Influence of lipophilicity on the interactions of N-alkyl-4-phenyl-1,2,3,6-tetrahydropyridines and their positively charged N-alkyl-4-phenylpyridinium metabolites with cytochrome P450 2D6
Kalgutkar, Amit S, Zhou, Sue, Fahmi, Odette A, Taylor, Timothy J
Published in Drug metabolism and disposition (01.05.2003)
Published in Drug metabolism and disposition (01.05.2003)
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Optimization of the physicochemical and pharmacokinetic attributes in a 6-azauracil series of P2X 7 receptor antagonists leading to the discovery of the clinical candidate CE-224,535
Duplantier, Allen J., Dombroski, Mark A., Subramanyam, Chakrapani, Beaulieu, Aimee M., Chang, Shang-Poa, Gabel, Christopher A., Jordan, Crystal, Kalgutkar, Amit S., Kraus, Kenneth G., Labasi, Jeff M., Mussari, Christopher, Perregaux, David G., Shepard, Rick, Taylor, Timothy J., Trevena, Kristen A., Whitney-Pickett, Carrie, Yoon, Kwansik
Published in Bioorganic & medicinal chemistry letters (15.06.2011)
Published in Bioorganic & medicinal chemistry letters (15.06.2011)
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Journal Article
Optimization of the physicochemical and pharmacokinetic attributes in a 6-azauracil series of P2X sub(7 receptor antagonists leading to the discovery of the clinical candidate CE-224,535)
Duplantier, Allen J, Dombroski, Mark A, Subramanyam, Chakrapani, Beaulieu, Aimee M, Chang, Shang-Poa, Gabel, Christopher A, Jordan, Crystal, Kalgutkar, Amit S, Kraus, Kenneth G, Labasi, Jeff M, Mussari, Christopher, Perregaux, David G, Shepard, Rick, Taylor, Timothy J, Trevena, Kristen A, Whitney-Pickett, Carrie, Yoon, Kwansik
Published in Bioorganic & medicinal chemistry letters (15.06.2011)
Published in Bioorganic & medicinal chemistry letters (15.06.2011)
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Journal Article
Preclinical pharmacokinetics and metabolism of 6-(4-(2,5-difluorophenyl)oxazol-5-yl)-3-isopropyl-[1,2,4]-triazolo[4,3-a]pyridine, a novel and selective p38α inhibitor: identification of an active metabolite in preclinical species and human liver microsomes
Kalgutkar, Amit S., Hatch, Heather L., Kosea, Frederick, Nguyen, Hang T., Choo, Edna F., McClure, Kim F., Taylor, Timothy J., Henne, Kirk R., Kuperman, Alexander V., Dombroski, Mark A., Letavic, Michael A.
Published in Biopharmaceutics & drug disposition (01.11.2006)
Published in Biopharmaceutics & drug disposition (01.11.2006)
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Influence of Lipophilicity on the Interactions ofN-Alkyl-4-phenyl-1,2,3,6-tetrahydropyridines and Their Positively Charged N-Alkyl-4-phenylpyridinium Metabolites with Cytochrome P450 2D6
Amit S. Kalgutkar, Sue Zhou, Odette A. Fahmi, Timothy J. Taylor
Published in Drug metabolism and disposition (01.05.2003)
Published in Drug metabolism and disposition (01.05.2003)
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Journal Article
Influence of lipophilicity on the interactions of N-alkyl-4-phenyl-1,2,3,6-tetrahydropyridines and their positively charged N-alkyl-4-phenylpyridinium metabolites with cytochrome Pp450 2D6
KALGUTKAR, Amit S, ZHOU, Sue, FAHMI, Odette A, TAYLOR, Timothy J
Published in Drug metabolism and disposition (2003)
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Published in Drug metabolism and disposition (2003)
Journal Article
HYPOCHLORITE BASED HARD SURFACE DISINFECTANTS
BOROKHOV, OLGA, CARRIER, ROBERT, SOM, ABHIGYAN, TAYLOR, TIMOTHY J, JANI, HARISH, JACKSON, ANABELL
Year of Publication 02.08.2022
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Year of Publication 02.08.2022
Patent
HYPOCHLORITE BASED HARD SURFACE DISINFECTANTS
Som, Abhigyan, Jackson, Anabell, Jani, Harish, Carrier, Robert, Borokhov, Olga, Taylor, Timothy J
Year of Publication 13.05.2021
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Year of Publication 13.05.2021
Patent
Preclinical pharmacokinetics and metabolism of 6-(4-(2,5-difluorophenyl)oxazol-5-yl)-3-isopropyl-[1,2,4]-triazolo[4,3-a]pyridine, a novel and selective p38alpha inhibitor: identification of an active metabolite in preclinical species and human liver microsomes
Kalgutkar, Amit S, Hatch, Heather L, Kosea, Frederick, Nguyen, Hang T, Choo, Edna F, McClure, Kim F, Taylor, Timothy J, Henne, Kirk R, Kuperman, Alexander V, Dombroski, Mark A, Letavic, Michael A
Published in Biopharmaceutics & drug disposition (01.11.2006)
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Published in Biopharmaceutics & drug disposition (01.11.2006)
Journal Article
Hypochlorite based hard surface disinfectants
Som, Abhigyan, Jackson, Anabell, Jani, Harish, Carrier, Robert, Borokhov, Olga, Taylor, Timothy J
Year of Publication 26.01.2021
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Year of Publication 26.01.2021
Patent
Preclinical pharmacokinetics and metabolism of 6-(4-(2,5-difluorophenyl)oxazol-5-yl)-3 -isopropyl -[1,2,4 ] -triazolo [4,3-a] pyridine, a novel and selective p38a inhibitor : Identification of an active metabolite in preclinical species and human liver microsomes
KALGUTKAR, Amit S, HATCH, Heather L, LETAVIC, Michael A, KOSEA, Frederick, NGUYEN, Hang T, CHOO, Edna F, MCCLURE, Kim F, TAYLOR, Timothy J, HENNE, Kirk R, KUPERMAN, Alexander V, DOMBROSKI, Mark A
Published in Biopharmaceutics & drug disposition (2006)
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Published in Biopharmaceutics & drug disposition (2006)
Journal Article
Preclinical pharmacokinetics and metabolism of 6-(4-(2,5- difluorophenyl)oxazol-5-yl)-3-isopropyl-[1,2,4]-triazolo[4,3-a]pyr idine , a novel and selective p38 alpha inhibitor: identification of an active metabolite in preclinical species and human liver microsomes
Kalgutkar, Amit S, Hatch, Heather L, Kosea, Frederick, Nguyen, Hang T, Choo, Edna F, McClure, Kim F, Taylor, Timothy J, Henne, Kirk R, Kuperman, Alexander V, Dombroski, Mark A, Letavic, Michael A
Published in Biopharmaceutics & drug disposition (01.01.2006)
Published in Biopharmaceutics & drug disposition (01.01.2006)
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Journal Article
Identification of criticality in neuronal avalanches: II. A theoretical and empirical investigation of the driven case
Hartley, Caroline, Taylor, Timothy J, Kiss, Istvan Z, Farmer, Simon F, Berthouze, Luc
Published in arXiv.org (13.09.2013)
Published in arXiv.org (13.09.2013)
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