Tyr115 is the key residue for determining agonist selectivity in the V1a vasopressin receptor
Chini, B., Mouillac, B., Ala, Y., Balestre, M.N., Trumpp-Kallmeyer, S., Hoflack, J., Elands, J., Hibert, M., Manning, M., Jard, S.
Published in The EMBO journal (01.05.1995)
Published in The EMBO journal (01.05.1995)
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Journal Article
Pyrido[2,3-d]pyrimidin-7-one Inhibitors of Cyclin-Dependent Kinases
Barvian, Mark, Boschelli, Diane H, Cossrow, Jennifer, Dobrusin, Ellen, Fattaey, Ali, Fritsch, Alex, Fry, David, Harvey, Patricia, Keller, Paul, Garrett, Michelle, La, Frances, Leopold, Wilbur, McNamara, Dennis, Quin, Maire, Trumpp-Kallmeyer, Susanne, Toogood, Peter, Wu, Zhipei, Zhang, Erli
Published in Journal of medicinal chemistry (30.11.2000)
Published in Journal of medicinal chemistry (30.11.2000)
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Journal Article
Three-dimensional models of neurotransmitter G-binding protein-coupled receptors
Hibert, M F, Trumpp-Kallmeyer, S, Bruinvels, A, Hoflack, J
Published in Molecular pharmacology (01.07.1991)
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Published in Molecular pharmacology (01.07.1991)
Journal Article
Identification of a Single Residue Responsible for Agonist Selectivity in the Oxytocin-Vasopressin Receptors
CHINI, B., MOUILLAC, B., ALA, Y., BALESTRE, M. N., TRUMPP-KALLMEYER, S., HOFLACK, J., ELANDS, J., HIBERT, M., MANNING, M., JARD, S., BARBERIS, C.
Published in Annals of the New York Academy of Sciences (01.05.1997)
Published in Annals of the New York Academy of Sciences (01.05.1997)
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Journal Article
Tyr115 is the key residue for determining agonist selectivity in the V1a vasopressin receptor
Chini, B., Mouillac, B., Ala, Y., Balestre, M.N., Trumpp‐Kallmeyer, S., Hoflack, J., Elands, J., Hibert, M., Manning, M., Jard, S.
Published in The EMBO journal (15.05.1995)
Published in The EMBO journal (15.05.1995)
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Journal Article
Functional architecture of vasopressin/oxytocin receptors
Hibert, M, Hoflack, J, Trumpp-Kallmeyer, S, Mouillac, B, Chini, B, Mahé, E, Cotte, N, Jard, S, Manning, M, Barberis, C
Published in Journal of receptors and signal transduction (01.01.1999)
Published in Journal of receptors and signal transduction (01.01.1999)
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Journal Article
3D MODELS OF HORMONE RECEPTORS : EXPERIMENTAL VALIDATION
HIBERT, Marcel, HOFLACK, Jan, TRUMPP-KALLMEYER, Suzanne, PAQUET, Jean-Luc, LEPPIK, Raymond, BARBERIS, Claude, Mouillac, Bernard, CHINI, Bice, JARD, Serge
Published in European journal of medicinal chemistry (1995)
Published in European journal of medicinal chemistry (1995)
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Journal Article
Conference Proceeding
Specific, Irreversible Inactivation of the Epidermal Growth Factor Receptor and erbB2, by a New Class of Tyrosine Kinase Inhibitor
Fry, David W., Bridges, Alexander J., Denny, William A., Doherty, Annette, Greis, Kenneth D., Hicks, James L., Hook, Kenneth E., Keller, Paul R., Leopold, Wilbur R., Loo, Joseph A., McNamara, Dennis J., Nelson, James M., Sherwood, Veronika, Smaill, Jeff B., Trumpp-Kallmeyer, Susanne, Dobrusin, Ellen M.
