Discovery of A‑971432, An Orally Bioavailable Selective Sphingosine-1-Phosphate Receptor 5 (S1P5) Agonist for the Potential Treatment of Neurodegenerative Disorders
Hobson, Adrian D, Harris, Christopher M, van der Kam, Elizabeth L, Turner, Sean C, Abibi, Ayome, Aguirre, Ana L, Bousquet, Peter, Kebede, Tegest, Konopacki, Donald B, Gintant, Gary, Kim, Youngjae, Larson, Kelly, Maull, John W, Moore, Nigel S, Shi, Dan, Shrestha, Anurupa, Tang, Xiubo, Zhang, Peng, Sarris, Kathy K
Published in Journal of medicinal chemistry (10.12.2015)
Published in Journal of medicinal chemistry (10.12.2015)
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Microwave-Assisted Synthesis of Novel (5-Nitropyridin-2-yl)alkyl and (5-Nitropyridin-3-yl)alkyl Carbamates
Henry, Christophe, Haupt, Andreas, Turner, Sean C
Published in Journal of organic chemistry (06.03.2009)
Published in Journal of organic chemistry (06.03.2009)
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Setting International Standards in Analyzing Patient-Reported Outcomes and Quality of Life Endpoints in Cancer Clinical Trials-Innovative Medicines Initiative (SISAQOL-IMI): stakeholder views, objectives, and procedures
Alanya, Ahu, Falk, Ragnhild Sorum, Bjordal, Kristin, Chang, Jane, Cislo, Paul, Coens, Corneel, Dirven, Linda, Speck, Rebecca M, Fitzgerald, Kristina, Galinsky, Jayne, Giesinger, Johannes M, Holzner, Bernhard, Le Cessie, Saskia, O'Connor, Daniel, Oliver, Kathy, Quinten, Chantal, Schlichting, Michael, Ren, Jinma, Roychoudhury, Satrajit, Taphoorn, Martin J B, Velikova, Galina, Wintner, Lisa M, Bottomley, Andrew, Bui, Cat, Kamalakar, Rajesh, Sail, Kavita, Sen, Rohini, Turner, Sean C, Cocks, Kim, Su, Yun, Peil, Barbara, Voorhaar, Maarten, Wong, Brendon, Dekanic Arbanas, Gracia, Kuljanic, Karin, Rede, Ivana, Arraras, Juan, Coons, Stephen Joel, Murray, Lindsey, Pignatti, Francesco, Martinelli, Francesca, Musoro, Jammbe, Dafni, Ourania, De Vries, Elisabeth, Gyawali, Bishal, Kiesewetter, Barbara, Roitberg, Felipe, Schoepf, Felix, Tschuggnall, Michael, Sasseville, Maxime, Soltys, Katherine, Ferrer, Montserrat, Garin, Olatz, Vilagut, Gemma, Schürmann, Christoph, Wieseler, Beate, Snyder, Claire, Alonso Abad, Ariel, Bogaerts, Kris, Brackx, Febe, Molenberghs, Geert, Verbeke, Geert, Choi, Jan, Thomassen, Doranne, Geissler, Jan, Sauerbrei, Willi, Pilz, Micha Johannes, Campbell, Lisa, Rantell, Khadija, Desplanques, Gregoire, Regnault, Antoine, Morgan, Kate, Plate, Ananda, ten Seldam, Silene, Terada, Mitsumi, Mizusawa, Junki, Wilder Smith, Ashley, Reksten, Tove Ragna, Cappelleri, Joseph, de Besi, Patrizia, Russell-Smith, Alexander, Sandin, Rickard, Mamolo, Carla, Tu, Dongsheng, Petersen, Morten, Cleeland, Charlie, Williams, Lori, Calvert, Melanie, Cruz Rivera, Samantha, Aiyegbusi, Olalekan Lee, Goetghebeur, Els, Van Lancker, Kelly, Boele, Florien, Gilbert, Alexandra, Peacock, Rosemary, King, Madeleine, Bhatnagar, Vishal, Fiero, Mallorie, Johnson, Laura Lee, Rodriguez, Lisa
Published in The lancet oncology (01.06.2023)
Published in The lancet oncology (01.06.2023)
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eTRANSAFE: data science to empower translational safety assessment
