Advances in Bacterial Methionine Aminopeptidase Inhibition
Helgren, Travis R, Wangtrakuldee, Phumvadee, Staker, Bart L, Hagen, Timothy J
Published in Current topics in medicinal chemistry (01.01.2016)
Published in Current topics in medicinal chemistry (01.01.2016)
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A single Leishmania adenylate forming enzyme of the ANL superfamily generates both acetyl- and acetoacetyl-CoA
Jezewski, Andrew J., Esan, Taiwo E., Propp, Jonah, Fuller, Andrew J., Daraji, Drashti G., Lail, Charles, Staker, Bart L., Woodward, Elijah L., Liu, Linjun, Battaile, Kevin P., Lovell, Scott, Hagen, Timothy J., Krysan, Damian J.
Published in The Journal of biological chemistry (10.10.2024)
Published in The Journal of biological chemistry (10.10.2024)
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Design and Synthesis of Selective Phosphodiesterase 4D (PDE4D) Allosteric Inhibitors for the Treatment of Fragile X Syndrome and Other Brain Disorders
Gurney, Mark E, Nugent, Richard A, Mo, Xuesheng, Sindac, Janice A, Hagen, Timothy J, Fox, David, O’Donnell, James M, Zhang, Chong, Xu, Ying, Zhang, Han-Ting, Groppi, Vincent E, Bailie, Marc, White, Ronald E, Romero, Donna L, Vellekoop, A. Samuel, Walker, Joel R, Surman, Matthew D, Zhu, Lei, Campbell, Robert F
Published in Journal of medicinal chemistry (23.05.2019)
Published in Journal of medicinal chemistry (23.05.2019)
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The synthesis, antimalarial activity and CoMFA analysis of novel aminoalkylated quercetin analogs
Helgren, Travis R., Sciotti, Richard J., Lee, Patricia, Duffy, Sandra, Avery, Vicky M., Igbinoba, Osayawemwen, Akoto, Matthew, Hagen, Timothy J.
Published in Bioorganic & medicinal chemistry letters (15.01.2015)
Published in Bioorganic & medicinal chemistry letters (15.01.2015)
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Structural and biophysical characterization of the Burkholderia pseudomallei IspF inhibitor L-tryptophan hydroxamate
Blain, Joy M., Grote, Dakota L., Watkins, Sydney M., Goshu, Gashaw M., Muller, Chanté, Gorman, James L., Ranieri, Gina, Walter, Richard L., Hofstetter, Heike, Horn, James R., Hagen, Timothy J.
Published in Bioorganic & medicinal chemistry letters (15.09.2021)
Published in Bioorganic & medicinal chemistry letters (15.09.2021)
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Structural Characterization of the Reaction and Substrate Specificity Mechanisms of Pathogenic Fungal Acetyl-CoA Synthetases
Jezewski, Andrew J, Alden, Katy M, Esan, Taiwo E, DeBouver, Nicholas D, Abendroth, Jan, Bullen, Jameson C, Calhoun, Brandy M, Potts, Kristy T, Murante, Daniel M, Hagen, Timothy J, Fox, David, Krysan, Damian J
Published in ACS chemical biology (20.08.2021)
Published in ACS chemical biology (20.08.2021)
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Bacterial structural genomics target enabled by a recently discovered potent fungal acetyl‐CoA synthetase inhibitor
DeBouver, Nicholas D., Bolejack, Madison J., Esan, Taiwo E., Krysan, Damian J., Hagen, Timothy J., Abendroth, Jan
Published in Acta crystallographica. Section F, Structural biology communications (01.06.2023)
Published in Acta crystallographica. Section F, Structural biology communications (01.06.2023)
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Traditional Kenyan herbal medicine: exploring natural products’ therapeutics against schistosomiasis
Ndegwa, Fidensio K., Kondam, Chaitanya, Aboagye, Samuel Y., Esan, Taiwo E., Waxali, Zohra Sattar, Miller, Margaret E., Gikonyo, Nicholas K., Mbugua, Paul K., Okemo, Paul O., Williams, David L., Hagen, Timothy J.
Published in Journal of helminthology (03.03.2022)
Published in Journal of helminthology (03.03.2022)
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Compound D159687, a phosphodiesterase 4D inhibitor, induces weight and fat mass loss in aged mice without changing lean mass, physical and cognitive function
Muo, Ijeoma M., Park, Sung-Jun, Smith, Antoine, A. Springer, Danielle, Allen, Michele D., Hagen, Timothy J., Chung, Jay H.
