Synthesis of Selective Estrogen Receptor Degrader GDC-0810 via Stereocontrolled Assembly of a Tetrasubstituted All-Carbon Olefin
Savage, Scott, McClory, Andrew, Zhang, Haiming, Cravillion, Theresa, Lim, Ngiap-Kie, Masui, Colin, Robinson, Sarah J, Han, Chong, Ochs, Christoph, Rege, Pankaj D, Gosselin, Francis
Published in Journal of organic chemistry (05.10.2018)
Published in Journal of organic chemistry (05.10.2018)
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Journal Article
Synthesis of PI3K inhibitor GDC-0077 via a stereocontrolled N-arylation of α-amino acids
Han, Chong, Kelly, Sean M., Cravillion, Theresa, Savage, Scott J., Nguyen, Tina, Gosselin, Francis
Published in Tetrahedron (09.08.2019)
Published in Tetrahedron (09.08.2019)
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Journal Article
Palladium-Catalyzed Site-Selective Amidation of Dichloroazines
Young, Ian S, Glass, Anna-Lena, Cravillion, Theresa, Han, Chong, Zhang, Haiming, Gosselin, Francis
Published in Organic letters (06.07.2018)
Published in Organic letters (06.07.2018)
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Journal Article
Highly Stereoselective Synthesis of Tetrasubstituted Acyclic All-Carbon Olefins via Enol Tosylation and Suzuki–Miyaura Coupling
Li, Beryl X, Le, Diane N, Mack, Kyle A, McClory, Andrew, Lim, Ngiap-Kie, Cravillion, Theresa, Savage, Scott, Han, Chong, Collum, David B, Zhang, Haiming, Gosselin, Francis
Published in Journal of the American Chemical Society (09.08.2017)
Published in Journal of the American Chemical Society (09.08.2017)
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Journal Article
Synthesis of a Selective Estrogen Receptor Degrader via a Stereospecific Elimination Approach
Lim, Ngiap-Kie, Cravillion, Theresa, Savage, Scott, McClory, Andrew, Han, Chong, Zhang, Haiming, DiPasquale, Antonio, Gosselin, Francis
Published in Organic letters (16.02.2018)
Published in Organic letters (16.02.2018)
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Journal Article
Stereocontrolled Synthesis of Arylomycin-Based Gram-Negative Antibiotic GDC-5338
Wong, Nicholas, Petronijević, Filip, Hong, Allen Y, Linghu, Xin, Kelly, Sean M, Hou, Haiyun, Cravillion, Theresa, Lim, Ngiap-Kie, Robinson, Sarah J, Han, Chong, Molinaro, Carmela, Sowell, C. Gregory, Gosselin, Francis
Published in Organic letters (15.11.2019)
Published in Organic letters (15.11.2019)
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Journal Article
Development of an Efficient Manufacturing Process for Reversible Bruton’s Tyrosine Kinase Inhibitor GDC-0853
Zhang, Haiming, Cravillion, Theresa, Lim, Ngiap-Kie, Tian, Qingping, Beaudry, Danial, Defreese, Jessica L, Fettes, Alec, James, Philippe, Linder, David, Malhotra, Sushant, Han, Chong, Angelaud, Remy, Gosselin, Francis
Published in Organic process research & development (17.08.2018)
Published in Organic process research & development (17.08.2018)
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Journal Article
PROCESS FOR PREPARING BTK INHIBITORS
TIAN QINGPING, ALEXANDER GMEHLING, SUSHANT MALHOTRA, DANIAL BEAUDRY, THERESA CRAVILLION, ZHANG HAIMING, LIM NGIAP-KIE, ALEC FETTES, FRANCIS GOSSELIN, STEFAN BACHMANN
Year of Publication 18.03.2021
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Year of Publication 18.03.2021
Patent
PROCESS FOR PREPARING BTK INHIBITORS
MALHOTRA, SUSHANT, GOSSELIN, FRANCIS, LIM, NGIAP-KIE, BACHMANN, STEPHAN, CRAVILLION, THERESA, TIAN, QINGPING, ZHANG, HAIMING, BEAUDRY, DANIAL, GMEHLING, ALEXANDER, FETTES, ALEC
Year of Publication 19.09.2023
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Year of Publication 19.09.2023
Patent
PROCESS FOR PREPARING BTK INHIBITORS
BACHMANN, Stephan, CRAVILLION, Theresa, ZHANG, Haiming, GMEHLING, Alexander, FETTES, Alec, BEAUDRY, Danial, MALHOTRA, Sushant, GOSSELIN, Francis, LIM, Ngiap-Kie, TIAN, Qingping
Year of Publication 10.08.2023
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Year of Publication 10.08.2023
Patent
Process for preparing BTK inhibitors
Beaudry, Danial, Fettes, Alec, Cravillion, Theresa, Malhotra, Sushant, Tian, Qingping, Gosselin, Francis, Lim, Ngiap-Kie, Gmehling, Alexander, Zhang, Haiming, Bachmann, Stephan
Year of Publication 30.05.2023
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Year of Publication 30.05.2023
Patent