Yuya, SAITO, Hiroshi, TAKAGI, Ken-Ichiro, OCHIAI, Eiji, ISHIZUKA, Seiichi, TAKENOUCHI, Kazuya, KITTAKA, Atsushi
Published in Journal of steroid biochemistry and molecular biology (01.07.2010)
Published in Journal of steroid biochemistry and molecular biology (01.07.2010)
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Conference Proceeding
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Retracted: CDP/Cut is an osteoblastic coactivator of the vitamin D receptor (VDR)
Ochiai, Eiji, Kitagawa, Hirochika, Takada, Ichiro, Fujiyama, Sally, Sawatsubashi, Shun, Kim, Mi‐sun, Mezaki, Yoshihiro, Tsushima, Yu, Takagi, Ken‐ichiro, Azuma, Yoshiaki, Takeyama, Ken‐ichi, Yamaoka, Kazuyoshi, Kato, Shigeaki, Kamimura, Takashi
Published in Journal of bone and mineral research (01.02.2013)
Published in Journal of bone and mineral research (01.02.2013)
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Journal Article
CDP/Cut Is an Osteoblastic Coactivator of the Vitamin D Receptor (VDR)
OCHIAI, Eiji, KITAGAWA, Hirochika, TAKEYAMA, Ken-Ichi, YAMAOKA, Kazuyoshi, KATO, Shigeaki, KAMIMURA, Takashi, TAKADA, Ichiro, FUJIYAMA, Sally, SAWATSUBASHI, Shun, KIM, Mi-Sun, MEZAKI, Yoshihiro, TSUSHIMA, Yu, TAKAGI, Ken-Ichiro, AZUMA, Yoshiaki
Published in Journal of bone and mineral research (01.05.2010)
Published in Journal of bone and mineral research (01.05.2010)
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Journal Article
Synthesis of 2α-substituted-14-epi-previtamin D3 and its genomic activity
SAWADA, Daisuke, KATAYAMA, Tomoyuki, KITTAKA, Atsushi, TSUKUDA, Yuya, SAITO, Nozomi, TAKANO, Masashi, SAITO, Hiroshi, TALCAGI, Ken-Ichiro, OCHIAI, Eiji, ISHIZUKA, Seiichi, TALCENOUCHI, Kazuya
Published in Bioorganic & medicinal chemistry letters (15.09.2009)
Published in Bioorganic & medicinal chemistry letters (15.09.2009)
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Journal Article
Retracted: CDP/cut is an osteoblastic coactivator of the vitamin D receptor (VDR)
Ochiai, Eiji, Kitagawa, Hirochika, Takada, Ichiro, Fujiyama, Sally, Sawatsubashi, Shun, Kim, Mi‐sun, Mezaki, Yoshihiro, Tsushima, Yu, Takagi, Ken‐ichiro, Azuma, Yoshiaki, Takeyama, Ken‐ichi, Yamaoka, Kazuyoshi, Kato, Shigeaki, Kamimura, Takashi
Published in Journal of bone and mineral research (01.05.2010)
Published in Journal of bone and mineral research (01.05.2010)
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Journal Article
Sequence of xynC and properties of XynC, a major component of the Clostridium thermocellum cellulosome
Hayashi, H, Takagi, K I, Fukumura, M, Kimura, T, Karita, S, Sakka, K, Ohmiya, K
Published in Journal of Bacteriology (01.07.1997)
Published in Journal of Bacteriology (01.07.1997)
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Journal Article
METHOD FOR SCREENING FOR VITAMIN D RECEPTOR LIGAND
OCHIAI, EIJI, TSUSHIMA, YU, KITAGAWA, HIROCHIKA, YAMAOKA, KAZUYOSHI, TAKAGI, KEN-ICHIRO, KATO, SHIGEAKI, TAKADA, ICHIRO
Year of Publication 07.02.2008
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Year of Publication 07.02.2008
Patent
Synthesis of 2 alpha-Heteroarylalkyl Active Vitamin D-3 with Therapeutic Effect on Enhancing Bone Mineral Density in Vivo
Matsuo, Mild, Hasegawa, Asami, Takano, Masashi, Saito, Hiroshi, Kakuda, Shinji, Chida, Takayuld, Takagi, Ken-ichiro, Ochiai, Eiji, Horie, Kyohei, Harada, Yoshifumi, Takimoto-Kamimura, Midori, Takenouchi, Kazuya, Sawada, Daisuke, Kittaka, Atsushi
Published in ACS medicinal chemistry letters (11.07.2013)
Published in ACS medicinal chemistry letters (11.07.2013)
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Journal Article
New C15-Substituted Active Vitamin D-3
Shindo, Kanako, Kumagai, Go, Takano, Masashi, Sawada, Daisuke, Saito, Nozomi, Saito, Hiroshi, Kakuda, Shinji, Takagi, Ken-ichiro, Ochiai, Eiji, Horie, Kyohei, Takimoto-Kamimura, Midori, Ishizuka, Seiichi, Takenouchi, Kazuya, Kittaka, Atsushi
Published in Organic letters (03.06.2011)
Published in Organic letters (03.06.2011)
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Journal Article
Synthesis and Biological Activities of 1 alpha,4 alpha,25-and 1 alpha,4 beta,25-Trihydroxyvitamin D-3 and Their Metabolism by Human CYP24A1 and UDP-Glucuronosyltransferase
Sawada, Daisuke, Tsukuda, Yuya, Yasuda, Kaori, Sakaki, Toshiyuki, Saito, Hiroshi, Takagi, Ken-ichiro, Takenouchi, Kazuya, Chen, Tai C., Reddy, G. Satyanarayana, Kittaka, Atsushi
Published in Chemical & pharmaceutical bulletin (01.10.2012)
Published in Chemical & pharmaceutical bulletin (01.10.2012)
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Journal Article