Sanz, Ferran, Pognan, François, Steger-Hartmann, Thomas, Díaz, Carlos, Asakura, Shoji, Amberg, Alexander, Bécourt-Lhote, Nathalie, Blomberg, Niklas, Bosc, Nicolas, Briggs, Katharine, Bringezu, Frank, Brulle-Wohlhueter, Claire, Brunak, Søren, Bueters, Ruud, Callegaro, Giulia, Capella-Gutierrez, Salvador, Centeno, Emilio, Corvi, Javier, Cronin, Mark T D, Drew, Philip, Duchateau-Nguyen, Guillemette, Ecker, Gerhard F, Escher, Sylvia, Felix, Eloy, Ferreiro, Miguel, Frericks, Markus, Furlong, Laura I, Geiger, Robert, George, Catherine, Grandits, Melanie, Ivanov-Draganov, Dragomir, Kilgour-Christie, Jean, Kiziloren, Tevfik, Kors, Jan A, Koyama, Naoki, Kreuchwig, Annika, Leach, Andrew R, Mayer, Miguel-Angel, Monecke, Peter, Muster, Wolfgang, Nakazawa, Chihiro Miyamoto, Nicholson, Gavin, Parry, Rowan, Pastor, Manuel, Piñero, Janet, Oberhauser, Nils, Ramírez-Anguita, Juan Manuel, Rodrigo, Adrián, Smajic, Aljosa, Schaefer, Markus, Schieferdecker, Sebastian, Soininen, Inari, Terricabras, Emma, Trairatphisan, Panuwat, Turner, Sean C, Valencia, Alfonso, van de Water, Bob, van der Lei, Johan L, van Mulligen, Erik M, Vock, Esther, Wilkinson, David
Published in Nature reviews. Drug discovery (01.08.2023)
Published in Nature reviews. Drug discovery (01.08.2023)
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Anticonvulsant effects of structurally diverse GABA(B) positive allosteric modulators in the DBA/2J audiogenic seizure test: Comparison to baclofen and utility as a pharmacodynamic screening model
Brown, Jordan W, Moeller, Achim, Schmidt, Martin, Turner, Sean C, Nimmrich, Volker, Ma, Junli, Rueter, Lynne E, van der Kam, Elizabeth, Zhang, Min
Published in Neuropharmacology (01.02.2016)
Published in Neuropharmacology (01.02.2016)
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The discovery of a new class of large-conductance Ca2+-activated K+ channel opener targeted for overactive bladder: Synthesis and structure-activity relationships of 2-amino-4-azaindoles
TURNER, Sean C, CARROLL, William A, SULLIVAN, James P, WHITE, Tammie K, GOPALAKRISHNAN, Murali, COGHLAN, Michael J, SHIEH, Char-Chang, ZHANG, Xu-Feng, PARIHAR, Ashutosh S, BUCKNER, Steven A, MILICIC, Ivan
Published in Bioorganic & medicinal chemistry letters (16.06.2003)
Published in Bioorganic & medicinal chemistry letters (16.06.2003)
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A national study of the processes and outcomes of paediatric formulary applications in Australia
Sinha, Yashwant K, Craig, Jonathan C, Barclay, Peter G, Miller, Hugh, Turner, Sean C, Whitehouse, Joseph P, Brien, Jo-anne E
Published in Medical journal of Australia (19.05.2014)
Published in Medical journal of Australia (19.05.2014)
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α-Methylation at benzylic fragment of N-aryl- N′-benzyl ureas provides TRPV1 antagonists with better pharmacokinetic properties and higher efficacy in inflammatory pain model
Gomtsyan, Arthur, Bayburt, Erol K., Keddy, Ryan, Turner, Sean C., Jinkerson, Tammie K., Didomenico, Stanley, Perner, Richard J., Koenig, John R., Drizin, Irene, McDonald, Heath A., Surowy, Carol S., Honore, Prisca, Mikusa, Joe, Marsh, Kennan C., Wetter, Jill M., Faltynek, Connie R., Lee, Chih-Hung
