Evaluation of the Anti-Schistosoma mansoni Activity of Thiosemicarbazones and Thiazoles
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Published in Antimicrobial Agents and Chemotherapy (01.01.2014)
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Antitumor and immunomodulatory activities of thiosemicarbazones and 1,3-Thiazoles in Jurkat and HT-29 cells
dos Santos, Thiago André R, da Silva, Aline Caroline, Silva, Elany Barbosa, Gomes, Paulo André Teixeira de Moraes, Espíndola, José Wanderlan Pontes, Cardoso, Marcos Veríssimo de Oliveira, Moreira, Diogo Rodrigo Magalhaes, Leite, Ana Cristina Lima, Pereira, Valéria R.A
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Published in Biomedicine & pharmacotherapy (01.08.2016)
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PA‑Int5: An isatin‑thiosemicarbazone derivative that exhibits anti‑nociceptive and anti‑inflammatory effects in Swiss mice
Da Fonseca, Aldilane Goncalves, De Sena Fernandes Ribeiro Dantas, Luzia Leiros, Rodrigues, Joquebede Pereira, Da Costa Alencar Filho, Marco Polo, De Melo Rego, Moacyr Jesus Barreto, Da Rocha Pitta, Maira Galdino, De Moraes Gomes, Paulo Andre Teixeira, De Melo Silva, Vanessa Gouveia, Leite, Ana Cristina Lima, Furtado, Allanny Alves, De Freitas Fernandes Pedrosa, Matheus, Gavioli, Elaine Cristina, Lemos, Telma Maria Araujo Moura
Published in Biomedical reports (01.07.2021)
Published in Biomedical reports (01.07.2021)
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Phthalimido-thiazoles as building blocks and their effects on the growth and morphology of Trypanosoma cruzi
Gomes, Paulo André Teixeira de Moraes, Oliveira, Arsênio Rodrigues, Cardoso, Marcos Veríssimo de Oliveira, Santiago, Edna de Farias, Barbosa, Miria de Oliveira, de Siqueira, Lucianna Rabelo Pessoa, Moreira, Diogo Rodrigo Magalhães, Bastos, Tanira Matutino, Brayner, Fábio André, Soares, Milena Botelho Pereira, Mendes, Andresa Pereira de Oliveira, de Castro, Maria Carolina Accioly Brelaz, Pereira, Valéria Rego Alves, Leite, Ana Cristina Lima
Published in European journal of medicinal chemistry (23.03.2016)
Published in European journal of medicinal chemistry (23.03.2016)
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Thiazolyl-isatin derivatives: Synthesis, in silico studies, in vitro biological profile against breast cancer cells, mRNA expression, P-gp modulation, and interactions of Akt2 and VIM proteins
Freitas, Luiz Alberto Barros, Sousa, Carolina, Lima, Beatriz Silva, Duarte, Denise, Gomes, Paulo André Teixeira de Moraes, Ramos, Camila Gabriela Costa, Costa, Valécia de Cássia Mendonça, Pitta, Maira Galdino da Rocha, Rêgo, Moacyr Jesus Barreto de Melo, de Simone, Carlos Alberto, Videira, Mafalda, Leite, Ana Cristina Lima
Published in Chemico-biological interactions (01.05.2024)
Published in Chemico-biological interactions (01.05.2024)
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Phthalimido-thiazole as privileged scaffold: activity against immature and adult worms of Schistosoma mansoni
de Oliveira, Sheilla Andrade, de Oliveira Barbosa, Miria, Filho, Carlos André Laranjeira Miranda, Oliveira, Arsênio Rodrigues, de Sousa, Fabiano Amaro, de Farias Santiago, Edna, de Oliveira Filho, Gevanio Bezerra, de Moraes Gomes, Paulo André Teixeira, da Conceição, Juliana Maria, Brayner, Fábio André, Alves, Luiz Carlos, Leite, Ana Cristina Lima
Published in Parasitology research (1987) (01.07.2018)
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Novel phthalimide derivatives with TNF-α and IL-1β expression inhibitory and apoptotic inducing properties
Coêlho, Lucas Cunha Duarte, Cardoso, Marcos Veríssimo de Oliveira, Moreira, Diogo Rodrigo Magalhães, Gomes, Paulo André Teixeira de Moraes, Cavalcanti, Suellen Melo Tibúrcio, Oliveira, Arsenio Rodrigues, Filho, Gevanio Bezerra de Oliveira, Siqueira, Lucianna Rabelo Pessoa de, Barbosa, Miria de Oliveira, Borba, Elizabeth Fernanda de Oliveira, Silva, Teresinha Gonçalves da, Kaskow, Belinda, Karimi, Mahdad, Abraham, Lawrence J, Leite, Ana Cristina Lima
Published in MedChemComm (2014)
Published in MedChemComm (2014)
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Identification of Novel Zika Virus Inhibitors: A Screening using Thiosemicarbazones and Thiazoles Templates
