Design and synthesis of cell potent BACE-1 inhibitors: Structure–activity relationship of P1′ substituents
Sealy, Jennifer M., Truong, Anh P., Tso, Luke, Probst, Gary D., Aquino, Jose, Hom, Roy K., Jagodzinska, Barbara M., Dressen, Darren, Wone, David W.G., Brogley, Louis, John, Varghese, Tung, Jay S., Pleiss, Michael A., Tucker, John A., Konradi, Andrei W., Dappen, Michael S., Toth, Gergely, Pan, Hu, Ruslim, Lany, Miller, Jim, Bova, Michael P., Sinha, Sukanto, Quinn, Kevin P., Sauer, John-Michael
Published in Bioorganic & medicinal chemistry letters (15.11.2009)
Published in Bioorganic & medicinal chemistry letters (15.11.2009)
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Journal Article
A high throughput drug screening assay to identify compounds that promote oligodendrocyte differentiation using acutely dissociated and purified oligodendrocyte precursor cells
Lariosa-Willingham, Karen D, Rosler, Elen S, Tung, Jay S, Dugas, Jason C, Collins, Tassie L, Leonoudakis, Dmitri
Published in BMC research notes (05.09.2016)
Published in BMC research notes (05.09.2016)
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Journal Article
Development of a high throughput drug screening assay to identify compounds that protect oligodendrocyte viability and differentiation under inflammatory conditions
Lariosa-Willingham, Karen D, Rosler, Elen S, Tung, Jay S, Dugas, Jason C, Collins, Tassie L, Leonoudakis, Dmitri
Published in BMC research notes (05.09.2016)
Published in BMC research notes (05.09.2016)
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Journal Article
Design and Synthesis of Hydroxyethylene-Based Peptidomimetic Inhibitors of Human β-Secretase
Hom, Roy K, Gailunas, Andrea F, Mamo, Shumeye, Fang, Larry Y, Tung, Jay S, Walker, Donald E, Davis, David, Thorsett, Eugene D, Jewett, Nancy E, Moon, Joseph B, John, Varghese
Published in Journal of medicinal chemistry (01.01.2004)
Published in Journal of medicinal chemistry (01.01.2004)
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Journal Article
Design and synthesis of hydroxyethylamine (HEA) BACE-1 inhibitors: Prime side chromane-containing inhibitors
Ng, Raymond A., Sun, Minghua, Bowers, Simeon, Hom, Roy K., Probst, Gary D., John, Varghese, Fang, Lawrence Y., Maillard, Michel, Gailunas, Andrea, Brogley, Louis, Neitz, R. Jeffrey, Tung, Jay S., Pleiss, Michael A., Konradi, Andrei W., Sham, Hing L., Dappen, Michael S., Adler, Marc, Yao, Nanhua, Zmolek, Wes, Nakamura, David, Quinn, Kevin P., Sauer, John-Michael, Bova, Michael P., Ruslim, Lany, Artis, Dean R., Yednock, Ted A.
Published in Bioorganic & medicinal chemistry letters (15.08.2013)
Published in Bioorganic & medicinal chemistry letters (15.08.2013)
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Journal Article
Design of Substrate-Based Inhibitors of Human β-Secretase
Tung, Jay S, Davis, David L, Anderson, John P, Walker, Don E, Mamo, Shumeye, Jewett, Nancy, Hom, Roy K, Sinha, Sukanto, Thorsett, Eugene D, John, Varghese
Published in Journal of medicinal chemistry (17.01.2002)
Published in Journal of medicinal chemistry (17.01.2002)
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Journal Article
Preparation and Optimization of a Series of 3-Carboxamido-5-phenacylaminopyrazole Bradykinin B1 Receptor Antagonists
Dressen, Darren, Garofalo, Albert W, Hawkinson, Jon, Hom, Dennis, Jagodzinski, Jacek, Marugg, Jennifer L, Neitzel, Martin L, Pleiss, Michael A, Szoke, Balazs, Tung, Jay S, Wone, David W. G, Wu, Jing, Zhang, Heather
Published in Journal of medicinal chemistry (18.10.2007)
Published in Journal of medicinal chemistry (18.10.2007)
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Journal Article
Improving the permeability of the hydroxyethylamine BACE-1 inhibitors: Structure–activity relationship of P2′ substituents
Truong, Anh P., Probst, Gary D., Aquino, Jose, Fang, Larry, Brogley, Louis, Sealy, Jennifer M., Hom, Roy K., Tucker, John A., John, Varghese, Tung, Jay S., Pleiss, Michael A., Konradi, Andrei W., Sham, Hing L., Dappen, Michael S., Tóth, Gergley, Yao, Nanhua, Brecht, Eric, Pan, Hu, Artis, Dean R., Ruslim, Lany, Bova, Michael P., Sinha, Sukanto, Yednock, Ted A., Zmolek, Wes, Quinn, Kevin P., Sauer, John-Michael
Published in Bioorganic & medicinal chemistry letters (15.08.2010)
Published in Bioorganic & medicinal chemistry letters (15.08.2010)
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Journal Article
Design and synthesis of hydroxyethylamine (HEA) BACE-1 inhibitors: Structure–activity relationship of the aryl region
