Discovery of pyrido[2,3-d]pyrimidine-based inhibitors of HCV NS5A
DeGoey, David A., Betebenner, David A., Grampovnik, David J., Liu, Dachun, Pratt, John K., Tufano, Michael D., He, Wenping, Krishnan, Preethi, Pilot-Matias, Tami J., Marsh, Kennan C., Molla, Akhteruzzaman, Kempf, Dale J., Maring, Clarence J.
Published in Bioorganic & medicinal chemistry letters (15.06.2013)
Published in Bioorganic & medicinal chemistry letters (15.06.2013)
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Synthesis and Biological Characterization of Aryl Uracil Inhibitors of Hepatitis C Virus NS5B Polymerase: Discovery of ABT-072, a trans-Stilbene Analog with Good Oral Bioavailability
Randolph, John T, Krueger, A. Chris, Donner, Pamela L, Pratt, John K, Liu, Dachun, Motter, Christopher E, Rockway, Todd W, Tufano, Michael D, Wagner, Rolf, Lim, Hock B, Beyer, Jill M, Mondal, Rubina, Panchal, Neeta S, Colletti, Lynn, Liu, Yaya, Koev, Gennadiy, Kati, Warren M, Hernandez, Lisa E, Beno, David W. A, Longenecker, Kenton L, Stewart, Kent D, Dumas, Emily O, Molla, Akhteruzzaman, Maring, Clarence J
Published in Journal of medicinal chemistry (08.02.2018)
Published in Journal of medicinal chemistry (08.02.2018)
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Novel Hepatitis C virus replicon inhibitors: Synthesis and structure–activity relationships of fused pyrimidine derivatives
Chris Krueger, A., Madigan, Darold L., Beno, David W., Betebenner, David A., Carrick, Robert, Green, Brian E., He, Wenping, Liu, Dachun, Maring, Clarence J., McDaniel, Keith F., Mo, Hongmei, Molla, Akhteruzzaman, Motter, Christopher E., Pilot-Matias, Tami J., Tufano, Michael D., Kempf, Dale J.
Published in Bioorganic & medicinal chemistry letters (15.03.2012)
Published in Bioorganic & medicinal chemistry letters (15.03.2012)
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ANTI-VIRAL COMPOUNDS
ALLAN C KRUEGER, BETEBENNER DAVID A, HUTCHINSON DOUGLAS K, ROCKWAY TODD W, JEAN C CALIFANO, FLENTGE CHARLES A, CHARLES W HUTCHINS, SARRIS KATHY, GAO YI, DEGOEY DAVID A, KATI WARREN M, KEDDY RYAN G, MATULENKO MARK A, TAMMIE K JINKERSON, MARING CLARENCE J, DONNER PAMELA L, PRATT JOHN K, NELSON LISSA T, WAGNER ROLF, SACHIN V PATEL, WAGAW SABLE H, RANDOLPH JOHN T, TUFANO MICHAEL D, WILLIAM A CARROLL, MOTTER CHRISTOPHER E, LIU DACHUN, DANIEL D CASPI, LI WENKE, BELLIZZI MARY E, KEVIN R WOLLER
Year of Publication 04.03.2021
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Year of Publication 04.03.2021
Patent
ANTI-VIRAL COMPOUNDS
