Reevaluating the Substrate Specificity of the L‑Type Amino Acid Transporter (LAT1)
Chien, Huan-Chieh, Colas, Claire, Finke, Karissa, Springer, Seth, Stoner, Laura, Zur, Arik A., Venteicher, Brooklynn, Campbell, Jerome, Hall, Colton, Flint, Andrew, Augustyn, Evan, Hernandez, Christopher, Heeren, Nathan, Hansen, Logan, Anthony, Abby, Bauer, Justine, Fotiadis, Dimitrios, Schlessinger, Avner, Giacomini, Kathleen M., Thomas, Allen A.
Published in Journal of medicinal chemistry (23.08.2018)
Published in Journal of medicinal chemistry (23.08.2018)
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LAT1 activity of carboxylic acid bioisosteres: Evaluation of hydroxamic acids as substrates
Zur, Arik A., Chien, Huan-Chieh, Augustyn, Evan, Flint, Andrew, Heeren, Nathan, Finke, Karissa, Hernandez, Christopher, Hansen, Logan, Miller, Sydney, Lin, Lawrence, Giacomini, Kathleen M., Colas, Claire, Schlessinger, Avner, Thomas, Allen A.
Published in Bioorganic & medicinal chemistry letters (15.10.2016)
Published in Bioorganic & medicinal chemistry letters (15.10.2016)
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Osmium-Catalyzed Dihydroxylation of Olefins in Acidic Media: Old Process, New Tricks
Dupau, Philippe, Epple, Robert, Thomas, Allen A., Fokin, Valery V., Sharpless, K. Barry
Published in Advanced synthesis & catalysis (01.06.2002)
Published in Advanced synthesis & catalysis (01.06.2002)
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Describing inhibitor specificity for the amino acid transporter LAT1 from metainference simulations
Hutchinson, Keino, Silva, Dina Buitrago, Bohlke, Joshua, Clausen, Chase, Thomas, Allen A., Bonomi, Massimiliano, Schlessinger, Avner
Published in Biophysical journal (06.12.2022)
Published in Biophysical journal (06.12.2022)
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Synthesis of ribavirin 1,2,3- and 1,2,4-triazolyl analogs with changes at the amide and cytotoxicity in breast cancer cell lines
Way, Hannah, Roh, Joshua, Venteicher, Brooklynn, Chandra, Surabhi, Thomas, Allen A.
Published in Nucleosides, nucleotides & nucleic acids (2023)
Published in Nucleosides, nucleotides & nucleic acids (2023)
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Experimental and Theoretical Kinetic Isotope Effects for Asymmetric Dihydroxylation. Evidence Supporting a Rate-Limiting “(3 + 2)” Cycloaddition
DelMonte, Albert J, Haller, Jan, Houk, K. N, Sharpless, K. Barry, Singleton, Daniel A, Strassner, Thomas, Thomas, Allen A
Published in Journal of the American Chemical Society (15.10.1997)
Published in Journal of the American Chemical Society (15.10.1997)
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l-Type amino acid transporter 1 activity of 1,2,3-triazolyl analogs of l-histidine and l-tryptophan
Hall, Colton, Wolfe, Hannah, Wells, Alyssa, Chien, Huan-Chieh, Colas, Claire, Schlessinger, Avner, Giacomini, Kathleen M., Thomas, Allen A.
Published in Bioorganic & medicinal chemistry letters (15.08.2019)
Published in Bioorganic & medicinal chemistry letters (15.08.2019)
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Evaluation of Rhodanine Indolinones as AANAT Inhibitors
Hagemeister, Mackenzie, Hamilton, Luke, Wandrey, Nicole, Hill, Mackinzi, Mounce, Emery, Mosel, Noah, Lytle, Katie, Redinger, Makenna, Boley, Jake, Fancher, Nathan, Haynes, Alexis, Fill, Ianna, Cole, Philip A., Hill, Evan, Moxley, Michael A., Thomas, Allen A.
Published in ChemMedChem (02.01.2024)
Published in ChemMedChem (02.01.2024)
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LAT-1 activity of meta-substituted phenylalanine and tyrosine analogs
Augustyn, Evan, Finke, Karissa, Zur, Arik A., Hansen, Logan, Heeren, Nathan, Chien, Huan-Chieh, Lin, Lawrence, Giacomini, Kathleen M., Colas, Claire, Schlessinger, Avner, Thomas, Allen A.
Published in Bioorganic & medicinal chemistry letters (01.06.2016)
Published in Bioorganic & medicinal chemistry letters (01.06.2016)
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Cellular fatty acid level regulates the effect of tolylfluanid on mitochondrial dysfunction and insulin sensitivity in C2C12 skeletal myotubes
Davis, A'Lexxus F., Thomas, Allen A., Shorter, Kimberly S., Brown, Stephan L., Baumgarner, Bradley L.
Published in Biochemical and biophysical research communications (28.10.2018)
Published in Biochemical and biophysical research communications (28.10.2018)
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The Effects of Prodrug Size and a Carbonyl Linker on l‐Type Amino Acid Transporter 1‐Targeted Cellular and Brain Uptake
Venteicher, Brooklynn, Merklin, Kasey, Ngo, Huy X., Chien, Huan‐Chieh, Hutchinson, Keino, Campbell, Jerome, Way, Hannah, Griffith, Joseph, Alvarado, Cesar, Chandra, Surabhi, Hill, Evan, Schlessinger, Avner, Thomas, Allen A.
