Discovery of the Soluble Guanylate Cyclase Stimulator Vericiguat (BAY 1021189) for the Treatment of Chronic Heart Failure
Follmann, Markus, Ackerstaff, Jens, Redlich, Gorden, Wunder, Frank, Lang, Dieter, Kern, Armin, Fey, Peter, Griebenow, Nils, Kroh, Walter, Becker-Pelster, Eva-Maria, Kretschmer, Axel, Geiss, Volker, Li, Volkhart, Straub, Alexander, Mittendorf, Joachim, Jautelat, Rolf, Schirok, Hartmut, Schlemmer, Karl-Heinz, Lustig, Klemens, Gerisch, Michael, Knorr, Andreas, Tinel, Hanna, Mondritzki, Thomas, Trübel, Hubert, Sandner, Peter, Stasch, Johannes-Peter
Published in Journal of medicinal chemistry (22.06.2017)
Published in Journal of medicinal chemistry (22.06.2017)
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Journal Article
Reversal of rivaroxaban anticoagulation by haemostatic agents in rats and primates
Perzborn, Elisabeth, Gruber, András, Tinel, Hanna, Marzec, Ulla M, Buetehorn, Ulf, Buchmueller, Anja, Heitmeier, Stefan, Laux, Volker
Published in Thrombosis and haemostasis (2013)
Published in Thrombosis and haemostasis (2013)
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Journal Article
Transcriptome Characterization of Estrogen-Treated Human Myocardium Identifies Myosin Regulatory Light Chain Interacting Protein as a Sex-Specific Element Influencing Contractile Function
Kararigas, Georgios, PhD, Bito, Virginie, PhD, Tinel, Hanna, PhD, Becher, Eva, PhD, Baczko, Istvan, MD, PhD, Knosalla, Christoph, MD, Albrecht-Küpper, Barbara, PhD, Sipido, Karin R., MD, PhD, Regitz-Zagrosek, Vera, MD
Published in Journal of the American College of Cardiology (24.01.2012)
Published in Journal of the American College of Cardiology (24.01.2012)
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Journal Article
Inhaled mosliciguat (BAY 1237592): targeting pulmonary vasculature via activating apo-sGC
Becker-Pelster, Eva M., Hahn, Michael G., Delbeck, Martina, Dietz, Lisa, Hüser, Jörg, Kopf, Johannes, Kraemer, Thomas, Marquardt, Tobias, Mondritzki, Thomas, Nagelschmitz, Johannes, Nikkho, Sylvia M., Pires, Philippe V., Tinel, Hanna, Weimann, Gerrit, Wunder, Frank, Sandner, Peter, Schuhmacher, Joachim, Stasch, Johannes-Peter, Truebel, Hubert K. F.
Published in Respiratory research (01.10.2022)
Published in Respiratory research (01.10.2022)
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Journal Article
Chymase Inhibition Resolves and Prevents Deep Vein Thrombosis Without Increasing Bleeding Time in the Mouse Model
Lapointe, Catherine, Vincent, Laurence, Giguère, Hugo, Auger-Messier, Mannix, Schwertani, Adel, Jin, Denan, Takai, Shinji, Pejler, Gunnar, Sirois, Martin G, Tinel, Hanna, Heitmeier, Stefan, D'Orléans-Juste, Pedro
Published in Journal of the American Heart Association (21.02.2023)
Published in Journal of the American Heart Association (21.02.2023)
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Journal Article
Effects of PDE5 Inhibitors and sGC Stimulators in a Rat Model of Artificial Ureteral Calculosis
Sandner, Peter, Tinel, Hanna, Affaitati, Giannapia, Costantini, Raffaele, Giamberardino, Maria Adele
Published in PloS one (28.10.2015)
Published in PloS one (28.10.2015)
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Journal Article
Discovery of the Soluble Guanylate Cyclase Activator Runcaciguat (BAY 1101042)
Hahn, Michael G, Lampe, Thomas, El Sheikh, Sherif, Griebenow, Nils, Woltering, Elisabeth, Schlemmer, Karl-Heinz, Dietz, Lisa, Gerisch, Michael, Wunder, Frank, Becker-Pelster, Eva-Maria, Mondritzki, Thomas, Tinel, Hanna, Knorr, Andreas, Kern, Armin, Lang, Dieter, Hueser, Joerg, Schomber, Tibor, Benardeau, Agnes, Eitner, Frank, Truebel, Hubert, Mittendorf, Joachim, Kumar, Vijay, van den Akker, Focco, Schaefer, Martina, Geiss, Volker, Sandner, Peter, Stasch, Johannes-Peter
Published in Journal of medicinal chemistry (13.05.2021)
Published in Journal of medicinal chemistry (13.05.2021)
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Journal Article
The Novel Potent and Selective Vasopressin V1a Antagonist BAY2327949 Blocks Arginine Vasopressin-Mediated Decline of Renal Blood Flow and Tissue Oxygenation: PO0647