ALLAN C KRUEGER, BETEBENNER DAVID A, HUTCHINSON DOUGLAS K, ROCKWAY TODD W, JEAN C CALIFANO, FLENTGE CHARLES A, CHARLES W HUTCHINS, SARRIS KATHY, GAO YI, DEGOEY DAVID A, KATI WARREN M, KEDDY RYAN G, MATULENKO MARK A, TAMMIE K JINKERSON, MARING CLARENCE J, DONNER PAMELA L, PRATT JOHN K, NELSON LISSA T, WAGNER ROLF, SACHIN V PATEL, WAGAW SABLE H, RANDOLPH JOHN T, TUFANO MICHAEL D, WILLIAM A CARROLL, MOTTER CHRISTOPHER E, LIU DACHUN, DANIEL D CASPI, LI WENKE, BELLIZZI MARY E, KEVIN R WOLLER
Year of Publication 16.04.2020
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Year of Publication 16.04.2020
Patent
ANTI-VIRAL COMPOUNDS FOR TREATING HCV INFECTION
ALLAN C KRUEGER, BETEBENNER DAVID A, HUTCHINSON DOUGLAS K, ROCKWAY TODD W, JEAN C CALIFANO, FLENTGE CHARLES A, CHARLES W HUTCHINS, SARRIS KATHY, GAO YI, DEGOEY DAVID A, KATI WARREN M, KEDDY RYAN G, MATULENKO MARK A, TAMMIE K JINKERSON, MARING CLARENCE J, DONNER PAMELA L, PRATT JOHN K, NELSON LISSA T, WAGNER ROLF, SACHIN V PATEL, WAGAW SABLE H, RANDOLPH JOHN T, TUFANO MICHAEL D, MOTTER CHRISTOPHER E, LIU DACHUN, DANIEL D CASPI, LI WENKE, BELLIZZI MARY E, KEVIN R WOLLER
Year of Publication 07.11.2019
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Year of Publication 07.11.2019
Patent
ANTI-VIRUS COMPOUND
ALLAN C KRUEGER, BETEBENNER DAVID A, HUTCHINSON DOUGLAS K, ROCKWAY TODD W, JEAN C CALIFANO, FLENTGE CHARLES A, CHARLES W HUTCHINS, SARRIS KATHY, GAO YI, DEGOEY DAVID A, KATI WARREN M, KEDDY RYAN G, MATULENKO MARK A, TAMMIE K JINKERSON, MARING CLARENCE J, DONNER PAMELA L, PRATT JOHN K, NELSON LISSA T, WAGNER ROLF, SACHIN V PATEL, WAGAW SABLE H, RANDOLPH JOHN T, TUFANO MICHAEL D, WILLIAM A CARROLL, MOTTER CHRISTOPHER E, LIU DACHUN, DANIEL D CASPI, LI WENKE, BELLIZZI MARY E, KEVIN R WOLLER
Year of Publication 26.04.2018
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Year of Publication 26.04.2018
Patent
ANTI-VIRAL COMPOUNDS
HUTCHINS CHARLES W, WOLLER KEVIN R, WAGAW SEBEL H, BETEBENNER DAVID A, HUTCHINSON DOUGLAS K, ROCKWAY TODD W, FLENTGE CHARLES A, JINKERSON TAMMIE K, SARRIS KATHY, GAO YI, DEGOEY DAVID A, KATI WARREN M, KEDDY RYAN G, MATULENKO MARK A, CALIFANO JEAN C, CASPI DANIEL D, MARING CLARENCE J, DONNER PAMELA L, PRATT JOHN K, NELSON LISSA T, WAGNER ROLF, RANDOLPH JOHN T, CARROLL WILLIAM A, TUFANO MICHAEL D, KRUEGER ALLAN C, MOTTER CHRISTOPHER E, LIU DACHUN, PATEL SACHEL V, LI WENKE, BELLIZZI MARY E
Year of Publication 13.03.2018
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Year of Publication 13.03.2018
Patent
ANTI-VIRAL COMPOUNDS TO TREAT HCV INFECTION
