Identification of Atuveciclib (BAY 1143572), the First Highly Selective, Clinical PTEFb/CDK9 Inhibitor for the Treatment of Cancer
Lücking, Ulrich, Scholz, Arne, Lienau, Philip, Siemeister, Gerhard, Kosemund, Dirk, Bohlmann, Rolf, Briem, Hans, Terebesi, Ildiko, Meyer, Kirstin, Prelle, Katja, Denner, Karsten, Bömer, Ulf, Schäfer, Martina, Eis, Knut, Valencia, Ray, Ince, Stuart, von Nussbaum, Franz, Mumberg, Dominik, Ziegelbauer, Karl, Klebl, Bert, Choidas, Axel, Nussbaumer, Peter, Baumann, Matthias, Schultz‐Fademrecht, Carsten, Rühter, Gerd, Eickhoff, Jan, Brands, Michael
Published in ChemMedChem (08.11.2017)
Published in ChemMedChem (08.11.2017)
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Changing for the Better: Discovery of the Highly Potent and Selective CDK9 Inhibitor VIP152 Suitable for Once Weekly Intravenous Dosing for the Treatment of Cancer
Lücking, Ulrich, Kosemund, Dirk, Böhnke, Niels, Lienau, Philip, Siemeister, Gerhard, Denner, Karsten, Bohlmann, Rolf, Briem, Hans, Terebesi, Ildiko, Bömer, Ulf, Schäfer, Martina, Ince, Stuart, Mumberg, Dominik, Scholz, Arne, Izumi, Raquel, Hwang, Stuart, von Nussbaum, Franz
Published in Journal of medicinal chemistry (12.08.2021)
Published in Journal of medicinal chemistry (12.08.2021)
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Discovery of IRAK4 Inhibitors BAY1834845 (Zabedosertib) and BAY1830839
Bothe, Ulrich, Günther, Judith, Nubbemeyer, Reinhard, Siebeneicher, Holger, Ring, Sven, Bömer, Ulf, Peters, Michaele, Rausch, Alexandra, Denner, Karsten, Himmel, Herbert, Sutter, Andreas, Terebesi, Ildiko, Lange, Martin, Wengner, Antje M., Guimond, Nicolas, Thaler, Tobias, Platzek, Johannes, Eberspächer, Uwe, Schäfer, Martina, Steuber, Holger, Zollner, Thomas M., Steinmeyer, Andreas, Schmidt, Nicole
Published in Journal of medicinal chemistry (25.01.2024)
Published in Journal of medicinal chemistry (25.01.2024)
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Abstract 984: Identification of potent and highly selective PTEFb inhibitor BAY 1251152 for the treatment of cancer: from p.o. to i.v. application via scaffold hops
Luecking, Ulrich T., Scholz, Arne, Kosemund, Dirk, Bohlmann, Rolf, Briem, Hans, Lienau, Philip, Siemeister, Gerhard, Terebesi, Ildiko, Meyer, Kirstin, Prelle, Katja, Valencia, Ray, Ince, Stuart, Nussbaum, Franz von, Mumberg, Dominik, Ziegelbauer, Karl, Brands, Michael
Published in Cancer research (Chicago, Ill.) (01.07.2017)
Published in Cancer research (Chicago, Ill.) (01.07.2017)
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Abstract 2828: Rapid identification of potent and highly selective, oral PTEFb Inhibitor BAY 1143572 with first in class potential
Luecking, Ulrich TJ, Scholz, Arne, Lienau, Philip, Siemeister, Gerhard, Kosemund, Dirk, Bohlmann, Rolf, Eis, Knut, Gnoth, Mark, Terebesi, Ildiko, Meyer, Kirstin, Prelle, Katja, Valencia, Ray, Ince, Stuart, von Nussbaum, Franz, Mumberg, Dominik, Ziegelbauer, Karl, Klebl, Bert, Choidas, Axel, Nussbaumer, Peter, Baumann, Matthias, Schultz-Fademrecht, Carsten, Ruehter, Gerd, Eickhoff, Jan, Brands, Michael
Published in Cancer research (Chicago, Ill.) (01.08.2015)
Published in Cancer research (Chicago, Ill.) (01.08.2015)
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Year of Publication 28.01.2019
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Year of Publication 28.01.2019
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DIEFENBACH KONSTANZE, TEREBESI ILDIKO, FUNKE ADRIAN, SCHAEFERS MATTHIAS, GENERAL SASCHA
Year of Publication 31.08.2011
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Year of Publication 31.08.2011
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PRODRUG DERIVATIVES OF SUBSTITUTED TRIAZOLOPYRIDINES
LIENAU PHILIP, BIERER DONALD, TEREBESI ILDIKO, SCHULZE VOLKER, WENGNER ANTJE MARGRET, SIEMEISTER GERHARD, KOSEMUND DIRK, STOECKIGT DETLEF, BRUENING MICHAEL, LERCHEN HANS GEORG, KRENZ URSULA, LUECKING ULRICH
Year of Publication 19.02.2016
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Year of Publication 19.02.2016
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18-METHYL-6,7-METHYLENE-3-OXO-17-PREGN-4-ENE-21,17β-CARBOLACTONES, PHARMACEUTICAL PREPARATIONS CONTAINING SAID COMPOUNDS AND USE THEREOF IN THE TREATMENT OF ENDOMETRIOSIS
GALLUS NORBERT, TEREBESI ILDIKO, KUHNKE JOACHIM, BOHLMANN ROLF, HUEBNER JAN, GASHAW ISABELLA, NUBBEMEYER REINHARD, FISCHER OLIVER MARTIN
Year of Publication 09.07.2014
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Year of Publication 09.07.2014
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ESTRADIOL-CONTAINING DRUG DELIVERY SYSTEM
DIEFENBACH KONSTANZE, TEREBESI ILDIKO, FUNKE ADRIAN, ALINCIC KUNZ SOFIA, HOLLER THOMAS, ZURTH CHRISTIAN, SCHAEFERS MATTHIAS, GENERAL SASCHA
Year of Publication 30.11.2010
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Year of Publication 30.11.2010
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