Probst, Gary D., Bowers, Simeon, Sealy, Jennifer M., Stupi, Brian, Dressen, Darren, Jagodzinska, Barbara M., Aquino, Jose, Gailunas, Andrea, Truong, Anh P., Tso, Luke, Xu, Ying-Zi, Hom, Roy K., John, Varghese, Tung, Jay S., Pleiss, Michael A., Tucker, John A., Konradi, Andrei W., Sham, Hing L., Jagodzinski, Jacek, Toth, Gergely, Brecht, Eric, Yao, Nanhua, Pan, Hu, Lin, May, Artis, Dean R., Ruslim, Lany, Bova, Michael P., Sinha, Sukanto, Yednock, Ted A., Gauby, Shawn, Zmolek, Wes, Quinn, Kevin P., Sauer, John-Michael
Published in Bioorganic & medicinal chemistry letters (15.10.2010)
Published in Bioorganic & medicinal chemistry letters (15.10.2010)
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Journal Article
Design and Synthesis of Statine-Based Cell-Permeable Peptidomimetic Inhibitors of Human β-Secretase
Hom, Roy K, Fang, Larry Y, Mamo, Shumeye, Tung, Jay S, Guinn, Ashley C, Walker, Don E, Davis, David L, Gailunas, Andrea F, Thorsett, Eugene D, Sinha, Sukanto, Knops, Jeroen E, Jewett, Nancy E, Anderson, John P, John, Varghese
Published in Journal of medicinal chemistry (08.05.2003)
Published in Journal of medicinal chemistry (08.05.2003)
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Journal Article
Stereochemical Analysis of the Reaction Catalyzed by Yeast Protein Farnesyltransferase
Edelstein, Rebecca L, Weller, Valerie A, Distefano, Mark D, Tung, Jay S
Published in Journal of organic chemistry (07.08.1998)
Published in Journal of organic chemistry (07.08.1998)
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Journal Article
Characterization of Caspase Processing and Activation in HL-60 Cell Cytosol Under Cell-free Conditions
Mesner, Peter W., Bible, Keith C., Martins, Luis M., Kottke, Timothy J., Srinivasula, Srinivasa M., Svingen, Phyllis A., Chilcote, Tamie J., Basi, Guriq S., Tung, Jay S., Krajewski, Stan, Reed, John C., Alnemri, Emad S., Earnshaw, William C., Kaufmann, Scott H.
Published in The Journal of biological chemistry (06.08.1999)
Published in The Journal of biological chemistry (06.08.1999)
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Journal Article
Comparison of Apoptosis in Wild-Type and Fas-Resistant Cells: Chemotherapy-Induced Apoptosis Is Not Dependent on Fas/Fas Ligand Interactions
Eischen, Christine M., Kottke, Timothy J., Martins, Luis M., Basi, Guriqbal S., Tung, Jay S., Earnshaw, William C., Leibson, Paul J., Kaufmann, Scott H.
Published in Blood (01.08.1997)
Published in Blood (01.08.1997)
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A high-yield modification of the Pschorr phenanthrene synthesis
Duclos, Richard I, Tung, Jay S, Rapoport, Henry
Published in Journal of organic chemistry (01.12.1984)
Published in Journal of organic chemistry (01.12.1984)
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Journal Article
Activation of Multiple Interleukin-1β Converting Enzyme Homologues in Cytosol and Nuclei of HL-60 Cells during Etoposide-induced Apoptosis
Martins, Luis M., Kottke, Timothy, Mesner, Peter W., Basi, Guriqbal S., Sinha, Sukanto, Frigon, Normand, Tatar, Eric, Tung, Jay S., Bryant, Karin, Takahashi, Atsushi, Svingen, Phyllis A., Madden, Benjamin J., McCormick, Daniel J., Earnshaw, William C., Kaufmann, Scott H.
Published in The Journal of biological chemistry (14.03.1997)
Published in The Journal of biological chemistry (14.03.1997)
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Journal Article
Comparison of Caspase Activation and Subcellular Localization in HL-60 and K562 Cells Undergoing Etoposide-Induced Apoptosis
Martins, Luis M., Mesner, Peter W., Kottke, Timothy J., Basi, Guriqbal S., Sinha, Sukanto, Tung, Jay S., Svingen, Phyllis A., Madden, Benjamin J., Takahashi, Atsushi, McCormick, Daniel J., Earnshaw, William C., Kaufmann, Scott H.
Published in Blood (01.12.1997)
Published in Blood (01.12.1997)
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Journal Article
Characterization of caspase processing and activation in HL-60 cell cytosol under cell-free conditions. Nucleotide requirement and inhibitor profile
Mesner, Jr, P W, Bible, K C, Martins, L M, Kottke, T J, Srinivasula, S M, Svingen, P A, Chilcote, T J, Basi, G S, Tung, J S, Krajewski, S, Reed, J C, Alnemri, E S, Earnshaw, W C, Kaufmann, S H
Published in The Journal of biological chemistry (06.08.1999)
Published in The Journal of biological chemistry (06.08.1999)
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Journal Article
Methods and Compositions for the Treatment of Demyelinating Disorders
Dugas, Jason, Rosler, Elen, Tung, Jay S, Lariosa-Willingham, Karen, Leonoudakis, Dmitri, Collins, Tassie
Year of Publication 02.05.2019
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Year of Publication 02.05.2019
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