mTORC2 Regulates Amino Acid Metabolism in Cancer by Phosphorylation of the Cystine-Glutamate Antiporter xCT
Gu, Yuchao, Albuquerque, Claudio P., Braas, Daniel, Zhang, Wei, Villa, Genaro R., Bi, Junfeng, Ikegami, Shiro, Masui, Kenta, Gini, Beatrice, Yang, Huijun, Gahman, Timothy C., Shiau, Andrew K., Cloughesy, Timothy F., Christofk, Heather R., Zhou, Huilin, Guan, Kun-Liang, Mischel, Paul S.
Published in Molecular cell (06.07.2017)
Published in Molecular cell (06.07.2017)
Get full text
Journal Article
EGFR Mutation Promotes Glioblastoma through Epigenome and Transcription Factor Network Remodeling
Liu, Feng, Hon, Gary C., Villa, Genaro R., Turner, Kristen M., Ikegami, Shiro, Yang, Huijun, Ye, Zhen, Li, Bin, Kuan, Samantha, Lee, Ah Young, Zanca, Ciro, Wei, Bowen, Lucey, Greg, Jenkins, David, Zhang, Wei, Barr, Cathy L., Furnari, Frank B., Cloughesy, Timothy F., Yong, William H., Gahman, Timothy C., Shiau, Andrew K., Cavenee, Webster K., Ren, Bing, Mischel, Paul S.
Published in Molecular cell (15.10.2015)
Published in Molecular cell (15.10.2015)
Get full text
Journal Article
An LXR-Cholesterol Axis Creates a Metabolic Co-Dependency for Brain Cancers
Villa, Genaro R., Hulce, Jonathan J., Zanca, Ciro, Bi, Junfeng, Ikegami, Shiro, Cahill, Gabrielle L., Gu, Yuchao, Lum, Kenneth M., Masui, Kenta, Yang, Huijun, Rong, Xin, Hong, Cynthia, Turner, Kristen M., Liu, Feng, Hon, Gary C., Jenkins, David, Martini, Michael, Armando, Aaron M., Quehenberger, Oswald, Cloughesy, Timothy F., Furnari, Frank B., Cavenee, Webster K., Tontonoz, Peter, Gahman, Timothy C., Shiau, Andrew K., Cravatt, Benjamin F., Mischel, Paul S.
Published in Cancer cell (14.11.2016)
Published in Cancer cell (14.11.2016)
Get full text
Journal Article
Dual Targeting of Bromodomain and Extraterminal Domain Proteins, and WNT or MAPK Signaling, Inhibits c-MYC Expression and Proliferation of Colorectal Cancer Cells
Tögel, Lars, Nightingale, Rebecca, Chueh, Anderly C, Jayachandran, Aparna, Tran, Hoanh, Phesse, Toby, Wu, Rui, Sieber, Oliver M, Arango, Diego, Dhillon, Amardeep S, Dawson, Mark A, Diez-Dacal, Beatriz, Gahman, Timothy C, Filippakopoulos, Panagis, Shiau, Andrew K, Mariadason, John M
Published in Molecular cancer therapeutics (01.06.2016)
Published in Molecular cancer therapeutics (01.06.2016)
Get full text
Journal Article
A Cell Biologist's Field Guide to Aurora Kinase Inhibitors
de Groot, Christian O, Hsia, Judy E, Anzola, John V, Motamedi, Amir, Yoon, Michelle, Wong, Yao Liang, Jenkins, David, Lee, Hyun J, Martinez, Mallory B, Davis, Robert L, Gahman, Timothy C, Desai, Arshad, Shiau, Andrew K
Published in Frontiers in oncology (21.12.2015)
Published in Frontiers in oncology (21.12.2015)
Get full text
Journal Article
Reversible centriole depletion with an inhibitor of Polo-like kinase 4
Wong, Yao Liang, Anzola, John V., Davis, Robert L., Yoon, Michelle, Motamedi, Amir, Kroll, Ashley, Seo, Chanmee P., Hsia, Judy E., Kim, Sun K., Mitchell, Jennifer W., Mitchell, Brian J., Desai, Arshad, Gahman, Timothy C., Shiau, Andrew K., Oegema, Karen
Published in Science (American Association for the Advancement of Science) (05.06.2015)
Published in Science (American Association for the Advancement of Science) (05.06.2015)
Get full text
Journal Article
Inhibition of Nuclear PTEN Tyrosine Phosphorylation Enhances Glioma Radiation Sensitivity through Attenuated DNA Repair
Ma, Jianhui, Benitez, Jorge A., Li, Jie, Miki, Shunichiro, Ponte de Albuquerque, Claudio, Galatro, Thais, Orellana, Laura, Zanca, Ciro, Reed, Rachel, Boyer, Antonia, Koga, Tomoyuki, Varki, Nissi M., Fenton, Tim R., Nagahashi Marie, Suely Kazue, Lindahl, Erik, Gahman, Timothy C., Shiau, Andrew K., Zhou, Huilin, DeGroot, John, Sulman, Erik P., Cavenee, Webster K., Kolodner, Richard D., Chen, Clark C., Furnari, Frank B.