Cernecka, Hana, Droebner, Karoline, Tinel, Hanna, Pook, Eisabeth, Fuerstner, Chantal, Collin, Marie-Pierre L., Hein, Peter, Eitner, Frank, Kolkhof, Peter
Published in Journal of the American Society of Nephrology (01.10.2020)
Published in Journal of the American Society of Nephrology (01.10.2020)
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Journal Article
Telemetric long-term assessment of autonomic function in experimental heart failure
Boden, Katharina, Pongratanakul, Pailin, Vogel, Julia, Willemsen, Nicola, Jülke, Eva-Maria, Balitzki, Jakob, Tinel, Hanna, Truebel, Hubert, Dinh, Wilfried, Mondritzki, Thomas
Published in Journal of pharmacological and toxicological methods (01.11.2023)
Published in Journal of pharmacological and toxicological methods (01.11.2023)
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Journal Article
Identification and characterization of the new generation soluble guanylate cyclase stimulator BAY‐747 designed for the treatment of resistant hypertension
Wunder, Frank, Stasch, Johannes‐Peter, Knorr, Andreas, Mondritzki, Thomas, Brockschnieder, Damian, Becker‐Pelster, Eva‐Maria, Sandner, Peter, Tinel, Hanna, Redlich, Gorden, Hartung, Ingo V., Vakalopoulos, Alexandros, Follmann, Markus
Published in British journal of pharmacology (01.10.2023)
Published in British journal of pharmacology (01.10.2023)
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Journal Article
Synergistic effects of BAY 60-4552 and vardenafil on relaxation of corpus cavernosum tissue of patients with erectile dysfunction and clinical phosphodiesterase type 5 inhibitor failure
Albersen, Maarten, Linsen, Loes, Tinel, Hanna, Sandner, Peter, Van Renterghem, Koenraad
Published in Journal of sexual medicine (01.05.2013)
Published in Journal of sexual medicine (01.05.2013)
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Journal Article
Vascular Protection and Decongestion Without Renin-Angiotensin-Aldosterone System Stimulation Mediated by a Novel Dual-Acting Vasopressin V1a/V2 Receptor Antagonist
Kolkhof, Peter, Pook, Elisabeth, Pavkovic, Mira, Kretschmer, Axel, Buchmüller, Anja, Tinel, Hanna, Delbeck, Martina, Mondritzki, Thomas, Wasnaire, Pierre, Dinh, Wilfried, Truebel, Hubert, Hüser, Jörg, Schmeck, Carsten
Published in Journal of cardiovascular pharmacology (01.07.2019)
Published in Journal of cardiovascular pharmacology (01.07.2019)
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Journal Article
Additive effects of the Rho kinase inhibitor Y‐27632 and vardenafil on relaxation of the corpus cavernosum tissue of patients with erectile dysfunction and clinical phosphodiesterase type 5 inhibitor failure
Uvin, Pieter, Albersen, Maarten, Bollen, Ine, Falter, Maarten, Weyne, Emmanuel, Linsen, Loes, Tinel, Hanna, Sandner, Peter, Bivalacqua, Trinity J., De Ridder, Dirk J. M. K., Van der Aa, Frank, Brône, Bert, Van Renterghem, Koenraad
Published in BJU international (01.02.2017)
Published in BJU international (01.02.2017)
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Journal Article
7- 1---3- 7-SUBSTITUTED 1-ARYL-NAPHTHYRIDINE-3-CARBOXYLIC ACID AMIDES AND USE THEREOF
BRECHMANN MARKUS, TINEL HANNA, MONDRITZKI THOMAS, VAKALOPOULOS ALEXANDROS, FREUDENBERGER TILL, WITTWER MATTHIAS BEAT, KULLMANN MAXIMILIAN ANDREAS, MARQUARDT TOBIAS, BOULTADAKIS ARAPINIS MELISSA, TELLER HENRIK, STRAUB ALEXANDER
Year of Publication 13.03.2023
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Year of Publication 13.03.2023
Patent
MP47-20 INCREASED RHO-KINASE 2 AND AN INCREASE OF SYNTHETIC SMOOTH MUSCLE-SPECIFIC MARKER EXPRESSION IS OBSERVED IN THE CORPUS CAVERNOSUM OF PATIENTS WITH SEVERE ERECTILE DYSFUNCTION
Albersen, Maarten, Bivalacqua, Trinity, Hannan, Johanna, Linsen, Loes, Weyne, Emmanuel, Tinel, Hanna, Sandner, Peter, Uvin, Pieter, Van Renterghem, Koenraad
Published in The Journal of urology (01.04.2014)
Published in The Journal of urology (01.04.2014)
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