Published in Bioorganic & medicinal chemistry letters (15.07.2007)
Published in Bioorganic & medicinal chemistry letters (15.07.2007)
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In Vitro Structure−Activity Relationship and In Vivo Characterization of 1-(Aryl)-3-(4-(amino)benzyl)urea Transient Receptor Potential Vanilloid 1 Antagonists
Perner, Richard J, DiDomenico, Stanley, Koenig, John R, Gomtsyan, Arthur, Bayburt, Erol K, Schmidt, Robert G, Drizin, Irene, Zheng, Guo Zhu, Turner, Sean C, Jinkerson, Tammie, Brown, Brian S, Keddy, Ryan G, Lukin, Kurill, McDonald, Heath A, Honore, Prisca, Mikusa, Joe, Marsh, Kennan C, Wetter, Jill M, St. George, Karen, Jarvis, Michael F, Faltynek, Connie R, Lee, Chih-Hung
Published in Journal of medicinal chemistry (26.07.2007)
Published in Journal of medicinal chemistry (26.07.2007)
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Enantiospecific Synthesis of Annulated Nicotine Analogues from d- and l-Glutamic Acid. Pyridotropanes
Turner, Sean C, Zhai, Hongbin, Rapoport, Henry
Published in Journal of organic chemistry (11.02.2000)
Published in Journal of organic chemistry (11.02.2000)
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Perceived and actual paracetamol dosing in overweight and obese children
Wiese, Michael David, Sluggett, Janet Kathleen, Wilson, Courtenay Jay, Reuter, Stephanie E, Turner, Sean C, Evans, Allan M
Published in European journal of hospital pharmacy. Science and practice (01.10.2012)
Published in European journal of hospital pharmacy. Science and practice (01.10.2012)
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Synthesis and Structure−Activity Relationships of a Novel Series of Tricyclic Dihydropyridine-Based KATP Openers That Potently Inhibit Bladder Contractions in Vitro
Carroll, William A, Agrios, Konstantinos A, Altenbach, Robert J, Buckner, Steven A, Chen, Yiyuan, Coghlan, Michael J, Daza, Anthony V, Drizin, Irene, Gopalakrishnan, Murali, Henry, Rodger F, Kort, Michael E, Kym, Philip R, Milicic, Ivan, Smith, Jamie C, Tang, Rui, Turner, Sean C, Whiteaker, Kristi L, Zhang, Henry, Sullivan, James P
Published in Journal of medicinal chemistry (03.06.2004)
Published in Journal of medicinal chemistry (03.06.2004)
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Structure–activity studies of a novel series of 5,6-fused heteroaromatic ureas as TRPV1 antagonists
Drizin, Irene, Gomtsyan, Arthur, Bayburt, Erol K., Schmidt, Robert G., Zheng, Guo Zhu, Perner, Richard J., DiDomenico, Stanley, Koenig, John R., Turner, Sean C., Jinkerson, Tammie K., Brown, Brian S., Keddy, Ryan G., McDonald, Heath A., Honore, Prisca, Wismer, Carol T., Marsh, Kennan C., Wetter, Jill M., Polakowski, James S., Segreti, Jason A., Jarvis, Michael F., Faltynek, Connie R., Lee, Chih-Hung
Published in Bioorganic & medicinal chemistry (15.07.2006)
Published in Bioorganic & medicinal chemistry (15.07.2006)
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A new class of histamine H3-Receptor antagonists: Synthesis and structure-activity relationships of 7,8,9,10-tetrahydro-6H-cyclohepta[b]quinolines
TURNER, Sean C, ESBENSHADE, Timothy A, BENNANI, Youssef L, HANCOCK, Arthur A
