Angucyclines: Biosynthesis, mode-of-action, new natural products, and synthesis
Kharel, Madan K, Pahari, Pallab, Shepherd, Micah D, Tibrewal, Nidhi, Nybo, S. Eric, Shaaban, Khaled A, Rohr, Jrgen
Published in Natural product reports (01.02.2012)
Published in Natural product reports (01.02.2012)
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Journal Article
Origins of stereoselectivity in evolved ketoreductases
Noey, Elizabeth L., Tibrewal, Nidhi, Jiménez-Osés, Gonzalo, Osuna, Sílvia, Park, Jiyong, Bond, Carly M., Cascio, Duilio, Liang, Jack, Zhang, Xiyun, Huisman, Gjalt W., Tang, Yi, Houk, Kendall N.
Published in Proceedings of the National Academy of Sciences - PNAS (22.12.2015)
Published in Proceedings of the National Academy of Sciences - PNAS (22.12.2015)
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Journal Article
Selective inhibitors of mTORC1 activate 4EBP1 and suppress tumor growth
Lee, Bianca J., Boyer, Jacob A., Burnett, G. Leslie, Thottumkara, Arun P., Tibrewal, Nidhi, Wilson, Stacy L., Hsieh, Tientien, Marquez, Abby, Lorenzana, Edward G., Evans, James W., Hulea, Laura, Kiss, Gert, Liu, Hui, Lee, Dong, Larsson, Ola, McLaughlan, Shannon, Topisirovic, Ivan, Wang, Zhengping, Wang, Zhican, Zhao, Yongyuan, Wildes, David, Aggen, James B., Singh, Mallika, Gill, Adrian L., Smith, Jacqueline A. M., Rosen, Neal
Published in Nature chemical biology (01.10.2021)
Published in Nature chemical biology (01.10.2021)
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Journal Article
Amalgamation of Nucleosides and Amino Acids in Antibiotic Biosynthesis: Discovery of an l‑Threonine:Uridine-5′-Aldehyde Transaldolase
Barnard-Britson, Sandra, Chi, Xiuling, Nonaka, Koichi, Spork, Anatol P, Tibrewal, Nidhi, Goswami, Anwesha, Pahari, Pallab, Ducho, Christian, Rohr, Jurgen, Van Lanen, Steven G
Published in Journal of the American Chemical Society (14.11.2012)
Published in Journal of the American Chemical Society (14.11.2012)
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Journal Article
Author Correction: Selective inhibitors of mTORC1 activate 4EBP1 and suppress tumor growth
Lee, Bianca J., Boyer, Jacob A., Burnett, G. Leslie, Thottumkara, Arun P., Tibrewal, Nidhi, Wilson, Stacy L., Hsieh, Tientien, Marquez, Abby, Lorenzana, Edward G., Evans, James W., Hulea, Laura, Kiss, Gert, Liu, Hui, Lee, Dong, Larsson, Ola, McLaughlan, Shannon, Topisirovic, Ivan, Wang, Zhengping, Wang, Zhican, Zhao, Yongyuan, Wildes, David, Aggen, James B., Singh, Mallika, Gill, Adrian L., Smith, Jacqueline A. M., Rosen, Neal
Published in Nature chemical biology (01.08.2021)
Published in Nature chemical biology (01.08.2021)
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Journal Article
Author Correction: Selective inhibitors of mTORC1 activate 4EBP1 and suppress tumor growth
Lee, Bianca J., Boyer, Jacob A., Burnett, G. Leslie, Thottumkara, Arun P., Tibrewal, Nidhi, Wilson, Stacy L., Hsieh, Tientien, Marquez, Abby, Lorenzana, Edward G., Evans, James W., Hulea, Laura, Kiss, Gert, Liu, Hui, Lee, Dong, Larsson, Ola, McLaughlan, Shannon, Topisirovic, Ivan, Wang, Zhengping, Wang, Zhican, Zhao, Yongyuan, Wildes, David, Aggen, James B., Singh, Mallika, Gill, Adrian L., Smith, Jacqueline A. M., Rosen, Neal
Published in Nature chemical biology (01.11.2021)
Published in Nature chemical biology (01.11.2021)
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Journal Article
Functional Identification of Valerena-1,10-diene Synthase, a Terpene Synthase Catalyzing a Unique Chemical Cascade in the Biosynthesis of Biologically Active Sesquiterpenes in Valeriana officinalis
Yeo, Yun-Soo, Nybo, S. Eric, Chittiboyina, Amar G., Weerasooriya, Aruna D., Wang, Yan-Hong, Góngora-Castillo, Elsa, Vaillancourt, Brieanne, Buell, C. Robin, DellaPenna, Dean, Celiz, Mary Dawn, Jones, A. Daniel, Wurtele, Eve Syrkin, Ransom, Nick, Dudareva, Natalia, Shaaban, Khaled A., Tibrewal, Nidhi, Chandra, Suman, Smillie, Troy, Khan, Ikhlas A., Coates, Robert M., Watt, David S., Chappell, Joe
Published in The Journal of biological chemistry (01.02.2013)
Published in The Journal of biological chemistry (01.02.2013)
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Journal Article
Biocatalysts for natural product biosynthesis
Tibrewal, Nidhi, Tang, Yi
Published in Annual review of chemical and biomolecular engineering (01.01.2014)
Published in Annual review of chemical and biomolecular engineering (01.01.2014)
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Journal Article
Baeyer–Villiger C–C Bond Cleavage Reaction in Gilvocarcin and Jadomycin Biosynthesis
Tibrewal, Nidhi, Pahari, Pallab, Wang, Guojun, Kharel, Madan K, Morris, Caleb, Downey, Theresa, Hou, Yanpeng, Bugni, Tim S, Rohr, Jürgen
Published in Journal of the American Chemical Society (07.11.2012)
Published in Journal of the American Chemical Society (07.11.2012)
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Journal Article
Abstract IA17: Strategies to target the mTORC1/eIF4F axis in B-cell leukemia and lymphoma
Herzog, Lee-or, Lee, Bianca J., Vo, Thanh-Trang, Chiu, Honyin, Mallya, Sharmila, Fung, Amos, Singh, Mallika, Aggen, James, Tibrewal, Nidhi, Smith, Jacqueline A.M., Wildes, David, Ronai, Ze'ev, Ruggero, Davide, Fruman, David A.