Published in Cancer cell (18.03.2019)
Published in Cancer cell (18.03.2019)
Get full text
Journal Article
An inhibitor of the proteasomal deubiquitinating enzyme USP14 induces tau elimination in cultured neurons
Boselli, Monica, Lee, Byung-Hoon, Robert, Jessica, Prado, Miguel A., Min, Sang-Won, Cheng, Chialin, Silva, M. Catarina, Seong, Changhyun, Elsasser, Suzanne, Hatle, Ketki M., Gahman, Timothy C., Gygi, Steven P., Haggarty, Stephen J., Gan, Li, King, Randall W., Finley, Daniel
Published in The Journal of biological chemistry (24.11.2017)
Published in The Journal of biological chemistry (24.11.2017)
Get full text
Journal Article
Synthesis and SAR of thiophene containing kinesin spindle protein (KSP) inhibitors
Pinkerton, Anthony B., Lee, Tom T., Hoffman, Timothy Z., Wang, Yan, Kahraman, Mehmet, Cook, Travis G., Severance, Daniel, Gahman, Timothy C., Noble, Stewart A., Shiau, Andrew K., Davis, Robert L.
Published in Bioorganic & medicinal chemistry letters (01.07.2007)
Published in Bioorganic & medicinal chemistry letters (01.07.2007)
Get full text
Journal Article
Glioblastoma cellular cross-talk converges on NF-κB to attenuate EGFR inhibitor sensitivity
Zanca, Ciro, Villa, Genaro R, Benitez, Jorge A, Thorne, Amy Haseley, Koga, Tomoyuki, D'Antonio, Matteo, Ikegami, Shiro, Ma, Jianhui, Boyer, Antonia D, Banisadr, Afsheen, Jameson, Nathan M, Parisian, Alison D, Eliseeva, Olesja V, Barnabe, Gabriela F, Liu, Feng, Wu, Sihan, Yang, Huijun, Wykosky, Jill, Frazer, Kelly A, Verkhusha, Vladislav V, Isaguliants, Maria G, Weiss, William A, Gahman, Timothy C, Shiau, Andrew K, Chen, Clark C, Mischel, Paul S, Cavenee, Webster K, Furnari, Frank B
Published in Genes & development (15.06.2017)
Published in Genes & development (15.06.2017)
Get full text
Journal Article
Inhibition of Nuclear PTEN Tyrosine Phosphorylation Enhances Glioma Radiation Sensitivity through Attenuated DNA Repair
Ma, Jianhui, Benitez, Jorge A., Li, Jie, Miki, Shunichiro, Ponte de Albuquerque, Claudio, Galatro, Thais, Orellana, Laura, Zanca, Ciro, Reed, Rachel, Boyer, Antonia, Koga, Tomoyuki, Varki, Nissi M., Fenton, Tim R., Nagahashi Marie, Suely Kazue, Lindahl, Erik, Gahman, Timothy C., Shiau, Andrew K., Zhou, Huilin, DeGroot, John, Sulman, Erik P., Cavenee, Webster K., Kolodner, Richard D., Chen, Clark C., Furnari, Frank B.