ALLAN C KRUEGER, BETEBENNER DAVID A, HUTCHINSON DOUGLAS K, ROCKWAY TODD W, JEAN C CALIFANO, FLENTGE CHARLES A, CHARLES W HUTCHINS, SARRIS KATHY, GAO YI, DEGOEY DAVID A, KATI WARREN M, KEDDY RYAN G, MATULENKO MARK A, TAMMIE K JINKERSON, MARING CLARENCE J, DONNER PAMELA L, PRATT JOHN K, NELSON LISSA T, WAGNER ROLF, SACHIN V PATEL, WAGAW SABLE H, RANDOLPH JOHN T, TUFANO MICHAEL D, MOTTER CHRISTOPHER E, LIU DACHUN, DANIEL D CASPI, LI WENKE, BELLIZZI MARY E, KEVIN R WOLLER
Year of Publication 28.09.2017
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Year of Publication 28.09.2017
Patent
ANTI-VIRAL COMPOUNDS FOR TREATING HCV INFECTION
ALLAN C KRUEGER, BETEBENNER DAVID A, HUTCHINSON DOUGLAS K, ROCKWAY TODD W, JEAN C CALIFANO, FLENTGE CHARLES A, CHARLES W HUTCHINS, SARRIS KATHY, GAO YI, DEGOEY DAVID A, KATI WARREN M, KEDDY RYAN G, MATULENKO MARK A, TAMMIE K JINKERSON, MARING CLARENCE J, DONNER PAMELA L, PRATT JOHN K, NELSON LISSA T, WAGNER ROLF, SACHIN V PATEL, WAGAW SABLE H, RANDOLPH JOHN T, TUFANO MICHAEL D, MOTTER CHRISTOPHER E, LIU DACHUN, DANIEL D CASPI, LI WENKE, BELLIZZI MARY E, KEVIN R WOLLER
Year of Publication 14.07.2016
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Year of Publication 14.07.2016
Patent
ANTI-VIRUS COMPOUND
ALLAN C KRUEGER, BETEBENNER DAVID A, HUTCHINSON DOUGLAS K, ROCKWAY TODD W, JEAN C CALIFANO, FLENTGE CHARLES A, CHARLES W HUTCHINS, SARRIS KATHY, GAO YI, DEGOEY DAVID A, KATI WARREN M, KEDDY RYAN G, MATULENKO MARK A, TAMMIE K JINKERSON, MARING CLARENCE J, DONNER PAMELA L, PRATT JOHN K, NELSON LISSA T, WAGNER ROLF, SACHIN V PATEL, WAGAW SABLE H, RANDOLPH JOHN T, TUFANO MICHAEL D, WILLIAM A CARROLL, MOTTER CHRISTOPHER E, LIU DACHUN, DANIEL D CASPI, LI WENKE, BELLIZZI MARY E, KEVIN R WOLLER
Year of Publication 16.06.2016
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Year of Publication 16.06.2016
Patent
ANTIVIRAL COMPOUNDS AND USES THEREOF
WAGNER ROLF, ALLAN C KRUEGER, BETEBENNER DAVID A, HUTCHINSON DOUGLAS K, ROCKWAY TODD W, FLENTGE CHARLES A, RANDOLPH JOHN T, TUFANO MICHAEL D, LIU DACHUN, DEGOEY DAVID A, KATI WARREN M, KENTON L LONGENECKER, MARING CLARENCE J, PRATT JOHN K, DONNER PAMELA L
Year of Publication 29.01.2015
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Year of Publication 29.01.2015
Patent
URACIL OR THYMINE DERIVATIVE FOR TREATING HEPATITIS C
HENRY RODGER F, LIU YAYA, LOU XIAOCHUN, BETEBENNER DAVID A, HUTCHINSON DOUGLAS K, FRANCZYK II THADDEUS S, ROCKWAY TODD W, HUANG PEGGY P, FLENTGE CHARLES A, SARRIS KATHY, GAO YI, DEGOEY DAVID A, KATI WARREN M, MARING CLARENCE J, BARNES DAVID M, PRATT JOHN K, DONNER PAMELA L, CHEN SHUANG, WAGNER ROLF, HENGEVELD JOHN E, RANDOLPH JOHN T, TUFANO MICHAEL D, LONGENECKER KENTON L, MOTTER CHRISTOPHER E, LIU DACHUN, KRUEGER ALLAN C, KOTECKI BRIAN J, HAIGHT ANTHONY R, ZHANG GEOFF G. Z, STEWART KENT D
Year of Publication 20.10.2015