Published in Biochemical and biophysical research communications (02.12.2018)
Published in Biochemical and biophysical research communications (02.12.2018)
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Antibacterial activity of 2-amino-4-hydroxypyrimidine-5-carboxylates and binding to Burkholderia pseudomallei 2-C-methyl-d-erythritol-2,4-cyclodiphosphate synthase
Watkins, Sydney M., Ghose, Debarati, Blain, Joy M., Grote, Dakota L., Luan, Chi-Hao, Clare, Michael, Meganathan, R., Horn, James R., Hagen, Timothy J.
Published in Bioorganic & medicinal chemistry letters (15.10.2019)
Published in Bioorganic & medicinal chemistry letters (15.10.2019)
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Discovery of triazines as selective PDE4B versus PDE4D inhibitors
Hagen, Timothy J., Mo, Xuesheng, Burgin, Alex B., Fox, David, Zhang, Zheng, Gurney, Mark E.
Published in Bioorganic & medicinal chemistry letters (15.08.2014)
Published in Bioorganic & medicinal chemistry letters (15.08.2014)
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A concise synthesis of biaryl PDE4D allosteric modulators
Dalby, Amy, Mo, Xuesheng, Stoa, Robert, Wroblewski, Nathaniel, Zhang, Zheng, Hagen, Timothy J.
Published in Tetrahedron letters (22.05.2013)
Published in Tetrahedron letters (22.05.2013)
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Rickettsia prowazekii methionine aminopeptidase as a promising target for the development of antibacterial agents
Helgren, Travis R., Chen, Congling, Wangtrakuldee, Phumvadee, Edwards, Thomas E., Staker, Bart L., Abendroth, Jan, Sankaran, Banumathi, Housley, Nicole A., Myler, Peter J., Audia, Jonathon P., Horn, James R., Hagen, Timothy J.
Published in Bioorganic & medicinal chemistry (01.02.2017)
Published in Bioorganic & medicinal chemistry (01.02.2017)
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Dissemination of Imidacloprid Through Dairy Cattle Manure and Its Effect on the Biological Control Agent, Spalangia endius (Hymenoptera: Pteromalidae), and a Filth Fly Host, Musca domestica (Diptera: Muscidae)
Burgess, Edwin R., Watkins, Sydney M., King, Bethia H., Chantos-Davidson, Karley, Kremer, Aspen N., Tournear, Jennifer C., Morrow, Joseph, Hagen, Timothy J., Gaillard, Elizabeth R.
Published in Journal of economic entomology (21.03.2019)
Published in Journal of economic entomology (21.03.2019)
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Crystal structure and biophysical characterization of IspD from Burkholderia thailandensis and Mycobacterium paratuberculosis
Pierce, Phillip G, Hartnett, Brian E, Laughlin, Tosha M, Blain, Joy M, Mayclin, Stephen J, Bolejack, Madison J, Myers, Janette B, Higgins, Tate W, Dranow, David M, Sullivan, Amy, Lorimer, Donald D, Edwards, Thomas E, Hagen, Timothy J, Horn, James R, Myler, Peter J
Published in Acta crystallographica. Section F, Structural biology communications (01.02.2024)
Published in Acta crystallographica. Section F, Structural biology communications (01.02.2024)
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The identification of inhibitory compounds of Rickettsia prowazekii methionine aminopeptidase for antibacterial applications
Helgren, Travis R., Seven, Elif S., Chen, Congling, Edwards, Thomas E., Staker, Bart L., Abendroth, Jan, Myler, Peter J., Horn, James R., Hagen, Timothy J.
Published in Bioorganic & medicinal chemistry letters (01.05.2018)
Published in Bioorganic & medicinal chemistry letters (01.05.2018)
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Synthesis and biological evaluation of pyrazolopyrimidines as potential antibacterial agents
Goshu, Gashaw M., Ghose, Debarati, Bain, Joy M., Pierce, Phillip G., Begley, Darren W., Hewitt, Stephen N., Udell, Hannah S., Myler, Peter J., Meganathan, R., Hagen, Timothy J.
Published in Bioorganic & medicinal chemistry letters (15.12.2015)
Published in Bioorganic & medicinal chemistry letters (15.12.2015)
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