Published in Cancer cell (09.12.2019)
Published in Cancer cell (09.12.2019)
Get full text
Journal Article
Inhibition of Nuclear PTEN Tyrosine Phosphorylation Enhances Glioma Radiation Sensitivity through Attenuated DNA Repair
Ma, Jianhui, Benitez, Jorge A., Li, Jie, Miki, Shunichiro, Ponte de Albuquerque, Claudio, Galatro, Thais, Orellana, Laura, Zanca, Ciro, Reed, Rachel, Boyer, Antonia, Koga, Tomoyuki, Varki, Nissi M., Fenton, Tim R., Nagahashi Marie, Suely Kazue, Lindahl, Erik, Gahman, Timothy C., Shiau, Andrew K., Zhou, Huilin, DeGroot, John, Sulman, Erik P., Cavenee, Webster K., Kolodner, Richard D., Chen, Clark C., Furnari, Frank B.
Published in Cancer cell (13.05.2019)
Published in Cancer cell (13.05.2019)
Get full text
Journal Article
Chemical regulators of epithelial plasticity reveal a nuclear receptor pathway controlling myofibroblast differentiation
Carthy, Jon M, Stöter, Martin, Bellomo, Claudia, Vanlandewijck, Michael, Heldin, Angelos, Morén, Anita, Kardassis, Dimitris, Gahman, Timothy C, Shiau, Andrew K, Bickle, Marc, Zerial, Marino, Heldin, Carl-Henrik, Moustakas, Aristidis
Published in Scientific reports (19.07.2016)
Published in Scientific reports (19.07.2016)
Get full text
Journal Article
Identification and SAR of selective inducible nitric oxide synthase (iNOS) dimerization inhibitors
Gahman, Timothy C., Herbert, Mark R., Lang, Henk, Thayer, Angie, Symons, Kent T., Nguyen, Phan Manh, Massari, Mark E., Dozier, Sara, Zhang, Yan, Sablad, Marciano, Rao, Tadimeti S., Noble, Stewart A., Shiau, Andrew K., Hassig, Christian A.
Published in Bioorganic & medicinal chemistry letters (15.11.2011)
Published in Bioorganic & medicinal chemistry letters (15.11.2011)
Get full text
Journal Article
COMPOSITION AND METHOD FOR ENHANCING PROTEASOME ACTIVITY
TIMOTHY C GAHMAN, DANIEL FINLEY, LEE MIN JAE, RANDALL W KING, LEE BYUNG-HOON
Year of Publication 18.08.2016
Get full text
Year of Publication 18.08.2016
Patent
Inhibition of Nuclear PTEN Tyrosine Phosphorylation Enhances Glioma diation Sensitivity through Attenuated DNA Repair
Ma, Jianhui, Benite, Jorge A., Miki, Shunichiro, Albuquerqu, Claudio Ponte, Galatro, Thais, Orellana, Laura, Zanca, Ciro, Reed, Rachel, Boyer, Antonia, Koga, Tomoyuki, Varki, Nissi M., Fenton, Tim R., Marie, Suely Kazue Nagahashi, Lindahl, Erik, Gahman, Timothy C., Shiau, Andrew K., Zhou, Huilin, DeGroot, John, Sulman, Erik P., Cavenee, Webster K., Kolodner, Richard D., Chen, Clark C., Furnari, Frank B.
Published in Cancer cell (2019)
Published in Cancer cell (2019)
Get full text
Journal Article
Inhibition of inducible nitric oxide synthase expression by a novel small molecule activator of the unfolded protein response
Symons, Kent T, Massari, Mark E, Dozier, Sara J, Nguyen, Phan M, Jenkins, David, Herbert, Mark, Gahman, Timothy C, Noble, Stewart A, Rozenkrants, Natasha, Zhang, Yan, Rao, Tadimeti S, Shiau, Andrew K, Hassig, Christian A
Published in Current chemical genomics (27.09.2008)
Published in Current chemical genomics (27.09.2008)
Get full text
Journal Article
Cell biology. Reversible centriole depletion with an inhibitor of Polo-like kinase 4
Wong, Yao Liang, Anzola, John V, Davis, Robert L, Yoon, Michelle, Motamedi, Amir, Kroll, Ashley, Seo, Chanmee P, Hsia, Judy E, Kim, Sun K, Mitchell, Jennifer W, Mitchell, Brian J, Desai, Arshad, Gahman, Timothy C, Shiau, Andrew K, Oegema, Karen
Published in Science (American Association for the Advancement of Science) (05.06.2015)
Published in Science (American Association for the Advancement of Science) (05.06.2015)
Get full text
Journal Article