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Published in Journal of medicinal chemistry (12.03.2020)
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Published in Pharmacological reports (01.04.2020)
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Published in European journal of medicinal chemistry (15.08.2019)
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Published in Journal of medicinal chemistry (06.06.2002)
Published in Journal of medicinal chemistry (06.06.2002)
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Spiroxatrine derivatives towards 5-HT1A receptor selectivity
Sorbi, Claudia, Tait, Annalisa, Battisti, Umberto M., Brasili, Livio
Published in Pharmacological reports (01.04.2020)
Published in Pharmacological reports (01.04.2020)
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Novel Dithiolane-Based Ligands Combining Sigma and NMDA Receptor Interactions as Potential Neuroprotective Agents
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Published in ACS medicinal chemistry letters (14.05.2020)
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Scouting new sigma receptor ligands: Synthesis, pharmacological evaluation and molecular modeling of 1,3-dioxolane-based structures and derivatives
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Discovery of a benzothiophene-flavonol halting miltefosine and antimonial drug resistance in Leishmania parasites through the application of medicinal chemistry, screening and genomics
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Published in European journal of medicinal chemistry (01.12.2019)
Published in European journal of medicinal chemistry (01.12.2019)
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Medicinal Chemistry in Parasitology: New Avenues in Drug Discovery
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Borsari, Chiara, Luciani, Rosaria, Pozzi, Cecilia, Poehner, Ina, Henrich, Stefan, Trande, Matteo, Cordeiro-da-Silva, Anabela, Santarem, Nuno, Baptista, Catarina, Tait, Annalisa, Di Pisa, Flavio, Dello Iacono, Lucia, Landi, Giacomo, Gul, Sheraz, Wolf, Markus, Kuzikov, Maria, Ellinger, Bernhard, Reinshagen, Jeanette, Witt, Gesa, Gribbon, Philip, Kohler, Manfred, Keminer, Oliver, Behrens, Birte, Costantino, Luca, Tejera Nevado, Paloma, Bifeld, Eugenia, Eick, Julia, Clos, Joachim, Torrado, Juan, Jiménez-Antón, María D, Corral, María J, Alunda, José Ma, Pellati, Federica, Wade, Rebecca C, Ferrari, Stefania, Mangani, Stefano, Costi, Maria Paola
Published in Journal of medicinal chemistry (25.08.2016)
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Published in European journal of medicinal chemistry (24.11.2014)
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Borsari, Chiara, Santarem, Nuno, Torrado, Juan, Olías, Ana Isabel, Corral, María Jesús, Baptista, Catarina, Gul, Sheraz, Wolf, Markus, Kuzikov, Maria, Ellinger, Bernhard, Witt, Gesa, Gribbon, Philip, Reinshagen, Jeanette, Linciano, Pasquale, Tait, Annalisa, Costantino, Luca, Freitas-Junior, Lucio H., Moraes, Carolina B., Bruno dos Santos, Pascoalino, Alcântara, Laura Maria, Franco, Caio Haddad, Bertolacini, Claudia Danielli, Fontana, Vanessa, Tejera Nevado, Paloma, Clos, Joachim, Alunda, José María, Cordeiro-da-Silva, Anabela, Ferrari, Stefania, Costi, Maria Paola
Published in European journal of medicinal chemistry (27.01.2017)
Published in European journal of medicinal chemistry (27.01.2017)
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Synthesis and biological evaluation of 1,3-dioxolane-based 5-HT 1A receptor agonists for CNS disorders and neuropathic pain
Franchini, Silvia, Bencheva, Leda Ivanova, Battisti, Umberto Maria, Tait, Annalisa, Sorbi, Claudia, Fossa, Paola, Cichero, Elena, Ronsisvalle, Simone, Aricò, Giuseppina, Denora, Nunzio, Iacobazzi, Rosa Maria, Cilia, Antonio, Pirona, Lorenza, Brasili, Livio
Published in Future medicinal chemistry (01.09.2018)
Published in Future medicinal chemistry (01.09.2018)
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Structure-Activity Relationships within a Series of sigma(1) and sigma(2) Receptor Ligands: Identification of a sigma(2) Receptor Agonist (BS148) with Selective Toxicity against Metastatic Melanoma
Franchini, Silvia, Sorbi, Claudia, Battisti, Umberto Maria, Tait, Annalisa, Bencheva, Leda Ivanova, Cichero, Elena, Fossa, Paola, Cilia, Antonio, Prezzavento, Orazio, Ronsisvalle, Simone, Arico, Giuseppina, Benassi, Luisa, Vaschieri, Cristina, Azzoni, Paola, Magnoni, Cristina, Brasili, Livio
Published in ChemMedChem (22.11.2017)
Published in ChemMedChem (22.11.2017)
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Journal Article
Structure–Activity Relationships within a Series of σ1 and σ2 Receptor Ligands: Identification of a σ2 Receptor Agonist (BS148) with Selective Toxicity against Metastatic Melanoma
Franchini, Silvia, Sorbi, Claudia, Battisti, Umberto Maria, Tait, Annalisa, Bencheva, Leda Ivanova, Cichero, Elena, Fossa, Paola, Cilia, Antonio, Prezzavento, Orazio, Ronsisvalle, Simone, Aricò, Giuseppina, Benassi, Luisa, Vaschieri, Cristina, Azzoni, Paola, Magnoni, Cristina, Brasili, Livio
Published in ChemMedChem (22.11.2017)
Published in ChemMedChem (22.11.2017)
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Diastereoselective Synthesis of (1,3-Dioxan-4-yl)pyrimidine and Purin Nucleoside Analogues
Battisti, Umberto M., Sorbi, Claudia, Quotadamo, Antonio, Franchini, Silvia, Tait, Annalisa, Schols, Dominique, Jeong, Lak Shin, Lee, Sang Kook, Song, Jayoung, Brasili, Livio
Published in European journal of organic chemistry (01.02.2015)
Published in European journal of organic chemistry (01.02.2015)
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Silvia Franchini, Umberto M. Battisti, Claudia Sorbi, Annalisa Tait, Andrea Cornia, 정낙신, 이상국, 송자영, Roberta Loddo, Silvia Madeddu, Giuseppina Sanna, Livio Brasili
Published in Archives of pharmacal research (01.05.2017)
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Published in Archives of pharmacal research (01.05.2017)
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Synthesis and Structure-Activity Relationships of Triazaspirodecanone Derivatives as Nociceptin/Orphanin FQ Receptor Ligands
Corrado, Sandra, Battisti, Umberto M., Sorbi, Claudia, Tait, Annalisa, Malfacini, Davide, Camarda, Valeria, Calò, Girolamo, Brasili, Livio
Published in Chemical biology & drug design (01.10.2015)
Published in Chemical biology & drug design (01.10.2015)
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