Published in Proceedings of the National Academy of Sciences - PNAS (29.09.1998)
Published in Proceedings of the National Academy of Sciences - PNAS (29.09.1998)
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Journal Article
Three-dimensional models of gonado-thyrotropin hormone receptor transmembrane domain
Hoflack, J, Hibert, M F, Trumpp-Kallmeyer, S, Bidart, J M
Published in Drug design and discovery (01.06.1993)
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Published in Drug design and discovery (01.06.1993)
Journal Article
G-Protein Coupled Receptors: Models, Mutagenesis, and Drug Design
Bikker, Jack Andrew, Trumpp-Kallmeyer, Susanne, Humblet, Christine
Published in Journal of medicinal chemistry (30.07.1998)
Published in Journal of medicinal chemistry (30.07.1998)
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Journal Article
The binding site of neuropeptide vasopressin V1a receptor. Evidence for a major localization within transmembrane regions
Mouillac, B, Chini, B, Balestre, M N, Elands, J, Trumpp-Kallmeyer, S, Hoflack, J, Hibert, M, Jard, S, Barberis, C
Published in The Journal of biological chemistry (27.10.1995)
Published in The Journal of biological chemistry (27.10.1995)
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Journal Article
Design and synthesis of potent, orally active, inhibitors of carboxypeptidase U (TAFIa)
POLLA, Magnus O, TOTTIE, Louise, SANDBERG, Marcel, THURMOND, John, PENG YU, HATEGAN, Georgeta, ANDERSON, Herb, NORDEN, Carita, LINSCHOTEN, Marcel, MÜSIL, Djordje, TRUMPP-KALLMEYER, Susanne, AUKRUST, Inger R, RINGOM, Rune, HOLM, Kjetil H, NESET, Siren M
Published in Bioorganic & medicinal chemistry (01.03.2004)
Published in Bioorganic & medicinal chemistry (01.03.2004)
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Journal Article
Tyrosine Kinase Inhibitors. 11. Soluble Analogues of Pyrrolo- and Pyrazoloquinazolines as Epidermal Growth Factor Receptor Inhibitors: Synthesis, Biological Evaluation, and Modeling of the Mode of Binding
Palmer, Brian D, Trumpp-Kallmeyer, Susanne, Fry, David W, Nelson, James M, Showalter, H. D. Hollis, Denny, William A
Published in Journal of medicinal chemistry (09.05.1997)
Published in Journal of medicinal chemistry (09.05.1997)
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Journal Article
Development of a Binding Model to Protein Tyrosine Kinases for Substituted Pyrido[2,3-d]pyrimidine Inhibitors
Trumpp-Kallmeyer, Susanne, Rubin, J. Ronald, Humblet, Christine, Hamby, James M, Hollis Showalter, H. D
Published in Journal of medicinal chemistry (21.05.1998)
Published in Journal of medicinal chemistry (21.05.1998)
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Journal Article
Two aromatic residues regulate the response of the human oxytocin receptor to the partial agonist arginine vasopressin
Chini, Bice, Mouillac, Bernard, Balestre, Marie-Nöelle, Trumpp-Kallmeyer, Susanne, Hoflack, Jan, Hibert, Marcel, Andriolo, Maria, Pupier, Sandrine, Jard, Serge, Barberis, Claude
Published in FEBS letters (18.11.1996)
Published in FEBS letters (18.11.1996)
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Journal Article
Site-directed mutagenesis of the putative human muscarinic M 2 receptor binding site
Heitz, Freddy, Holzwarth, James A, Gies, Jean-Pierre, Pruss, Rebecca M, Trumpp-Kallmeyer, Suzanne, Hibert, Marcel F, Guenet, Chantal
Published in European journal of pharmacology (10.09.1999)
Published in European journal of pharmacology (10.09.1999)
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Journal Article
Site-directed mutagenesis of the putative human muscarinic M2 receptor binding site
Heitz, F, Holzwarth, J A, Gies, J P, Pruss, R M, Trumpp-Kallmeyer, S, Hibert, M F, Guenet, C
Published in European journal of pharmacology (10.09.1999)
Published in European journal of pharmacology (10.09.1999)
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Journal Article
This is not a G protein-coupled receptor
Hibert, Marcel F., Trumpp-Kallmeyer, Susanne, Hoflack, Jan, Bruinvels, Anne
Published in Trends in Pharmacological Sciences (1993)
Published in Trends in Pharmacological Sciences (1993)
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Book Review
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