Search Results - "THOMASON, Jennifer" :: K.UTB vyhledávací portál | TBU Library Retrieval Portal

Discovery of novel N-hydroxy-2-arylisoindoline-4-carboxamides as potent and selective inhibitors of HDAC11

Discovery of novel N-hydroxy-2-arylisoindoline-4-carboxamides as potent and selective inhibitors of HDAC11

by Martin, Matthew W., Lee, Jennifer Y., Lancia, David R., Ng, Pui Yee, Han, Bingsong, Thomason, Jennifer R., Lynes, Maureen S., Marshall, C. Gary, Conti, Chiara, Collis, Alan, Morales, Monica Alvarez, Doshi, Kshama, Rudnitskaya, Aleksandra, Yao, Lili, Zheng, Xiaozhang
Published in Bioorganic & medicinal chemistry letters (01.07.2018)

Get full text

Journal Article

Diazine Indole Acetic Acids as Potent, Selective, and Orally Bioavailable Antagonists of Chemoattractant Receptor Homologous Molecule Expressed on Th2 Cells (CRTH2) for the Treatment of Allergic Inflammatory Diseases

Diazine Indole Acetic Acids as Potent, Selective, and Orally Bioavailable Antagonists of Chemoattractant Receptor Homologous Molecule Expressed on Th2 Cells (CRTH2) for the Treatment of Allergic Inflammatory Diseases

by Kaila, Neelu, Huang, Adrian, Moretto, Alessandro, Follows, Bruce, Janz, Kristin, Lowe, Michael, Thomason, Jennifer, Mansour, Tarek S, Hubeau, Cedric, Page, Karen, Morgan, Paul, Fish, Susan, Xu, Xin, Williams, Cara, Saiah, Eddine
Published in Journal of medicinal chemistry (14.06.2012)

Get full text

Journal Article

Potent, selective, and orally bioavailable matrix metalloproteinase-13 inhibitors for the treatment of osteoarthritis

Potent, selective, and orally bioavailable matrix metalloproteinase-13 inhibitors for the treatment of osteoarthritis

by Hu, Yonghan, Xiang, Jason S., DiGrandi, Martin J., Du, Xuemei, Ipek, Manus, Laakso, Leif M., Li, Jianchang, Li, Wei, Rush, Thomas S., Schmid, Jean, Skotnicki, Jerauld S., Tam, Steve, Thomason, Jennifer R., Wang, Qin, Levin, Jeremy I.
Published in Bioorganic & medicinal chemistry (15.12.2005)

Get full text

Journal Article

Inhibition of Tpl2 kinase and TNFα production with quinoline-3-carbonitriles for the treatment of rheumatoid arthritis

Inhibition of Tpl2 kinase and TNFα production with quinoline-3-carbonitriles for the treatment of rheumatoid arthritis

by Hu, Yonghan, Green, Neal, Gavrin, Lori K., Janz, Kristin, Kaila, Neelu, Li, Huan-Qiu, Thomason, Jennifer R., Cuozzo, John W., Hall, J. Perry, Hsu, Sang, Nickerson-Nutter, Cheryl, Telliez, Jean-Baptiste, Lin, Lih-Ling, Tam, Steve
Published in Bioorganic & medicinal chemistry letters (01.12.2006)

Get full text

Journal Article

Winter swarming behavior by the exotic cladoceran Daphnia lumholtzi Sars, 1885 in a Kentucky (USA) reservoir

Winter swarming behavior by the exotic cladoceran Daphnia lumholtzi Sars, 1885 in a Kentucky (USA) reservoir

by Beaver, John, Renicker, Thomas, Tausz, Claudia, Young, Jade, Thomason, Jennifer, Wolf, Zachary, Russell, Amber, Cherry, Mac, Scotese, Kyle, Koenig, Dawn
Published in Bioinvasions records (01.03.2018)

Get full text

Journal Article

Continued exploration of biphenylsulfonamide scaffold as a platform for aggrecanase-1 inhibition

Continued exploration of biphenylsulfonamide scaffold as a platform for aggrecanase-1 inhibition

by Hu, Yonghan, Xing, Li, Thomason, Jennifer R., Xiang, Jason, Ipek, Manus, Guler, Satenig, Li, Huanqiu, Sabatini, Joshua, Chockalingam, Priya, Reifenberg, Erica, Sheldon, Richard, Morris, Elisabeth A., Georgiadis, Katy E., Tam, Steve
Published in Bioorganic & medicinal chemistry letters (15.11.2011)

