Pharmacological characterization of the human vasopressin receptor subtypes stably expressed in Chinese hamster ovary cells
Tahara, Atsuo, Saito, Masayuki, Sugimoto, Toru, Tomura, Yuichi, Wada, Koh‐ichi, Kusayama, Toshiyuki, Tsukada, Junko, Ishii, Noe, Yatsu, Takeyuki, Uchida, Wataru, Tanaka, Akihiro
Published in British journal of pharmacology (01.12.1998)
Published in British journal of pharmacology (01.12.1998)
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Preparation of Highly Potent and Selective Non-Peptide Antagonists of the Arginine Vasopressin V1A Receptor by Introduction of a 2-Ethyl-1H-1-imidazolyl Group
Shimada, Yoshiaki, Akane, Hiroaki, Taniguchi, Nobuaki, Matsuhisa, Akira, Kawano, Noriyuki, Kikuchi, Kazumi, Yatsu, Takeyuki, Tahara, Atsuo, Tomura, Yuichi, Kusayama, Toshiyuki, Wada, Koh-ichi, Tsukada, Junko, Tsunoda, Takashi, Tanaka, Akihiro
Published in Chemical & pharmaceutical bulletin (01.07.2005)
Published in Chemical & pharmaceutical bulletin (01.07.2005)
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Antihypertensive activity of a nonpeptide angiotensin II receptor antagonist, YM358, in rats and dogs
Shibasaki, Masayuki, Fujimori, Akira, Kusayama, Toshiyuki, Tokioka, Tomoko, Satoh, Yasuko, Okazaki, Toshio, Uchida, Wataru, Inagaki, Osamu, Yanagisawa, Isao
Published in European journal of pharmacology (24.09.1997)
Published in European journal of pharmacology (24.09.1997)
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Pharmacological profile of YM358, a novel nonpeptide angiotensin AT1 receptor antagonist
Shibasaki, Masayuki, Fujimori, Akira, Takanashi, Masahiro, Kusayama, Toshiyuki, Tokioka, Tomoko, Satoh, Yasuko, Okazaki, Toshio, Uchida, Wataru, Inagaki, Osamu, Yanagisawa, Isao
Published in European journal of pharmacology (24.09.1997)
Published in European journal of pharmacology (24.09.1997)
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Abstract A76: MDV3100, a novel androgen receptor signaling inhibitor, promotes cell apoptosis and tumor regression in both in vitro and in vivo models of castration-resistant prostate cancer
Bernales, Sebastian, Guerrero, Javier, Gomez, Francisco, Alfaro, Ivan E., Iguchi, Kanako, Kusayama, Toshiyuki, Protter, Andrew A.
Published in Molecular cancer therapeutics (12.11.2011)
Published in Molecular cancer therapeutics (12.11.2011)
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Binding of a Catechol Derivative of Denopamine (T-0509) and N-tert-Butylnoradrenaline (Colterol) to .BETA.1- and .BETA.2-Adrenoceptors
KUSAYAMA, Toshiyuki, OKA, Junichiro, YABANA, Hideo, ADACHI-AKAHANE, Satomi, NAGAO, Taku
Published in Biological & pharmaceutical bulletin (1994)
Published in Biological & pharmaceutical bulletin (1994)
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Effects of YM471, a nonpeptide AVP V 1A and V 2 receptor antagonist, on human AVP receptor subtypes expressed in CHO cells and oxytocin receptors in human uterine smooth muscle cells
Tsukada, Junko, Tahara, Atsuo, Tomura, Yuichi, Wada, Koh‐ichi, Kusayama, Toshiyuki, Ishii, Noe, Yatsu, Takeyuki, Uchida, Wataru, Taniguchi, Nobuaki, Tanaka, Akihiro
Published in British journal of pharmacology (29.01.2009)
Published in British journal of pharmacology (29.01.2009)
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Effects of YM218, a nonpeptide vasopressin V1A receptor-selective antagonist, on human vasopressin and oxytocin receptors
Tahara, Atsuo, Tsukada, Junko, Tomura, Yuichi, Kusayama, Toshiyuki, Wada, Koh-Ichi, Ishii, Noe, Taniguchi, Nobuaki, Suzuki, Takeshi, Yatsu, Takeyuki, Uchida, Wataru, Shibasaki, Masayuki
Published in Pharmacological research (01.03.2005)
Published in Pharmacological research (01.03.2005)
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Pharmacologic properties of YM218, a novel, potent, nonpeptide vasopressin V1A receptor-selective antagonist
Tsukada, Junko, Tahara, Atsuo, Tomura, Yuichi, Kusayama, Toshiyuki, Wada, Koh-ichi, Ishii, Noe, Taniguchi, Nobuaki, Suzuki, Takeshi, Yatsu, Takeyuki, Uchida, Wataru, Shibasaki, Masayuki
Published in Vascular pharmacology (01.01.2005)
Published in Vascular pharmacology (01.01.2005)
