Aurora Kinase Inhibitors Based on the Imidazo[1,2-a]pyrazine Core: Fluorine and Deuterium Incorporation Improve Oral Absorption and Exposure
Kerekes, Angela D, Esposite, Sara J, Doll, Ronald J, Tagat, Jayaram R, Yu, Tao, Xiao, Yushi, Zhang, Yonglian, Prelusky, Dan B, Tevar, Seema, Gray, Kimberly, Terracina, Gaby A, Lee, Suining, Jones, Jennifer, Liu, Ming, Basso, Andrea D, Smith, Elizabeth B
Published in Journal of medicinal chemistry (13.01.2011)
Published in Journal of medicinal chemistry (13.01.2011)
Get full text
Journal Article
암을 치료하기 위한 항-CCR8 항체
SELBY MARK J, LEE JOHN K, ADELAKUN OLUFEMI A, CAMPBELL JOSEPH RICHARD, MCDONALD BRYAN, LEE PETER SUNG KEUN, MESKO PAUL BLAINE, LU KAI, GREENAWALT DANIELLE M, LIANG LINDA, JAIN RENU, LAN RUTH YIN ZONG, RAJPAL ARVIND, TERRACINA GABY A, FINDEISEN FELIX, SAMBANTHAMOORTHY SHARMILA, BARMAN ISHITA, SIEMERS NATHAN O, DIONG SJ JIAN ZHE, STROP PAVEL, WANG XI TAO, JHATAKIA AMY D
Year of Publication 29.11.2022
Get full text
Year of Publication 29.11.2022
Patent
ANTI-IDO ANTIBODY AND USES THEREOF
MESKO, Paul Blaine, WANG, Xi-Tao, CHUNTHARAPAI, Anan, SPIRES, JR., Thomas E, TERRACINA, Gaby A
Year of Publication 30.12.2021
Get full text
Year of Publication 30.12.2021
Patent
ANTI-IDO ANTIBODY AND USES THEREOF
MESKO, Paul Blaine, WANG, Xi-Tao, CHUNTHARAPAI, Anan, SPIRES, Thomas E, TERRACINA, Gaby A
Year of Publication 11.06.2020
Get full text
Year of Publication 11.06.2020
Patent
ANTI-CCR8 ANTIBODIES FOR TREATING CANCER
Wang, Xi-Tao, McDonald, Bryan, Rajpal, Arvind, Diong, SJ Jian Zhe, Greenawalt, Danielle M, Mesko, Paul, Lee, John K, Sambanthamoorthy, Sharmila, Selby, Mark J, Lee, Peter S.K, Siemers, Nathan O, Jain, Renu, Lan, Ruth Yin-Zong, Jhatakia, Amy D, Lu, Kai, Barman, Ishita, Findeisen, Felix, Adelakun, Olufemi A, Campbell, Joseph, Terracina, Gaby A, Liang, Linda, Strop, Pavel
Year of Publication 20.04.2023
Get full text
Year of Publication 20.04.2023
Patent
ANTI-CCR8 ANTIBODIES FOR TREATING CANCER
MESKO, Paul Blaine, SIEMERS, Nathan O, LEE, John K, DIONG, SJ Jian Zhe, STROP, Pavel, SELBY, Mark J, RAJPAL, Arvind, JHATAKIA, Amy D, BARMAN, Ishita, FINDEISEN, Felix, MCDONALD, Bryan, GREENAWALT, Danielle M, WANG, Xi-Tao, SAMBANTHAMOORTHY, Sharmila, LEE, Peter Sung Keun, JAIN, Renu, LU, Kai, LAN, Ruth Yin-Zong, TERRACINA, Gaby A, ADELAKUN, Olufemi A, LIANG, Linda, CAMPBELL, Joseph Richard
Year of Publication 08.02.2023
Get full text
Year of Publication 08.02.2023
Patent
Anti-CCR8 antibodies for treating cancer
MESKO, Paul Blaine, SIEMERS, Nathan O, LEE, John K, DIONG, SJ Jian Zhe, STROP, Pavel, SELBY, Mark J, RAJPAL, Arvind, JHATAKIA, Amy D, BARMAN, Ishita, FINDEISEN, Felix, MCDONALD, Bryan, GREENAWALT, Danielle M, WANG, Xi-Tao, SAMBANTHAMOORTHY, Sharmila, LEE, Peter Sung Keun, JAIN, Renu, LU, Kai, LAN, Ruth Yin-Zong, TERRACINA, Gaby A, ADELAKUN, Olufemi A, LIANG, Linda, CAMPBELL, Joseph Richard