Published in ChemMedChem (03.03.2021)
Published in ChemMedChem (03.03.2021)
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Spirocyclic β‑Site Amyloid Precursor Protein Cleaving Enzyme 1 (BACE1) Inhibitors: From Hit to Lowering of Cerebrospinal Fluid (CSF) Amyloid β in a Higher Species
Hunt, Kevin W, Cook, Adam W, Watts, Ryan J, Clark, Christopher T, Vigers, Guy, Smith, Darin, Metcalf, Andrew T, Gunawardana, Indrani W, Burkard, Michael, Cox, April A, Geck Do, Mary K, Dutcher, Darrin, Thomas, Allen A, Rana, Sumeet, Kallan, Nicholas C, DeLisle, Robert K, Rizzi, James P, Regal, Kelly, Sammond, Douglas, Groneberg, Robert, Siu, Michael, Purkey, Hans, Lyssikatos, Joseph P, Marlow, Allison, Liu, Xingrong, Tang, Tony P
Published in Journal of medicinal chemistry (25.04.2013)
Published in Journal of medicinal chemistry (25.04.2013)
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Discovery of 7‑Tetrahydropyran-2-yl Chromans: β‑Site Amyloid Precursor Protein Cleaving Enzyme 1 (BACE1) Inhibitors That Reduce Amyloid β‑Protein (Aβ) in the Central Nervous System
Thomas, Allen A, Hunt, Kevin W, Volgraf, Matthew, Watts, Ryan J, Liu, Xingrong, Vigers, Guy, Smith, Darin, Sammond, Douglas, Tang, Tony P, Rhodes, Susan P, Metcalf, Andrew T, Brown, Karin D, Otten, Jennifer N, Burkard, Michael, Cox, April A, Do, Mary K. Geck, Dutcher, Darrin, Rana, Sumeet, DeLisle, Robert K, Regal, Kelly, Wright, Albion D, Groneberg, Robert, Scearce-Levie, Kimberly, Siu, Michael, Purkey, Hans E, Lyssikatos, Joseph P, Gunawardana, Indrani W
Published in Journal of medicinal chemistry (13.02.2014)
Published in Journal of medicinal chemistry (13.02.2014)
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8‑Tetrahydropyran-2-yl Chromans: Highly Selective Beta-Site Amyloid Precursor Protein Cleaving Enzyme 1 (BACE1) Inhibitors
Thomas, Allen A, Hunt, Kevin W, Newhouse, Brad, Watts, Ryan J, Liu, Xingrong, Vigers, Guy, Smith, Darin, Rhodes, Susan P, Brown, Karin D, Otten, Jennifer N, Burkard, Michael, Cox, April A, Geck Do, Mary K, Dutcher, Darrin, Rana, Sumeet, DeLisle, Robert K, Regal, Kelly, Wright, Albion D, Groneberg, Robert, Liao, Jiangpeng, Scearce-Levie, Kimberly, Siu, Michael, Purkey, Hans E, Lyssikatos, Joseph P
Published in Journal of medicinal chemistry (11.12.2014)
Published in Journal of medicinal chemistry (11.12.2014)
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Synthesis, characterization, and PK/PD studies of a series of spirocyclic pyranochromene BACE1 inhibitors
Volgraf, Matthew, Chan, Lina, Huestis, Malcolm P., Purkey, Hans E., Burkard, Michael, Geck Do, Mary, Harris, Julie, Hunt, Kevin W., Liu, Xingrong, Lyssikatos, Joseph P., Rana, Sumeet, Thomas, Allen A., Vigers, Guy P.A., Siu, Michael
Published in Bioorganic & medicinal chemistry letters (01.06.2014)
Published in Bioorganic & medicinal chemistry letters (01.06.2014)
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Mechanistic pharmacokinetic-pharmacodynamic modeling of BACE1 inhibition in monkeys: development of a predictive model for amyloid precursor protein processing
Liu, Xingrong, Wong, Harvey, Scearce-Levie, Kimberly, Watts, Ryan J, Coraggio, Melis, Shin, Young G, Peng, Kun, Wildsmith, Kristin R, Atwal, Jasvinder K, Mango, Jason, Schauer, Stephen P, Regal, Kelly, Hunt, Kevin W, Thomas, Allen A, Siu, Michael, Lyssikatos, Joseph, Deshmukh, Gauri, Hop, Cornelis E C A
Published in Drug metabolism and disposition (01.07.2013)
Published in Drug metabolism and disposition (01.07.2013)
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Journal Article
Synthesis, in vitro and in vivo activity of thiamine antagonist transketolase inhibitors
Thomas, Allen A., Le Huerou, Y., De Meese, J., Gunawardana, Indrani, Kaplan, Tomas, Romoff, Todd T., Gonzales, Stephen S., Condroski, Kevin, Boyd, Steven A., Ballard, Josh, Bernat, Bryan, DeWolf, Walter, Han, May, Lee, Patrice, Lemieux, Christine, Pedersen, Robin, Pheneger, Jed, Poch, Greg, Smith, Darin, Sullivan, Francis, Weiler, Solly, Wright, S. Kirk, Lin, Jie, Brandhuber, Barb, Vigers, Guy
Published in Bioorganic & medicinal chemistry (15.03.2008)
Published in Bioorganic & medicinal chemistry (15.03.2008)
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Journal Article
Non-charged thiamine analogs as inhibitors of enzyme transketolase
Thomas, Allen A., De Meese, J., Le Huerou, Y., Boyd, Steven A., Romoff, Todd T., Gonzales, Steven S., Gunawardana, Indrani, Kaplan, Tomas, Sullivan, Francis, Condroski, Kevin, Lyssikatos, Joseph P., Aicher, Thomas D., Ballard, Josh, Bernat, Bryan, DeWolf, Walter, Han, May, Lemieux, Christine, Smith, Darin, Weiler, Solly, Wright, S. Kirk, Vigers, Guy, Brandhuber, Barb
Published in Bioorganic & medicinal chemistry (15.01.2008)
Published in Bioorganic & medicinal chemistry (15.01.2008)
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