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Cardiovascular and renal effects of conivaptan hydrochloride (YM087), a vasopressin V 1A and V 2 receptor antagonist, in dogs with pacing-induced congestive heart failure
Yatsu, Takeyuki, Tomura, Yuichi, Tahara, Atsuo, Wada, Koh-ichi, Kusayama, Toshiyuki, Tsukada, Junko, Tokioka, Tomoko, Uchida, Wataru, Inagaki, Osamu, Iizumi, Yuichi, Tanaka, Akihiro, Honda, Kazuo
Published in European journal of pharmacology (09.07.1999)
Published in European journal of pharmacology (09.07.1999)
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Pharmacological characterization of YM471, a novel potent vasopressin V1A and V2 receptor antagonist
TSUKADA, Junko, TAHARA, Atsuo, TANAKA, Akihiro, TOMURA, Yuichi, WADA, Koh-Ichi, KUSAYAMA, Toshiyuki, ISHII, Noe, AOKI, Motonori, YATSU, Takeyuki, UCHIDA, Wataru, TANIGUCHI, Nobuaki
Published in European journal of pharmacology (20.06.2002)
Published in European journal of pharmacology (20.06.2002)
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Effects of YM218, a nonpeptide vasopressin V 1A receptor-selective antagonist, on human vasopressin and oxytocin receptors
Tahara, Atsuo, Tsukada, Junko, Tomura, Yuichi, Kusayama, Toshiyuki, Wada, Koh-ichi, Ishii, Noe, Taniguchi, Nobuaki, Suzuki, Takeshi, Yatsu, Takeyuki, Uchida, Wataru, Shibasaki, Masayuki
Published in Pharmacological research (01.03.2005)
Published in Pharmacological research (01.03.2005)
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EFFECT OF CONIVAPTAN, A COMBINED VASOPRESSIN V 1a AND V 2 RECEPTOR ANTAGONIST, ON VASOPRESSIN-INDUCED CARDIAC AND HAEMODYNAMIC CHANGES IN ANAESTHETISED DOGS
YATSU, TAKEYUKI, KUSAYAMA, TOSHIYUKI, TOMURA, YUICHI, ARAI, YUKINORI, AOKI, MOTONORI, TAHARA, ATSUO, WADA, KOH-ICHI, TSUKADA, JUNKO
Published in Pharmacological research (01.11.2002)
Published in Pharmacological research (01.11.2002)
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Binding and Signal Transduction Characteristics of the Nonpeptide Vasopressin V1A Receptor-Selective Antagonist YM218 in Cultured Rat Mesangial Cells
Tahara, Atsuo, Tsukada, Junko, Tomura, Yuichi, Kusayama, Toshiyuki, Momose, Kazuhiro, Taniguchi, Nobuaki, Suzuki, Takeshi, Yatsu, Takeyuki, Shibasaki, Masayuki
Published in Pharmacology (2006)
Published in Pharmacology (2006)
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Synthesis and biological activity of novel 4,4-difluorobenzazepine derivatives as non-peptide antagonists of the arginine vasopressin V 1A receptor
Shimada, Yoshiaki, Taniguchi, Nobuaki, Matsuhisa, Akira, Akane, Hiroaki, Kawano, Noriyuki, Suzuki, Takeshi, Tobe, Takahiko, Kakefuda, Akio, Yatsu, Takeyuki, Tahara, Atsuo, Tomura, Yuichi, Kusayama, Toshiyuki, Wada, Koh-ichi, Tsukada, Junko, Orita, Masaya, Tsunoda, Takashi, Tanaka, Akihiro
Published in Bioorganic & medicinal chemistry (15.03.2006)
Published in Bioorganic & medicinal chemistry (15.03.2006)
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Synthesis and biological activity of novel 4,4-difluorobenzazepine derivatives as non-peptide antagonists of the arginine vasopressin V1A receptor
SHIMADA, Yoshiaki, TANIGUCHI, Nobuaki, TOMURA, Yuichi, KUSAYAMA, Toshiyuki, WADA, Koh-Ichi, TSUKADA, Junko, ORITA, Masaya, TSUNODA, Takashi, TANAKA, Akihiro, MATSUHISA, Akira, AKANE, Hiroaki, KAWANO, Noriyuki, SUZUKI, Takeshi, TOBE, Takahiko, KAKEFUDA, Akio, YATSU, Takeyuki, TAHARA, Atsuo
Published in Bioorganic & medicinal chemistry (15.03.2006)
Published in Bioorganic & medicinal chemistry (15.03.2006)
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Synthesis and biological activity of novel 4,4-difluorobenzazepine derivatives as non-peptide antagonists of the arginine vasopressin V sub(1A) receptor
Shimada, Yoshiaki, Taniguchi, Nobuaki, Matsuhisa, Akira, Akane, Hiroaki, Kawano, Noriyuki, Suzuki, Takeshi, Tobe, Takahiko, Kakefuda, Akio, Yatsu, Takeyuki, Tahara, Atsuo, Tomura, Yuichi, Kusayama, Toshiyuki, Wada, Koh-Ichi, Tsukada, Junko, Orita, Masaya, Tsunoda, Takashi, Tanaka, Akihiro
Published in Bioorganic & medicinal chemistry (01.01.2006)
Published in Bioorganic & medicinal chemistry (01.01.2006)
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