Year of Publication 24.11.2022
Get full text
Year of Publication 24.11.2022
Patent
Anti-ccr8 antibodies for treating cancer
FINDEISEN Felix, LEE Peter Sung Keun, SAMBANTHAMOORTHY Sharmila, CAMPBELL Joseph Richard, SIEMERS Nathan O, TERRACINA Gaby A, LEE John K, WANG Xi-Tao, MESKO Paul Blaine, MCDONALD Bryan, STROP Pavel, BARMAN Ishita, DIONG SJ Jian Zhe, RAJPAL Arvind, JHATAKIA Amy D, SELBY Mark J, LIANG Linda, GREENAWALT Danielle M, JAIN Renu, LU Kai, LAN Ruth Yin-Zong, ADELAKUN Olufemi A
Year of Publication 01.11.2022
Get full text
Year of Publication 01.11.2022
Patent
ANTI-CCR8 ANTIBODIES FOR TREATING CANCER
LIANG, LINDA, SELBY, MARK J, SIEMERS, NATHAN O, GREENAWALT, DANIELLE M, SAMBANTHAMOORTHY, SHARMILA, BARMAN, ISHITA, LAN, RUTH YIN-ZONG, LU, KAI, FINDEISEN, FELIX, MCDONALD, BRYAN, RAJPAL, ARVIND, LEE, JOHN K, JHATAKIA, AMY D, TERRACINA, GABY A, LEE, PETER SUNG KEUN, STROP, PAVEL, ADELAKUN, OLUFEMI A, JAIN, RENU, DIONG, SJ JIAN ZHE, WANG, XI-TAO, CAMPBELL, JOSEPH RICHARD, MESKO, PAUL BLAINE
Year of Publication 30.09.2021
Get full text
Year of Publication 30.09.2021
Patent
ANTI-CCR8 ANTIBODIES FOR TREATING CANCER
MESKO, Paul Blaine, SIEMERS, Nathan O, LEE, John K, DIONG, SJ Jian Zhe, STROP, Pavel, SELBY, Mark J, RAJPAL, Arvind, JHATAKIA, Amy D, BARMAN, Ishita, FINDEISEN, Felix, MCDONALD, Bryan, GREENAWALT, Danielle M, WANG, Xi-Tao, SAMBANTHAMOORTHY, Sharmila, LEE, Peter Sung Keun, JAIN, Renu, LU, Kai, LAN, Ruth Yin-Zong, TERRACINA, Gaby A, ADELAKUN, Olufemi A, LIANG, Linda, CAMPBELL, Joseph Richard
Year of Publication 30.09.2021
Get full text
Year of Publication 30.09.2021
Patent
ANTICUERPOS ANTI-CCR8 PARA EL TRATAMIENTO DEL CANCER
MESKO, Paul Blaine, SIEMERS, Nathan O, LEE, John K, DIONG, SJ Jian Zhe, STROP, Pavel, SELBY, Mark J, RAJPAL, Arvind, JHATAKIA, Amy D, BARMAN, Ishita, FINDEISEN, Felix, MCDONALD, Bryan, GREENAWALT, Danielle M, WANG, Xi-Tao, SAMBANTHAMOORTHY, Sharmila, LEE, Peter Sung Keun, JAIN, Renu, LU, Kai, LAN, Ruth Yin-Zong, TERRACINA, Gaby A, ADELAKUN, Olufemi A, LIANG, Linda, CAMPBELL, Joseph Richard
Year of Publication 19.05.2023
Get full text
Year of Publication 19.05.2023
Patent
Anticuerpos anti-ccr8 para el tratamiento del cáncer
Renu JAIN, Bryan MCDONALD, Linda LIANG, Mark J. SELBY, Felix FINDEISEN, Sharmila SAMBANTHAMOORTHY, Peter Sung Keun LEE, Ishita BARMAN, 2. Olufemi A. ADELAKUN, Joseph Richard CAMPBELL, Pavel STROP, Xi-Tao WANG, Paul Blaine MESKO, Kai LU, SJ Jian Zhe DIONG, John K. LEE, Nathan O. SIEMERS, Gaby A. TERRACINA, Amy D. JHATAKIA, Ruth Yin-Zong LAN, Arvind RAJPAL, Danielle M GREENAWALT