Get full text

Journal Article

Synthesis and SAR of highly selective MMP-13 inhibitors

Synthesis and SAR of highly selective MMP-13 inhibitors

by Li, Jianchang, Rush, Thomas S., Li, Wei, DeVincentis, Dianne, Du, Xuemei, Hu, Yonghan, Thomason, Jennifer R., Xiang, Jason S., Skotnicki, Jerauld S., Tam, Steve, Cunningham, Kristina M., Chockalingam, Priya S., Morris, Elisabeth A., Levin, Jeremy I.
Published in Bioorganic & medicinal chemistry letters (15.11.2005)

Get full text

Journal Article

Inhibition of Tpl2 kinase and TNF-α production with 1,7-naphthyridine-3-carbonitriles: Synthesis and structure–activity relationships

Inhibition of Tpl2 kinase and TNF-α production with 1,7-naphthyridine-3-carbonitriles: Synthesis and structure–activity relationships

by Gavrin, Lori Krim, Green, Neal, Hu, Yonghan, Janz, Kristin, Kaila, Neelu, Li, Huan-Qiu, Tam, Steve Y., Thomason, Jennifer R., Gopalsamy, Ariamala, Ciszewski, Greg, Cuozzo, John W., Hall, J. Perry, Hsu, Sang, Telliez, Jean-Baptiste, Lin, Lih-Ling
Published in Bioorganic & medicinal chemistry letters (01.12.2005)

Get full text

Journal Article

3,4-Disubstituted benzofuran P1′ MMP-13 inhibitors: Optimization of selectivity and reduction of protein binding

3,4-Disubstituted benzofuran P1′ MMP-13 inhibitors: Optimization of selectivity and reduction of protein binding

by Li, Wei, Hu, Yonghan, Li, Jianchang, Thomason, Jennifer R., DeVincentis, Dianne, Du, Xuemei, Wu, Junjun, Hotchandani, Rajeev, Rush, Thomas S., Skotnicki, Jerauld S., Tam, Steve, Chockalingam, Priya S., Morris, Elisabeth A., Levin, Jeremy I.
Published in Bioorganic & medicinal chemistry letters (15.08.2009)

Get full text

Journal Article

Synthesis and biological evaluation of biphenylsulfonamide carboxylate aggrecanase-1 inhibitors

Synthesis and biological evaluation of biphenylsulfonamide carboxylate aggrecanase-1 inhibitors

by Xiang, Jason S., Hu, Yonghan, Rush, Thomas S., Thomason, Jennifer R., Ipek, Manus, Sum, Phaik-Eng, Abrous, Leila, Sabatini, Joshua J., Georgiadis, Katy, Reifenberg, Erica, Majumdar, Manas, Morris, Elisabeth A., Tam, Steve
Published in Bioorganic & medicinal chemistry letters (15.01.2006)

Get full text

Journal Article

Discovery of Clinical Candidate 1‑{[(2S,3S,4S)‑3-Ethyl-4-fluoro-5-oxopyrrolidin-2-yl]methoxy}-7-methoxyisoquinoline-6-carboxamide (PF-06650833), a Potent, Selective Inhibitor of Interleukin‑1 Receptor Associated Kinase 4 (IRAK4), by Fragment-Based Drug Design

Discovery of Clinical Candidate 1‑{[(2S,3S,4S)‑3-Ethyl-4-fluoro-5-oxopyrrolidin-2-yl]methoxy}-7-methoxyisoquinoline-6-carboxamide (PF-06650833), a Potent, Selective Inhibitor of Interleukin‑1 Receptor Associated Kinase 4 (IRAK4), by Fragment-Based Drug Design

by Lee, Katherine L, Ambler, Catherine M, Anderson, David R, Boscoe, Brian P, Bree, Andrea G, Brodfuehrer, Joanne I, Chang, Jeanne S, Choi, Chulho, Chung, Seungwon, Curran, Kevin J, Day, Jacqueline E, Dehnhardt, Christoph M, Dower, Ken, Drozda, Susan E, Frisbie, Richard K, Gavrin, Lori K, Goldberg, Joel A, Han, Seungil, Hegen, Martin, Hepworth, David, Hope, Heidi R, Kamtekar, Satwik, Kilty, Iain C, Lee, Arthur, Lin, Lih-Ling, Lovering, Frank E, Lowe, Michael D, Mathias, John P, Morgan, Heidi M, Murphy, Elizabeth A, Papaioannou, Nikolaos, Patny, Akshay, Pierce, Betsy S, Rao, Vikram R, Saiah, Eddine, Samardjiev, Ivan J, Samas, Brian M, Shen, Marina W. H, Shin, Julia H, Soutter, Holly H, Strohbach, Joseph W, Symanowicz, Peter T, Thomason, Jennifer R, Trzupek, John D, Vargas, Richard, Vincent, Fabien, Yan, Jiangli, Zapf, Christoph W, Wright, Stephen W
Published in Journal of medicinal chemistry (13.07.2017)

