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Published in Journal of medicinal chemistry (14.11.2013)
Published in Journal of medicinal chemistry (14.11.2013)
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Synthesis and biological evaluation of novel orally available 1-phenyl-6-aminouracils containing dimethyldihydrobenzofuranol structure for the treatment of allergic skin diseases
Tobe, Masanori, Tsuboi, Katsunori, Hasegawa, Futoshi, Fujiwara, Norio, Inoue, Yoshifumi, Isobe, Masakazu, Isobe, Yoshiaki
Published in Bioorganic & medicinal chemistry letters (15.02.2016)
Published in Bioorganic & medicinal chemistry letters (15.02.2016)
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DAGLβ inhibition perturbs a lipid network involved in macrophage inflammatory responses
Hsu, Ku-Lung, Tsuboi, Katsunori, Adibekian, Alexander, Pugh, Holly, Masuda, Kim, Cravatt, Benjamin F
Published in Nature chemical biology (01.12.2012)
Published in Nature chemical biology (01.12.2012)
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Discovery of N-(6-(5-fluoro-2-(piperidin-1-yl)phenyl)pyridazin-3-yl)-1-(tetrahydro-2H-pyran-4-yl)methanesulfonamide as a brain-permeable and metabolically stable kynurenine monooxygenase inhibitor
Tsuboi, Katsunori, Kimura, Hidenori, Nakatsuji, Yoshie, Kassai, Momoe, Deai, Yoko, Isobe, Yoshiaki
Published in Bioorganic & medicinal chemistry letters (15.07.2021)
Published in Bioorganic & medicinal chemistry letters (15.07.2021)
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Discovery and Optimization of Piperidyl-1,2,3-Triazole Ureas as Potent, Selective, and in Vivo-Active Inhibitors of α/β-Hydrolase Domain Containing 6 (ABHD6)
Hsu, Ku-Lung, Tsuboi, Katsunori, Chang, Jae Won, Whitby, Landon R, Speers, Anna E, Pugh, Holly, Cravatt, Benjamin F
Published in Journal of medicinal chemistry (14.11.2013)
Published in Journal of medicinal chemistry (14.11.2013)
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Potent and Selective Inhibitors of Glutathione S-Transferase Omega 1 That Impair Cancer Drug Resistance
Tsuboi, Katsunori, Bachovchin, Daniel A, Speers, Anna E, Spicer, Timothy P, Fernandez-Vega, Virneliz, Hodder, Peter, Rosen, Hugh, Cravatt, Benjamin F
Published in Journal of the American Chemical Society (19.10.2011)
Published in Journal of the American Chemical Society (19.10.2011)
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STEREOCHEMISTRY OF AN ALLYL CYANATE-TO-ISOCYANATE REARRANGEMENT
ICHIKAWA, Y, TSUBOI, K, ISOBE, M
Published in Journal of the Chemical Society, Perkin Transactions 1 (1994)
Published in Journal of the Chemical Society, Perkin Transactions 1 (1994)
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Confirming Target Engagement for Reversible Inhibitors in Vivo by Kinetically Tuned Activity-Based Probes
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Published in Journal of the American Chemical Society (27.06.2012)
Published in Journal of the American Chemical Society (27.06.2012)
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LOAD MEASUREMENT UNIT AND LOAD MEASUREMENT METHOD
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Year of Publication 06.06.2019
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Year of Publication 06.06.2019
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3-(ARYL OR HETEROARYL) METHYLENEINDOLIN-2-ONE DERIVATIVES AS INHIBITORS OF CANCER STEM CELL PATHWAY KINASES FOR TREATMENT OF CANCER
LIU JI-FENG, AMANDA GIBEAU, HARRY ROGOFF, TOJO SHINGO, LEE WAI, KANAI TOSHIO, CHIANG J LI, TAKANASHI YOSUKE, KUBOTA KATSUMI, TSUBOI KATSUNORI, KODAMA TOMOHIRO
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Year of Publication 01.11.2018
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NOVEL BICYCLIC HETEROCYCLIC COMPOUND
TSUBOI, KATSUNORI, KINOSHITA, HIRONORI, YAMAI, YUSUKE, WATANABE, HITOSHI
Year of Publication 01.07.2010
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Year of Publication 01.07.2010
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3-(ARYL OR HETEROARYL)METHYLENEINDOLIN-2-ONE DERIVATIVES AS INHIBITORS OF CANCER STEM CELL PATHWAY KINASES FOR THE TREATMENT OF CANCER
ROGOFF HARRY, LIU JI FENG, TOJO SHINGO, KANAI TOSHIO, LI CHIANG J, LI WEI, TAKANASHI YOSUKE, KUBOTA KATSUMI, TSUBOI KATSUNORI, GIBEAU AMANDA, KODAMA TOMOHIRO
Year of Publication 16.11.2015
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Year of Publication 16.11.2015
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