Tumor‐infiltrating endothelial cells and endothelial precursor cells in inflammatory breast cancer
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Published in International journal of cancer (20.05.2002)
Published in International journal of cancer (20.05.2002)
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Angiogenic potential of perivascularly delivered aFGF in a porcine model of chronic myocardial ischemia
Lopez, John J, Edelman, Elazer R, Stamler, Alon, Hibberd, Mark G, Prasad, Pottumarthi, Thomas, Kenneth A, Disalvo, Jerry, Caputo, Ronald P, Carrozza, Joseph P, Douglas, Pamela S, Sellke, Frank W, Simons, Michael
Published in American journal of physiology. Heart and circulatory physiology (01.03.1998)
Published in American journal of physiology. Heart and circulatory physiology (01.03.1998)
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Vascular endothelial growth factor stimulates angiogenesis without improving collateral blood flow following hindlimb ischemia in rabbits
Hershey, James C, Baskin, Elizabeth P, Corcoran, Halea A, Bett, Andrew, Dougherty, Nancy M, Gilberto, David B, Mao, Xianzhi, Thomas, Kenneth A, Cook, Jacquelynn J
Published in Heart and vessels (01.07.2003)
Published in Heart and vessels (01.07.2003)
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Paracrine Expression of a Native Soluble Vascular Endothelial Growth Factor Receptor Inhibits Tumor Growth, Metastasis, and Mortality Rate
Goldman, Corey K., Kendall, Richard L., Cabrera, Gustavo, Soroceanu, Liliana, Heike, Yuji, Gillespie, G. Yancey, Siegal, Gene P., Mao, Xianzhi, Bett, Andrew J., Huckle, William R., Thomas, Kenneth A., Curiel, David T.
Published in Proceedings of the National Academy of Sciences - PNAS (21.07.1998)
Published in Proceedings of the National Academy of Sciences - PNAS (21.07.1998)
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Synthesis and Initial SAR Studies of 3,6-Disubstituted Pyrazolo[1,5- a]pyrimidines: A New Class of KDR Kinase Inhibitors
Fraley, Mark E., Hoffman, William F., Rubino, Robert S., Hungate, Randall W., Tebben, Andrew J., Rutledge, Ruth Z., McFall, Rosemary C., Huckle, William R., Kendall, Richard L., Coll, Kathleen E., Thomas, Kenneth A.
Published in Bioorganic & medicinal chemistry letters (07.10.2002)
Published in Bioorganic & medicinal chemistry letters (07.10.2002)
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Dynamic Contrast-Enhanced MRI Measurements of Passive Permeability through Blood Retinal Barrier in Diabetic Rats
Berkowitz, Bruce A, Roberts, Robin, Luan, Hongmei, Peysakhov, Jamie, Mao, Xianzhi, Thomas, Kenneth A
Published in Investigative ophthalmology & visual science (01.07.2004)
Published in Investigative ophthalmology & visual science (01.07.2004)
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Potent N-(1,3-Thiazol-2-yl)pyridin-2-amine Vascular Endothelial Growth Factor Receptor Tyrosine Kinase Inhibitors with Excellent Pharmacokinetics and Low Affinity for the hERG Ion Channel
Bilodeau, Mark T, Balitza, Adrienne E, Koester, Timothy J, Manley, Peter J, Rodman, Leonard D, Buser-Doepner, Carolyn, Coll, Kathleen E, Fernandes, Christine, Gibbs, Jackson B, Heimbrook, David C, Huckle, William R, Kohl, Nancy, Lynch, Joseph J, Mao, Xianzhi, McFall, Rosemary C, McLoughlin, Debra, Miller-Stein, Cynthia M, Rickert, Keith W, Sepp-Lorenzino, Laura, Shipman, Jennifer M, Subramanian, Raju, Thomas, Kenneth A, Wong, Bradley K, Yu, Sean, Hartman, George D
Published in Journal of medicinal chemistry (02.12.2004)
Published in Journal of medicinal chemistry (02.12.2004)
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Optimization of a pyrazolo[1,5- a]pyrimidine class of KDR kinase inhibitors: improvements in physical properties enhance cellular activity and pharmacokinetics
Fraley, Mark E., Rubino, Robert S., Hoffman, William F., Hambaugh, Scott R., Arrington, Kenneth L., Hungate, Randall W., Bilodeau, Mark T., Tebben, Andrew J., Rutledge, Ruth Z., Kendall, Richard L., McFall, Rosemary C., Huckle, William R., Coll, Kathleen E., Thomas, Kenneth A.
