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Part 3: Synthesis and biological evaluation of some analogs of the antitumor agents, 2-{4-[(7-chloro-2-quinoxalinyl)oxy]phenoxy}propionic acid, and 2-{4-[(7-bromo-2-quinolinyl)oxy]phenoxy}propionic acid
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Synthetic modification of the 2-oxypropionic acid moiety in 2-{4-[(7-chloro-2-quinoxalinyl)oxy]phenoxy}propionic acid (XK469), and consequent antitumor effects. Part 4
Hazeldine, Stuart T., Polin, Lisa, Kushner, Juiwanna, White, Kathryn, Corbett, Thomas H., Horwitz, Jerome P.
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Total Structures of Cryptophycins, Potent Antitumor Depsipeptides from the Blue-Green Alga Nostoc sp. Strain GSV 224
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Published in Journal of the American Chemical Society (01.06.1994)
Published in Journal of the American Chemical Society (01.06.1994)
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Structure determination, conformational analysis, chemical stability studies, and antitumor evaluation of the cryptophycins. Isolation of 18 new analogs from Nostoc sp. strain GSV 224
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Isolation, Structure Determination, and Biological Activity of Dolastatin 12 and Lyngbyastatin 1 from Lyngbya majuscula/Schizothrix calcicola Cyanobacterial Assemblages
Harrigan, George G, Yoshida, Wesley Y, Moore, Richard E, Nagle, Dale G, Park, Peter U, Biggs, Jason, Paul, Valerie J, Mooberry, Susan L, Corbett, Thomas H, Valeriote, Fred A
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Published in Journal of natural products (Washington, D.C.) (01.10.1998)
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Biological evaluation of cryptophycin 52 fragment A analogues: Effect of the multidrug resistance ATP binding cassette transporters on antitumor activity
Al-Awar, Rima S, Corbett, Thomas H, Ray, James E, Polin, Lisa, Kennedy, Joseph H, Wagner, Margaret M, Williams, Daniel C
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Published in Molecular cancer therapeutics (01.09.2004)
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Total Structure Determination of Apratoxin A, a Potent Novel Cytotoxin from the Marine Cyanobacterium Lyngbya majuscula
LUESCH, Hendrik, YOSHIDA, Wesley Y., MOORE, Richard E., PAUL, Valerie J., CORBETT, Thomas H.
Published in Journal of the American Chemical Society (13.06.2001)
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Isolation of Dolastatin 10 from the Marine Cyanobacterium Symploca Species VP642 and Total Stereochemistry and Biological Evaluation of Its Analogue Symplostatin 1
Luesch, Hendrik, Moore, Richard E, Paul, Valerie J, Mooberry, Susan L, Corbett, Thomas H
Published in Journal of natural products (Washington, D.C.) (01.07.2001)
Published in Journal of natural products (Washington, D.C.) (01.07.2001)
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Design, Synthesis, and Biological Evaluation of Analogues of the Antitumor Agent, 2-{4-[(7-Chloro-2-quinoxalinyl)oxy]phenoxy}propionic Acid (XK469)
Hazeldine, Stuart T, Polin, Lisa, Kushner, Juiwanna, Paluch, Jennifer, White, Kathryn, Edelstein, Matthew, Palomino, Eduardo, Corbett, Thomas H, Horwitz, Jerome P
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Published in Journal of medicinal chemistry (24.05.2001)
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Preclinical efficacy of thioxanthone SR271425 against transplanted solid tumors of mouse and human origin
Corbett, T H, Panchapor, C, Polin, L, Lowichik, N, Pugh, S, White, K, Kushner, J, Meyer, J, Czarnecki, J, Chinnukroh, S, Edelstein, M, LoRusso, P, Heilbrun, L, Horwitz, J P, Grieshaber, C, Perni, R, Wentland, M, Coughlin, S, Elenbaas, S, Philion, R, Rake, J
Published in Investigational new drugs (01.02.1999)
Published in Investigational new drugs (01.02.1999)
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II. Synthesis and Biological Evaluation of Some Bioisosteres and Congeners of the Antitumor Agent, 2-{4-[(7-Chloro-2-quinoxalinyl)oxy]phenoxy}propionic Acid (XK469)
Hazeldine, Stuart T, Polin, Lisa, Kushner, Juiwanna, White, Kathryn, Bouregeois, Nicole M, Crantz, Brianna, Palomino, Eduardo, Corbett, Thomas H, Horwitz, Jerome P
Published in Journal of medicinal chemistry (04.07.2002)
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Discovery of cryptophycin-1 and BCN-183577 : Examples of strategies and problems in the detection of antitumor activity in mice
CORBETT, T. H, VALERIOTE, F. A, WENTLAND, M, GOLAKOTI, T, HETZEL, C, OGINO, J, PATTERSON, G, MOORE, R, DEMCHIK, L, LOWICHIK, N, POLIN, L, PANCHAPOR, C, PUGH, S, WHITE, K, KUSHNER, J, RAKE, J
Published in Investigational new drugs (01.01.1997)
Published in Investigational new drugs (01.01.1997)
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Symplostatin 3, a New Dolastatin 10 Analogue from the Marine Cyanobacterium Symploca sp. VP452
Luesch, Hendrik, Yoshida, Wesley Y, Moore, Richard E, Paul, Valerie J, Mooberry, Susan L, Corbett, Thomas H
Published in Journal of natural products (Washington, D.C.) (01.01.2002)
Published in Journal of natural products (Washington, D.C.) (01.01.2002)
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Cryptophycins-309, 249 and other cryptophycin analogs: preclinical efficacy studies with mouse and human tumors
Liang, Jian, Moore, Richard E, Moher, Eric D, Munroe, John E, Al-awar, Rima S, Hay, David A, Varie, David L, Zhang, Tony Y, Aikins, James A, Martinelli, Michael J, Shih, Chuan, Ray, James E, Gibson, Lowell L, Vasudevan, Vasu, Polin, Lisa, White, Kathryn, Kushner, Juiwanna, Simpson, Chiab, Pugh, Susan, Corbett, Thomas H
Published in Investigational new drugs (01.06.2005)
Published in Investigational new drugs (01.06.2005)
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Synthesis and biological evaluation of conformationally constrained analogs of the antitumor agents XK469 and SH80. Part 5
Hazeldine, Stuart T., Polin, Lisa, Kushner, Juiwanna, White, Kathryn, Corbett, Thomas H., Horwitz, Jerome P.
Published in Bioorganic & medicinal chemistry (01.04.2006)
Published in Bioorganic & medicinal chemistry (01.04.2006)
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A Convergent Approach to Cryptophycin 52 Analogues: Synthesis and Biological Evaluation of a Novel Series of Fragment A Epoxides and Chlorohydrins
Al-awar, Rima S, Ray, James E, Schultz, Richard M, Andis, Sherri L, Kennedy, Joseph H, Moore, Richard E, Liang, Jian, Golakoti, Trimurtulu, Subbaraju, Gottumukkala V, Corbett, Thomas H
Published in Journal of medicinal chemistry (03.07.2003)
Published in Journal of medicinal chemistry (03.07.2003)
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