Published in Molecular cancer research (01.10.2020)
Published in Molecular cancer research (01.10.2020)
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Journal Article
Abstract PR04: 4EBP1 reactivation by potent and selective bi-steric inhibitors of mTORC1
Tibrewal, Nidhi, Aggen, James B., Bassan, Abraham I., Burnett, G. Leslie, Evans, Jim, Gliedt, Micah J., Hsieh, Daphne, Kiss, Gert, Lee, Bianca J., Lee, Dong, Lorenzana, Ed, Marquez, Abby, Thottumkara, Arun, Wang, Zhengping, Wilson, Stacy, Zhao, Frances, Goldsmith, Mark, Singh, Mallika, Wildes, Pete, Gill, Adrian L., Smith, Jacqueline A.M.
Published in Molecular cancer research (01.10.2020)
Published in Molecular cancer research (01.10.2020)
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Journal Article
Evaluation of hadacidin analogues
Tibrewal, Nidhi, Elliott, Gregory I.
Published in Bioorganic & medicinal chemistry letters (01.01.2011)
Published in Bioorganic & medicinal chemistry letters (01.01.2011)
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Journal Article
Abstract 4878: RMC-4550, an allosteric inhibitor of SHP2: Synthesis, structure, and anti-tumor activity
Koltun, Elena S., Aay, Naing, Buckl, Andreas, Jogalekar, Ashutosh S., Kiss, Gert, Marquez, Abby, Mellem, Kevin T., Mordec, Kasia, Saldajeno-Concar, Mae, Semko, Chris M., Tibrewal, Nidhi, Tzitzilonis, Christos, Won, Walter, Smith, Jacqueline A., Wilson, Susan E., Nichols, Robert J., Wang, Zhengping, Wilds, David, Singh, Mallika, Gill, Adrian L.
Published in Cancer research (Chicago, Ill.) (01.07.2018)
Published in Cancer research (Chicago, Ill.) (01.07.2018)
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854 HPK1 inhibition relieves suppression downstream of TCR activation to drive enhanced cytokine production and antigen-specific killing, an effect that is further enhanced by immune checkpoint blockade
Singh, Rajesh, Patel, Bindi, Rayaji, Rameshwari, Marubayashi, Sachie, Cho, Sean, Garrido-Shaqfeh, Stefan, Kulusich, Joseph, Meleza, Cesar, Tibrewal, Nidhi, Joice, Thomas, Nareddy, Pradeep, Sharif, Ehesan, Zhao, Sharon, Green, Dave, Leleti, Manmohan, Powers, Jay, Walters, Matt, DiRenzo, Daniel
Published in Journal for immunotherapy of cancer (01.11.2022)
Published in Journal for immunotherapy of cancer (01.11.2022)
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Journal Article
Origins of stereoselectivity in evolved ketoreductases
Noey, Elizabeth L., Tibrewal, Nidhi, Jiménez-Osés, Gonzalo, Osuna, Sílvia, Park, Jiyong, Bond, Carly M., Cascio, Duilio, Liang, Jack, Zhang, Xiyun, Huisman, Gjalt W., Tang, Yi, Houk, Kendall N.
Published in Proceedings of the National Academy of Sciences - PNAS (07.12.2015)
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Published in Proceedings of the National Academy of Sciences - PNAS (07.12.2015)
Journal Article
Roles of the Synergistic Reductive O‑Methyltransferase GilM and of O‑Methyltransferase GilMT in the Gilvocarcin Biosynthetic Pathway
Tibrewal, Nidhi, Downey, Theresa E, Van Lanen, Steven G, Ul Sharif, Ehesan, O’Doherty, George A, Rohr, Jürgen
Published in Journal of the American Chemical Society (01.08.2012)
Published in Journal of the American Chemical Society (01.08.2012)
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Abstract 1367: HPK1 inhibition enhances T cell activation and relieves the immunosuppressive phenotype of inhibitory signals found in the tumor microenvironment
Singh, Rajesh K., Rayaji, Rameshwari, Patel, Bindi, Zhang, Kristen, Marubayashi, Sachie, Cho, Soonweng, Garrido-Shaqfeh, Stefan, Kulusich, Joseph, Meleza, Cesar, Tibrewal, Nidhi, Thomas, Joice, Nareddy, Pradeep, Sharif, Ehesan, Zhao, Sharon, Green, David, Leleti, Manmohan R., Powers, Jay P., DiRenzo, Daniel, Walters, Matthew J.
Published in Cancer research (Chicago, Ill.) (15.06.2022)
Published in Cancer research (Chicago, Ill.) (15.06.2022)
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Journal Article
mTOR 억제제로서의 파라마이신 유사체
THOTTUMKARA ARUN P, KISS GERT, WANG GANG, BURNETT G. LESLIE, WON WALTER, SEMKO CHRISTOPHER, TIBREWAL NIDHI, PITZEN JENNIFER, GLIEDT MICAH JAMES EVANS, AGGEN JAMES BRADLEY, LEE JULIE CHU LI, GILL ADRIAN LIAM
Year of Publication 05.02.2020
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Year of Publication 05.02.2020
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