Get full text

Journal Article

Discovery of Isoquinolinone Indole Acetic Acids as Antagonists of Chemoattractant Receptor Homologous Molecule Expressed on Th2 Cells (CRTH2) for the Treatment of Allergic Inflammatory Diseases

Discovery of Isoquinolinone Indole Acetic Acids as Antagonists of Chemoattractant Receptor Homologous Molecule Expressed on Th2 Cells (CRTH2) for the Treatment of Allergic Inflammatory Diseases

by Kaila, Neelu, Follows, Bruce, Leung, Louis, Thomason, Jennifer, Huang, Adrian, Moretto, Alessandro, Janz, Kristin, Lowe, Michael, Mansour, Tarek S, Hubeau, Cedric, Page, Karen, Morgan, Paul, Fish, Susan, Xu, Xin, Williams, Cara, Saiah, Eddine
Published in Journal of medicinal chemistry (27.02.2014)

Get full text

Journal Article

Indole cytosolic phospholipase A(2) alpha inhibitors: Discovery and in vitro and in vivo characterization of 4-{3-[5-chloro-2-(2-{[(3,4-dichlorobenzyl)sulfonyl]amino}ethyl)-1-(diphenylmethyl)-1H-indol-3-yl]propyl}benzoic acid, efipladib

Indole cytosolic phospholipase A(2) alpha inhibitors: Discovery and in vitro and in vivo characterization of 4-{3-[5-chloro-2-(2-{[(3,4-dichlorobenzyl)sulfonyl]amino}ethyl)-1-(diphenylmethyl)-1H-indol-3-yl]propyl}benzoic acid, efipladib

by McKew, John C., Lee, Katherine L., Shen, Marina W. H., Thakker, Paresh, Foley, Megan A., Behnke, Mark L., Hu, Baihua, Sum, Fuk-Wah, Tam, Steve, Hu, Yonghan, Chen, Lihren, Kirincich, Steven J., Michalak, Ronald, Thomason, Jennifer, Ipek, Manus, Wu, Kun, Wooder, Lane, Ramarao, Manjunath K., Murphy, Elizabeth A., Goodwin, Debra G., Albert, Leo, Xu, Xin, Donahue, Frances, Ku, M. Sherry, Keith, James, Nickerson-Nutter, Cheryl L., Abraham, William M., Williams, Cara, Hegen, Martin, Clark, James D.
Published in Journal of medicinal chemistry (26.06.2008)

Get full text

Journal Article

Indole Cytosolic Phospholipase A2 α Inhibitors: Discovery and in Vitro and in Vivo Characterization of 4-{3-[5-Chloro-2-(2-{[(3,4-dichlorobenzyl)sulfonyl]amino}ethyl)-1-(diphenylmethyl)-1H-indol-3-yl]propyl}benzoic Acid, Efipladib

Indole Cytosolic Phospholipase A2 α Inhibitors: Discovery and in Vitro and in Vivo Characterization of 4-{3-[5-Chloro-2-(2-{[(3,4-dichlorobenzyl)sulfonyl]amino}ethyl)-1-(diphenylmethyl)-1H-indol-3-yl]propyl}benzoic Acid, Efipladib

by McKew, John C, Lee, Katherine L, Shen, Marina W. H, Thakker, Paresh, Foley, Megan A, Behnke, Mark L, Hu, Baihua, Sum, Fuk-Wah, Tam, Steve, Hu, Yonghan, Chen, Lihren, Kirincich, Steven J, Michalak, Ronald, Thomason, Jennifer, Ipek, Manus, Wu, Kun, Wooder, Lane, Ramarao, Manjunath K, Murphy, Elizabeth A, Goodwin, Debra G, Albert, Leo, Xu, Xin, Donahue, Frances, Ku, M. Sherry, Keith, James, Nickerson-Nutter, Cheryl L, Abraham, William M, Williams, Cara, Hegen, Martin, Clark, James D
Published in Journal of medicinal chemistry (26.06.2008)