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Year of Publication 20.10.2015
Patent
ANTI-VIRAL COMPOUNDS
HUTCHINS CHARLES W, WOLLER KEVIN R, WAGAW SEBEL H, BETEBENNER DAVID A, HUTCHINSON DOUGLAS K, ROCKWAY TODD W, FLENTGE CHARLES A, JINKERSON TAMMIE K, SARRIS KATHY, GAO YI, DEGOEY DAVID A, KATI WARREN M, KEDDY RYAN G, MATULENKO MARK A, CALIFANO JEAN C, CASPI DANIEL D, MARING CLARENCE J, DONNER PAMELA L, PRATT JOHN K, NELSON LISSA T, WAGNER ROLF, RANDOLPH JOHN T, CARROLL WILLIAM A, TUFANO MICHAEL D, KRUEGER ALLAN C, MOTTER CHRISTOPHER E, LIU DACHUN, PATEL SACHEL V, LI WENKE, BELLIZZI MARY E
Year of Publication 15.12.2014
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Year of Publication 15.12.2014
Patent
ANTI-VIRAL COMPOUNDS TO TREAT HCV INFECTION
HUTCHINS CHARLES W, WOLLER KEVIN R, BETEBENNER DAVID A, HUTCHINSON DOUGLAS K, ROCKWAY TODD W, FLENTGE CHARLES A, PATEL SACHIN V, JINKERSON TAMMIE K, SARRIS KATHY, GAO YI, DEGOEY DAVID A, KATI WARREN M, KEDDY RYAN G, MATULENKO MARK A, CALIFANO JEAN C, CASPI DANIEL D, MARING CLARENCE J, DONNER PAMELA L, PRATT JOHN K, NELSON LISSA T, WAGNER ROLF, RANDOLPH JOHN T, TUFANO MICHAEL D, KRUEGER ALLAN C, MOTTER CHRISTOPHER E, LIU DACHUN, WAGAW SEBLE H, LI WENKE, BELLIZZI MARY E
Year of Publication 27.03.2014
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Year of Publication 27.03.2014
Patent
ANTI-VIRAL COMPOUNDS
HUTCHINS CHARLES W, WOLLER KEVIN R, WAGAW SEBEL H, BETEBENNER DAVID A, HUTCHINSON DOUGLAS K, ROCKWAY TODD W, FLENTGE CHARLES A, JINKERSON TAMMIE K, SARRIS KATHY, GAO YI, DEGOEY DAVID A, KATI WARREN M, KEDDY RYAN G, MATULENKO MARK A, CALIFANO JEAN C, CASPI DANIEL D, MARING CLARENCE J, DONNER PAMELA L, PRATT JOHN K, NELSON LISSA T, WAGNER ROLF, RANDOLPH JOHN T, CARROLL WILLIAM A, TUFANO MICHAEL D, KRUEGER ALLAN C, MOTTER CHRISTOPHER E, LIU DACHUN, PATEL SACHEL V, LI WENKE, BELLIZZI MARY E
Year of Publication 14.03.2014
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Year of Publication 14.03.2014
Patent
ANTI-VIRAL COMPOUNDS TO TREAT HCV INFECTION
HUTCHINS CHARLES W, WOLLER KEVIN R, BETEBENNER DAVID A, HUTCHINSON DOUGLAS K, ROCKWAY TODD W, FLENTGE CHARLES A, PATEL SACHIN V, JINKERSON TAMMIE K, SARRIS KATHY, GAO YI, DEGOEY DAVID A, KATI WARREN M, KEDDY RYAN G, MATULENKO MARK A, CALIFANO JEAN C, CASPI DANIEL D, MARING CLARENCE J, DONNER PAMELA L, PRATT JOHN K, NELSON LISSA T, WAGNER ROLF, RANDOLPH JOHN T, TUFANO MICHAEL D, KRUEGER ALLAN C, MOTTER CHRISTOPHER E, LIU DACHUN, WAGAW SEBLE H, LI WENKE, BELLIZZI MARY E
Year of Publication 24.10.2012
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Year of Publication 24.10.2012
Patent