Year of Publication 17.03.2023
Get full text
Year of Publication 17.03.2023
Patent
ANTICORPOS ANTI-CCR8 PARA TRATAMENTO DE CÂNCER
JOHN K. LEE, NATHAN O. SIEMERS, AMY D JHATAKIA, FELIX FINDEISEN, OLUFEMI A. ADELAKUN, JOSEPH RICHARD CAMPBELL, SJ JIAN ZHE DIONG, MARK J. SELBY, BRYAN MCDONALD, DANIELLE M. GREENAWALT, LINDA LIANG, ARVIND RAJPAL, PAVEL STROP, RENU JAIN, XI-TAO WANG, ISHITA BARMAN, SHARMILA SAMBANTHAMOORTHY, PAUL BLAINE MESKO, KAI LU, PETER SUNG KEUN LEE, RUTH YIN-ZONG LAN, GABY A. TERRACINA
Year of Publication 31.01.2023
Get full text
Year of Publication 31.01.2023
Patent
Anticuerpos anti-ccr8 para el tratamiento del cáncer
MESKO, Paul Blaine, SIEMERS, Nathan O, LEE, John K, DIONG, SJ Jian Zhe, STROP, Pavel, SELBY, Mark J, RAJPAL, Arvind, JHATAKIA, Amy D, BARMAN, Ishita, FINDEISEN, Felix, MCDONALD, Bryan, GREENAWALT, Danielle M, WANG, Xi-Tao, SAMBANTHAMOORTHY, Sharmila, LEE, Peter Sung Keun, JAIN, Renu, LU, Kai, LAN, Ruth Yin-Zong, TERRACINA, Gaby A, ADELAKUN, Olufemi A, LIANG, Linda, CAMPBELL, Joseph Richard
Year of Publication 11.10.2022
Get full text
Year of Publication 11.10.2022
Patent
ANTI-CCR8 ANTIBODIES FOR TREATING CANCER
LEE Peter Sung Keun, FINDEISEN Felix, SAMBANTHAMOORTHY Sharmila, CAMPBELL Joseph Richard, SIEMERS Nathan O, LAN Ruth Yin-zong, TERRACINA Gaby A, LEE John K, WANG Xi-tao, MESKO Paul Blaine, STROP Pavel, DIONG Sj Jian Zhe, MCDONALD Bryan, BARMAN Ishita, RAJPAL Arvind, SELBY Mark J, JHATAKIA Amy D, LIANG Linda, GREENAWALT Danielle M, JAIN Renu, LU Kai, ADELAKUN Olufemi A
Year of Publication 07.10.2022
Get full text
Year of Publication 07.10.2022
Patent
ANTICUERPOS ANTI-CCR8 PARA EL TRATAMIENTO DEL CÁNCER
LIANG, LINDA, SELBY, MARK J, SIEMERS, NATHAN O, GREENAWALT, DANIELLE M, SAMBANTHAMOORTHY, SHARMILA, ZONG - ADELAKUN, OLUFEMI A, BARMAN, ISHITA, LU, KAI, FINDEISEN, FELIX, RAJPAL, ARVIND, LEE, JOHN K, MDONALD, BRYAN, JHATAKIA, AMY D, TERRACINA, GABY A, LEE, PETER SUNG KEUN, STROP, PAVEL, JAIN, RENU, WANG, XI, TAO - DIONG, SJ JIAN ZHE, LAN, RUTH YIN, CAMPBELL, JOSEPH RICHARD, MESKO, PAUL BLAINE
Year of Publication 22.06.2022
Get full text
Year of Publication 22.06.2022
Patent
Anti-CCR8 antibodies for treating cancer
LIANG, LINDA, SELBY, MARK J, SIEMERS, NATHAN O, GREENAWALT, DANIELLE M, SAMBANTHAMOORTHY, SHARMILA, BARMAN, ISHITA, LAN, RUTH YIN-ZONG, LU, KAI, FINDEISEN, FELIX, MCDONALD, BRYAN, RAJPAL, ARVIND, LEE, JOHN K, JHATAKIA, AMY D, TERRACINA, GABY A, LEE, PETER SUNG KEUN, STROP, PAVEL, ADELAKUN, OLUFEMI A, JAIN, RENU, WANG, XI-TAO, DIONG, SJ JIAN ZHE, CAMPBELL, JOSEPH RICHARD, MESKO, PAUL BLAINE
Year of Publication 16.01.2022
Get full text
Year of Publication 16.01.2022
Patent