Synthesis and biological evaluation of novel orally available 1-phenyl-6-aminouracils containing dimethyldihydrobenzofuranol structure for the treatment of allergic skin diseases
Tobe, Masanori, Tsuboi, Katsunori, Hasegawa, Futoshi, Fujiwara, Norio, Inoue, Yoshifumi, Isobe, Masakazu, Isobe, Yoshiaki
Published in Bioorganic & medicinal chemistry letters (15.02.2016)
Published in Bioorganic & medicinal chemistry letters (15.02.2016)
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Journal Article
New year greetings from editors of Drug Delivery System
Maruyama, Atsushi, Itaka, Keiji, Kawakami, Kohsaku, Koga, Yoshikatsu, Shiraishi, Koichi, Niidome, Takuro, Higuchi, Yuriko, Manabe, Shino, Ohta, Kotoe, Tobe, Masanori
Published in Drug Delivery System (25.01.2024)
Published in Drug Delivery System (25.01.2024)
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Journal Article
Asymmetric synthesis of the carbon-14-labeled selective glucocorticoid receptor modulator using cinchona alkaloid catalyzed addition of 6-bromoindole to ethyl trifluoropyruvate
Sumiyoshi, Takaaki, Urabe, Daisuke, Tojo, Kengo, Sakamoto, Masato, Niidome, Kazumi, Tsuboya, Norie, Nakajima, Tomoko, Tobe, Masanori
Published in Molecules (Basel, Switzerland) (30.05.2012)
Published in Molecules (Basel, Switzerland) (30.05.2012)
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Journal Article
The chemistry and biological activity of heterocycle-fused quinolinone derivatives: A review
Shiro, Tomoya, Fukaya, Takayuki, Tobe, Masanori
Published in European journal of medicinal chemistry (05.06.2015)
Published in European journal of medicinal chemistry (05.06.2015)
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Journal Article
New year greetings from editors of Drug Delivery System
Maruyama, Atsushi, Itaka, Keiji, Kawakami, Kohsaku, Koga, Yoshikatsu, Shiraishi, Koichi, Niidome, Takuro, Higuchi, Yuriko, Manabe, Shino, Ohta, Kotoe, Tobe, Masanori, 丸山 厚, 啓史, 位髙, 亘作, 川上, 宣勝, 古賀, 貢一, 白石, 琢郎, 新留, ゆり子, 樋口, 史乃, 眞鍋, 琴恵, 太田, 雅則, 戸邊
Published in Drug delivery system (01.01.2023)
Published in Drug delivery system (01.01.2023)
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Journal Article
Drug Delivery System編集委員/幹事からのご挨拶
丸山, 厚, 位髙, 啓史, 川上, 亘作, 古賀, 宣勝, 白石, 貢一, 新留, 琢郎, 樋口, ゆり子, 眞鍋, 史乃, 太田, 琴恵, 戸邊, 雅則
Published in Drug Delivery System (25.01.2024)
Published in Drug Delivery System (25.01.2024)
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Journal Article
Prodrugs of 9-Benzyl-8-hydroxy-2-(2-hydroxyethylthio)adenine: Potent Interferon Inducing Agents in Monkeys
Kurimoto, Ayumu, Tobe, Masanori, Ogita, Haruhisa, Ogino, Tetsuhiro, Takaku, Haruo, Ichii, Shinji, Kawakami, Hajime, Isobe, Yoshiaki
Published in Chemical & pharmaceutical bulletin (01.04.2004)
Published in Chemical & pharmaceutical bulletin (01.04.2004)
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Journal Article
Construction of 3,5-substituted 1,2,4-oxadiazole rings triggered by tetrabutylammonium hydroxide: a highly efficient and fluoride-free ring closure reaction of O-acylamidoximes
Otaka, Hiromichi, Ikeda, Junya, Tanaka, Daisuke, Tobe, Masanori
Published in Tetrahedron letters (29.01.2014)
Published in Tetrahedron letters (29.01.2014)
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Journal Article
Synthesis and Activity of a Metabolite of (S)-6-Amino-5-(6-hydroxy-2,5,7,8-tetramethylchroman-2-carboxamido)-3-methyl-1-phenyl-2,4-(1H,3H)-pyrimidinedione (CX-659S)
Isobe, Yoshiaki, Tobe, Masanori, Takahashi, Osamu, Goto, Yuso, Inoue, Yoshifumi, Obara, Fumihiro, Tsuchiya, Masami, Hayashi, Hideya
Published in Chemical & pharmaceutical bulletin (01.10.2002)
Published in Chemical & pharmaceutical bulletin (01.10.2002)
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Journal Article
Prodrugs of 9-Benzyl-8-hydroxy-2-(2-hydroxyethylthio)adenine:Potent Interferon Inducing Agents in Monkeys
Ayumu KURIMOTO, Masanori TOBE, Haruhisa OGITA, Tetsuhiro OGINO, Haruo TAKAKU, Shinji ICHII, Hajime KAWAKAMI, Yoshiaki ISOBE
Published in Chemical & Pharmaceutical Bulletin (2004)
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Published in Chemical & Pharmaceutical Bulletin (2004)
Journal Article
Structure–Activity Relationships of 6-Nitroquinazolines: Dual-Acting Compounds with Inhibitory Activities toward both TNF-α Production and T Cell Proliferation
Tobe, Masanori, Isobe, Yoshiaki, Tomizawa, Hideyuki, Nagasaki, Takahiro, Obara, Fumihiro, Matsumoto, Mitsuhiro, Hayashi, Hideya
Published in Chemical & pharmaceutical bulletin (01.08.2002)
Published in Chemical & pharmaceutical bulletin (01.08.2002)
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Journal Article
Synthesis and Evaluation of 6-Nitro-7-(1-piperazino)quinazolines: Dual-Acting Compounds with Inhibitory Activities toward Both Tumor Necrosis Factor-α (TNF-α) Production and T Cell Proliferation
Tobe, Masanori, Isobe, Yoshiaki, Tomizawa, Hideyuki, Nagasaki, Takahiro, Aoki, Masamitsu, Negishi, Toru, Hayashi, Hideya
Published in Chemical & pharmaceutical bulletin (2003)
Published in Chemical & pharmaceutical bulletin (2003)
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Journal Article
Design and synthesis of an aminopiperidine series of gamma-secretase modulators
Kobayashi, Tomonori, Iwama, Seiji, Fusano, Akira, Kato, Yoshihiro, Ikeda, Atsushi, Teranishi, Yasuhiro, Nishihara, Akemi, Tobe, Masanori
Published in Bioorganic & medicinal chemistry letters (01.01.2014)
Published in Bioorganic & medicinal chemistry letters (01.01.2014)
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Journal Article
Synthesis and structure―activity relationships of phenothiazine carboxylic acids having pyrimidine-dione as novel histamine H1 antagonists
KUBOTA, Katsumi, KUREBAYASHI, Hirotaka, MIYACHI, Hirotaka, TOBE, Masanori, ONISHI, Masako, ISOBE, Yoshiaki
Published in Bioorganic & medicinal chemistry letters (01.05.2009)
Published in Bioorganic & medicinal chemistry letters (01.05.2009)
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Journal Article
Synthesis and structure–activity relationships of phenothiazine carboxylic acids having pyrimidine-dione as novel histamine H 1 antagonists
Kubota, Katsumi, Kurebayashi, Hirotaka, Miyachi, Hirotaka, Tobe, Masanori, Onishi, Masako, Isobe, Yoshiaki
Published in Bioorganic & medicinal chemistry letters (15.05.2009)
Published in Bioorganic & medicinal chemistry letters (15.05.2009)
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