A new class of antibacterials, the imidazopyrazinones, reveal structural transitions involved in DNA gyrase poisoning and mechanisms of resistance
Germe, Thomas, Vörös, Judit, Jeannot, Frederic, Taillier, Thomas, Stavenger, Robert A, Bacqué, Eric, Maxwell, Anthony, Bax, Benjamin D
Published in Nucleic acids research (04.05.2018)
Published in Nucleic acids research (04.05.2018)
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Journal Article
Optimization of the Antibacterial Spectrum and the Developability Profile of the Novel-Class Natural Product Corramycin
Renard, Stephane, Versluys, Stéphanie, Taillier, Thomas, Dubarry, Nelly, Leroi-Geissler, Corinne, Rey, Astrid, Cornaire, Emilie, Sordello, Sylvie, Carry, Jean-Christophe B., Angouillant-Boniface, Odile, Gouyon, Thierry, Thompson, Fabienne, Lebourg, Gilles, Certal, Victor, Balazs, Laszlo, Arranz, Esther, Doerflinger, Gilles, Bretin, Francois, Gervat, Vincent, Brohan, Eric, Kraft, Volker, Boulenc, Xavier, Ducelier, Cécile, Bacqué, Eric, Couturier, Cédric
Published in Journal of medicinal chemistry (28.12.2023)
Published in Journal of medicinal chemistry (28.12.2023)
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Structure Elucidation, Total Synthesis, Antibacterial In Vivo Efficacy and Biosynthesis Proposal of Myxobacterial Corramycin
Couturier, Cédric, Groß, Sebastian, Tesmar, Alexander, Hoffmann, Judith, Deckarm, Selina, Fievet, Anouchka, Dubarry, Nelly, Taillier, Thomas, Pöverlein, Christoph, Stump, Heike, Kurz, Michael, Toti, Luigi, Haag Richter, Sabine, Schummer, Dietmar, Sizun, Philippe, Hoffmann, Michael, Prasad Awal, Ram, Zaburannyi, Nestor, Harmrolfs, Kirsten, Wink, Joachim, Lessoud, Emilie, Vermat, Thierry, Cazals, Veronique, Silve, Sandra, Bauer, Armin, Mourez, Michael, Fraisse, Laurent, Leroi‐Geissler, Corinne, Rey, Astrid, Versluys, Stéphanie, Bacqué, Eric, Müller, Rolf, Renard, Stephane
Published in Angewandte Chemie International Edition (19.12.2022)
Published in Angewandte Chemie International Edition (19.12.2022)
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Journal Article
Studies of antibacterial activity (in vitro and in vivo) and mode of action for des-acyl tridecaptins (DATs)
Couturier, Cédric, Ronzon, Quentin, Lattanzi, Giulia, Lingard, Iain, Coyne, Sebastien, Cazals, Veronique, Dubarry, Nelly, Yvon, Stephane, Leroi-Geissler, Corinne, Gracia, Obdulia Rabal, Teague, Joanne, Sordello, Sylvie, Corbett, David, Bauch, Caroline, Monlong, Chantal, Payne, Lloyd, Taillier, Thomas, Fuchs, Hazel, Broenstrup, Mark, Harrison, Peter H., Moynié, Lucile, Lakshminarayanan, Abirami, Gianga, Tiberiu-Marius, Hussain, Rohanah, Naismith, James H., Mourez, Michael, Bacqué, Eric, Björkling, Fredrik, Sabuco, Jean-Francois, Franzyk, Henrik
Published in European journal of medicinal chemistry (05.02.2024)
Published in European journal of medicinal chemistry (05.02.2024)
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Journal Article
A new class of antibacterials, the imidazopyrazinones, reveal structural transitions involved in DNA gyrase poisoning and mechanisms of resistance
Germe, Thomas, Vörös, Judit, Jeannot, Frederic, Taillier, Thomas, Stavenger, Robert A, Bacqué, Eric, Maxwell, Anthony, Bax, Benjamin D
Published in Nucleic acids research (04.05.2018)
Published in Nucleic acids research (04.05.2018)
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Journal Article
Imidazopyrazinones (IPYs): Non-Quinolone Bacterial Topoisomerase Inhibitors Showing Partial Cross-Resistance with Quinolones
Jeannot, Frédéric, Taillier, Thomas, Despeyroux, Pierre, Renard, Stéphane, Rey, Astrid, Mourez, Michaël, Poeverlein, Christoph, Khichane, Imène, Perrin, Marc-Antoine, Versluys, Stéphanie, Stavenger, Robert A, Huang, Jianzhong, Germe, Thomas, Maxwell, Anthony, Cao, Sha, Huseby, Douglas L, Hughes, Diarmaid, Bacqué, Eric
Published in Journal of medicinal chemistry (26.04.2018)
Published in Journal of medicinal chemistry (26.04.2018)
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Journal Article
Strukturaufklärung, Totalsynthese, In‐Vivo‐Aktivität und Potentieller Biosyntheseweg des Neuen Myxobakteriellen Antibiotikums Corramycin
Couturier, Cédric, Groß, Sebastian, von Tesmar, Alexander, Hoffmann, Judith, Deckarm, Selina, Fievet, Anouchka, Dubarry, Nelly, Taillier, Thomas, Pöverlein, Christoph, Stump, Heike, Kurz, Michael, Toti, Luigi, Haag Richter, Sabine, Schummer, Dietmar, Sizun, Philippe, Hoffmann, Michael, Prasad Awal, Ram, Zaburannyi, Nestor, Harmrolfs, Kirsten, Wink, Joachim, Lessoud, Emilie, Vermat, Thierry, Cazals, Veronique, Silve, Sandra, Bauer, Armin, Mourez, Michael, Fraisse, Laurent, Leroi‐Geissler, Corinne, Rey, Astrid, Versluys, Stéphanie, Bacqué, Eric, Müller, Rolf, Renard, Stephane
Published in Angewandte Chemie (19.12.2022)
Published in Angewandte Chemie (19.12.2022)
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Journal Article
Strukturaufklärung, Totalsynthese, In‐Vivo‐Aktivität und Potentieller Biosyntheseweg des Neuen Myxobakteriellen Antibiotikums Corramycin
Couturier, Cédric, Groß, Sebastian, Tesmar, Alexander, Hoffmann, Judith, Deckarm, Selina, Fievet, Anouchka, Dubarry, Nelly, Taillier, Thomas, Pöverlein, Christoph, Stump, Heike, Kurz, Michael, Toti, Luigi, Haag Richter, Sabine, Schummer, Dietmar, Sizun, Philippe, Hoffmann, Michael, Prasad Awal, Ram, Zaburannyi, Nestor, Harmrolfs, Kirsten, Wink, Joachim, Lessoud, Emilie, Vermat, Thierry, Cazals, Veronique, Silve, Sandra, Bauer, Armin, Mourez, Michael, Fraisse, Laurent, Leroi‐Geissler, Corinne, Rey, Astrid, Versluys, Stéphanie, Bacqué, Eric, Müller, Rolf, Renard, Stephane
Published in Angewandte Chemie (19.12.2022)
Published in Angewandte Chemie (19.12.2022)
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Journal Article