Published in Bioorganic & medicinal chemistry letters (16.12.2002)
Published in Bioorganic & medicinal chemistry letters (16.12.2002)
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Vascular Endothelial Growth Factor Receptor KDR Tyrosine Kinase Activity Is Increased by Autophosphorylation of Two Activation Loop Tyrosine Residues
Kendall, R L, Rutledge, R Z, Mao, X, Tebben, A J, Hungate, R W, Thomas, K A
Published in The Journal of biological chemistry (05.03.1999)
Published in The Journal of biological chemistry (05.03.1999)
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Purification and Characterization of a Naturally Occurring Vascular Endothelial Growth Factor · Placenta Growth Factor Heterodimer (∗)
DiSalvo, Jerry, Bayne, Marvin L., Conn, Greg, Kwok, Perry W., Trivedi, Prashant G., Soderman, Denis D., Palisi, Thomas M., Sullivan, Kathleen A., Thomas, Kenneth A.
Published in The Journal of biological chemistry (31.03.1995)
Published in The Journal of biological chemistry (31.03.1995)
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Optimization of the indolyl quinolinone class of KDR (VEGFR-2) kinase inhibitors: effects of 5-amido- and 5-sulphonamido-indolyl groups on pharmacokinetics and hERG binding
Fraley, Mark E., Arrington, Kenneth L., Buser, Carolyn A., Ciecko, Patrice A., Coll, Kathleen E., Fernandes, Christine, Hartman, George D., Hoffman, William F., Lynch, Joseph J., McFall, Rosemary C., Rickert, Keith, Singh, Romi, Smith, Sheri, Thomas, Kenneth A., Wong, Bradley K.
Published in Bioorganic & medicinal chemistry letters (19.01.2004)
Published in Bioorganic & medicinal chemistry letters (19.01.2004)
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Design and synthesis of 3,7-diarylimidazopyridines as inhibitors of the VEGF-receptor KDR
ZHICAI WU, FRALEY, Mark E, BIN SHI, SEPP-LORENZINO, Laura, THOMAS, Kenneth A, BILODEAU, Mark T, KAUFMAN, Mildred L, TASBER, Edward S, BALITZA, Adrienne E, HARTMAN, George D, COLL, Kathleen E, RICKERT, Keith, SHIPMAN, Jennifer
Published in Bioorganic & medicinal chemistry letters (23.02.2004)
Published in Bioorganic & medicinal chemistry letters (23.02.2004)
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The discovery of N-(1,3-thiazol-2-yl)pyridin-2-amines as potent inhibitors of KDR kinase
Bilodeau, Mark T., Rodman, Leonard D., McGaughey, Georgia B., Coll, Kathleen E., Koester, Timothy J., Hoffman, William F., Hungate, Randall W., Kendall, Richard L., McFall, Rosemary C., Rickert, Keith W., Rutledge, Ruth Z., Thomas, Kenneth A.
Published in Bioorganic & medicinal chemistry letters (07.06.2004)
Published in Bioorganic & medicinal chemistry letters (07.06.2004)
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Property-Based Design of KDR Kinase Inhibitors
Fraley, Mark E, Hoffman, William F, Arrington, Kenneth L, Hungate, Randy W, Hartman, George D, McFall, Rosemary C, Coll, Kathleen E, Rickert, Keith, Thomas, Kenneth A, McGaughey, Georgia B
Published in Current medicinal chemistry (01.03.2004)
Published in Current medicinal chemistry (01.03.2004)
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