The Hsp90 inhibitor IPI-504 rapidly lowers EML4-ALK levels and induces tumor regression in ALK-driven NSCLC models
NORMANT, E, PAEZ, G, PALOMBELLA, V. J, FRITZ, C. C, WEST, K. A, LIM, A. R, SLOCUM, K. L, TUNKEY, C, MCDOUGALL, J, WYLIE, A. A, ROBISON, K, CALIRI, K
Published in Oncogene (02.06.2011)
Published in Oncogene (02.06.2011)
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Quantitative analysis of gene regulation by seven clinically relevant progestins suggests a highly similar mechanism of action through progesterone receptors in T47D breast cancer cells
Bray, Jeffrey D., Jelinsky, Scott, Ghatge, Radhika, Bray, Jenifer A., Tunkey, Christopher, Saraf, Kathryn, Jacobsen, Britta M., Richer, Jennifer K., Brown, Eugene L., Winneker, Richard C., Horwitz, Kathryn B., Lyttle, C. Richard
Published in The Journal of steroid biochemistry and molecular biology (01.12.2005)
Published in The Journal of steroid biochemistry and molecular biology (01.12.2005)
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210 EML4-ALK is a sensitive client protein of Hsp90, and rearrangements of the ALK locus are associated with clinical response to IPI-504 (retaspimycin hydrochloride), a novel Hsp90 chaperone inhibitor, in patients with non-small cell lung cancer
Fritz, C, Lim, A, Slocum, K, Tunkey, C, Paez, G, West, K, Ross, R, Normant, E, Sequist, L, Palombella, V
Published in European journal of cancer supplements (2010)
Published in European journal of cancer supplements (2010)
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Global transcription profiling of estrogen activity: Estrogen receptor a regulates gene expression in the kidney
JELINSKY, Scott A, HARRIS, Heather A, BROWN, Eugene L, FLANAGAN, Kathryn, XIAOCHUN ZHANG, TUNKEY, Christopher, LAI, Kehdih, LANE, Malcolm V, SIMCOE, Donna K, EVANS, Mark J
Published in Endocrinology (Philadelphia) (01.02.2003)
Published in Endocrinology (Philadelphia) (01.02.2003)
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Safety and activity of IPI-504 (retaspimycin hydrochloride) and docetaxel in pretreated patients (pts) with metastatic non-small cell lung cancer (NSCLC)
Riely, G. J., Gettinger, S. N., Stoller, R. G., Gabrail, N. Y., Dy, G. K., Weiss, G. J., Tunkey, C., Skliris, G., Strychor, S., Dunbar, J., DeLucia, D., Ross, R. W., Gray, J. E.
Published in Journal of clinical oncology (20.05.2011)
Published in Journal of clinical oncology (20.05.2011)
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Exploiting genotypic differences to identify genes important for EAE development
Jelinsky, Scott A., Miyashiro, Joy S., Saraf, Kathryn A., Tunkey, Christopher, Reddy, Padma, Newcombe, Jia, Oestreicher, Judith L., Brown, Eugene, Trepicchio, William L., Leonard, John P., Marusic, Suzana
Published in Journal of the neurological sciences (15.12.2005)
Published in Journal of the neurological sciences (15.12.2005)
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