Get full text

Journal Article

HDAC 억제제로서의 이소인돌린

HDAC 억제제로서의 이소인돌린

by RUDNITSKAYA ALEKSANDRA, THOMASON JENNIFER R, HAN BINGSONG, ZHENG XIAOZHANG, MARTIN MATTHEW W, NG PUI YEE, LANCIA JR. DAVID R
Year of Publication 13.04.2021

Get full text

Patent

Inhibitors of Tumor Progression Loci-2 (Tpl2) Kinase and Tumor Necrosis Factor α (TNF-α) Production: Selectivity and in Vivo Antiinflammatory Activity of Novel 8-Substituted-4-anilino-6-aminoquinoline-3-carbonitriles

Inhibitors of Tumor Progression Loci-2 (Tpl2) Kinase and Tumor Necrosis Factor α (TNF-α) Production: Selectivity and in Vivo Antiinflammatory Activity of Novel 8-Substituted-4-anilino-6-aminoquinoline-3-carbonitriles

by Green, Neal, Hu, Yonghan, Janz, Kristin, Li, Huan-Qiu, Kaila, Neelu, Guler, Satenig, Thomason, Jennifer, Joseph-McCarthy, Diane, Tam, Steve Y, Hotchandani, Rajeev, Wu, Junjun, Huang, Adrian, Wang, Qin, Leung, Louis, Pelker, Jefferey, Marusic, Suzana, Hsu, Sang, Telliez, Jean-Baptiste, Hall, J. Perry, Cuozzo, John W, Lin, Lih-Ling
Published in Journal of medicinal chemistry (20.09.2007)

Get full text

Journal Article

Perspectives on Teacher Leadership: Implications for Practice and Teacher Leadership Development

Perspectives on Teacher Leadership: Implications for Practice and Teacher Leadership Development

by Thomason, Jennifer, Sanzo, Karen L, Scribner, Jay Paredes
Published in International Journal of Educational Leadership Preparation (2023)

Get full text

Journal Article

Synthesis and biological evaluation of ((4-keto)-phenoxy)methyl biphenyl-4-sulfonamides: A class of potent aggrecanase-1 inhibitors

Synthesis and biological evaluation of ((4-keto)-phenoxy)methyl biphenyl-4-sulfonamides: A class of potent aggrecanase-1 inhibitors

by Hopper, Darrin W., Vera, Matthew D., How, David, Sabatini, Joshua, Xiang, Jason S., Ipek, Manus, Thomason, Jennifer, Hu, Yonghan, Feyfant, Eric, Wang, Qin, Georgiadis, Katy E., Reifenberg, Erica, Sheldon, Richard T., Keohan, Cristin C., Majumdar, Manas K., Morris, Elisabeth A., Skotnicki, Jerauld, Sum, Phaik-Eng
Published in Bioorganic & medicinal chemistry letters (01.05.2009)

Get full text

Journal Article

Identification of a novel class of selective Tpl2 kinase inhibitors: 4-Alkylamino-[1,7]naphthyridine-3-carbonitriles

Identification of a novel class of selective Tpl2 kinase inhibitors: 4-Alkylamino-[1,7]naphthyridine-3-carbonitriles

by Kaila, Neelu, Green, Neal, Li, Huan-Qiu, Hu, Yonghan, Janz, Kristin, Gavrin, Lori Krim, Thomason, Jennifer, Tam, Steve, Powell, Dennis, Cuozzo, John, Hall, J. Perry, Telliez, Jean-Baptiste, Hsu, Sang, Nickerson-Nutter, Cheryl, Wang, Qin, Lin, Lih-Ling
Published in Bioorganic & medicinal chemistry (01.10.2007)

Get full text

Journal Article

HDAC8 억제제로서의 알파-신나미드 화합물 및 조성물

HDAC8 억제제로서의 알파-신나미드 화합물 및 조성물

by RUDNITSKAYA ALEKSANDRA, LIU CUIXIAN, THOMASON JENNIFER R, HAN BINGSONG, LANCIA DAVID R. JR, ZHENG XIAOZHANG, MARTIN MATTHEW W, NG PUI YEE, BAIR KENNETH W, BARCZAK NICHOLAS, ZABLOCKI MARY MARGARET
Year of Publication 10.11.2017

Get full text

Patent

1
2
3
4
5
6
7
8
9
10
11
Next
[12]