Published in Bioorganic & medicinal chemistry letters (07.07.2003)
Published in Bioorganic & medicinal chemistry letters (07.07.2003)
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Journal Article
In vitro and in vivo characterization of a novel naphthylamide ATP‐sensitive K+ channel opener, A‐151892
Gopalakrishnan, Murali, Buckner, Steven A, Shieh, Char‐Chang, Fey, Thomas, Fabiyi, Adebola, Whiteaker, Kristi L, Davis‐Taber, Rachel, Milicic, Ivan, Daza, Anthony V, Scott, Victoria E S, Castle, Neil A, Printzenhoff, David, London, Brecht, Turner, Sean C, Carroll, William A, Sullivan, James P, Coghlan, Michael J, Brune, Michael E
Published in British journal of pharmacology (01.09.2004)
Published in British journal of pharmacology (01.09.2004)
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Journal Article
Structure–activity relationship of a novel class of naphthyl amide KATP channel openers
Turner, Sean C, Carroll, William A, White, Tammie K, Brune, Michael E, Buckner, Steven A, Gopalakrishnan, Murali, Fabiyi, Adebola, Coghlan, Michael J, Scott, Victoria E, Castle, Neil A, Daza, Anthony V, Milicic, Ivan, Sullivan, James P
Published in Bioorganic & medicinal chemistry letters (19.05.2003)
Published in Bioorganic & medicinal chemistry letters (19.05.2003)
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Journal Article
ARYLSULFONYLMETHYL OR ARYLSULFONAMIDE SUBSTITUTED AROMATIC COMPOUNDS SUITABLE FOR TREATING DISORDERS THAT RESPOND TO MODULATION OF THE DOPAMINE D3 RECEPTOR
DRESCHER KARLA, UNGER LILIANE, HAUPT ANDREAS, BRAJE WILFRIED, GRANDEL ROLAND, TURNER SEAN C, HENRY CHRISTOPHE
Year of Publication 20.03.2013
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Year of Publication 20.03.2013
Patent
Synthesis and Structure−Activity Relationships of a Novel Series of 2,3,5,6,7,9-Hexahydrothieno[3,2-b]quinolin-8(4H)-one 1,1-Dioxide KATP Channel Openers: Discovery of (−)-(9S)-9-(3-Bromo-4-fluorophenyl)-2,3,5,6,7,9- hexahydrothieno[3,2-b]quinolin-8(4H)-one 1,1-Dioxide (A-278637), a Potent KATP Opener That Selectively Inhibits Spontaneous Bladder Contractions
Carroll, William A, Altenbach, Robert J, Bai, Hao, Brioni, Jorge D, Brune, Michael E, Buckner, Steven A, Cassidy, Christopher, Chen, Yiyuan, Coghlan, Michael J, Daza, Anthony V, Drizin, Irene, Fey, Thomas A, Fitzgerald, Michael, Gopalakrishnan, Murali, Gregg, Robert J, Henry, Rodger F, Holladay, Mark W, King, Linda L, Kort, Michael E, Kym, Philip R, Milicic, Ivan, Tang, Rui, Turner, Sean C, Whiteaker, Kristi L, Yi, Lin, Zhang, Henry, Sullivan, James P
Published in Journal of medicinal chemistry (03.06.2004)
Published in Journal of medicinal chemistry (03.06.2004)
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Journal Article
MODULATORS OF 5-HT RECEPTORS AND METHODS OF USE THEREOF
NOEL S WILSON, ALAN F GASIECKI, ZHAO HONGYU, ANA-LUCIA RELO, CHRISTINA M THOMPSON, BRAJE WILFRIED, ALBERT W KRUGER, DENNIE S WELCH, TURNER SEAN C, LI HUANQIU, ZHANG MIN, IRINI AKRITOPOULOU-ZANZE, SHASHANK SHEKHAR, GANDARILLA JORGE, STEVAN W DJURIC
Year of Publication 14.01.2016
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Year of Publication 14.01.2016
Patent