de Moraes Gomes, Paulo André Teixeira, Barros Freitas, Luiz Alberto, Pessoa Siqueira, Luciana Rabelo, da Conceição, Juliana Maria, Dos Santos, Ignes Regina, Pinto, Aline Ferreira, de Melo Silva, Vanessa Gouveia, Nunes, Janine Siqueira, de Oliveira Cardoso, Marcos Veríssimo, Pena, Lindomar José, Lima Leite, Ana Cristina
Published in Current topics in medicinal chemistry (01.01.2023)
Published in Current topics in medicinal chemistry (01.01.2023)
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New 1,3-thiazole derivatives and their biological and ultrastructural effects on Trypanosoma cruzi
de Moraes Gomes, Paulo André Teixeira, de Oliveira Barbosa, Miria, Farias Santiago, Edna, de Oliveira Cardoso, Marcos Veríssimo, Capistrano Costa, Natáli Tereza, Hernandes, Marcelo Zaldini, Moreira, Diogo Rodrigo Magalhães, da Silva, Aline Caroline, dos Santos, Thiago André Ramos, Pereira, Valéria Rêgo Alves, Brayner dos Santosd, Fábio André, do Nascimento Pereira, Glaécia Aparecida, Ferreira, Rafaela Salgado, Leite, Ana Cristina Lima
Published in European journal of medicinal chemistry (04.10.2016)
Published in European journal of medicinal chemistry (04.10.2016)
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Conformational restriction of aryl thiosemicarbazones produces potent and selective anti-Trypanosoma cruzi compounds which induce apoptotic parasite death
Magalhaes Moreira, Diogo Rodrigo, de Oliveira, Ana Daura Travassos, Teixeira de Moraes Gomes, Paulo André, de Simone, Carlos Alberto, Villela, Filipe Silva, Ferreira, Rafaela Salgado, da Silva, Aline Caroline, dos Santos, Thiago André Ramos, Brelaz de Castro, Maria Carolina Accioly, Pereira, Valéria Rego Alves, Leite, Ana Cristina Lima
Published in European journal of medicinal chemistry (21.03.2014)
Published in European journal of medicinal chemistry (21.03.2014)
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Dual Parasiticidal Activities of Phthalimides: Synthesis and Biological Profile against Trypanosoma cruzi and Plasmodium falciparum
Teixeira de Moraes Gomes, Paulo André, Veríssimo de Oliveira Cardoso, Marcos, Santos, Ignes Regina, Amaro de Sousa, Fabiano, Conceição, Juliana Maria, Gouveia de Melo Silva, Vanessa, Duarte, Denise, Pereira, Raquel, Oliveira, Rafael, Nogueira, Fátima, Alves, Luiz Carlos, Brayner, Fabio André, Silva Santos, Aline Caroline, Rêgo Alves Pereira, Valéria, Lima Leite, Ana Cristina
Published in ChemMedChem (18.11.2020)
Published in ChemMedChem (18.11.2020)
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Synthesis, anticancer activity and mechanism of action of new thiazole derivatives
de Santana, Temístocles Italo, Barbosa, Miria de Oliveira, Gomes, Paulo André Teixeira de Moraes, da Cruz, Anne Cecília Nascimento, da Silva, Teresinha Gonçalves, Leite, Ana Cristina Lima
Published in European journal of medicinal chemistry (20.01.2018)
Published in European journal of medicinal chemistry (20.01.2018)
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Multi-target compounds acting in cancer progression: Focus on thiosemicarbazone, thiazole and thiazolidinone analogues
de Siqueira, Lucianna Rabelo Pessoa, de Moraes Gomes, Paulo André Teixeira, de Lima Ferreira, Larissa Pelágia, de Melo Rêgo, Moacyr Jesus Barreto, Leite, Ana Cristina Lima
Published in European journal of medicinal chemistry (15.05.2019)
Published in European journal of medicinal chemistry (15.05.2019)
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Structural improvement of new thiazolyl-isatin derivatives produces potent and selective trypanocidal and leishmanicidal compounds
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Published in Chemico-biological interactions (25.08.2021)
Published in Chemico-biological interactions (25.08.2021)
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Compound profiling and 3D-QSAR studies of hydrazone derivatives with activity against intracellular Trypanosoma cruzi
Costa, Lívia Bandeira, Cardoso, Marcos Veríssimo de Oliveira, de Oliveira Filho, Gevanio Bezerra, de Moraes Gomes, Paulo André Teixeira, Espíndola, José Wanderlan Pontes, de Jesus Silva, Thays Gabrielle, Torres, Pedro Henrique Monteiro, Silva, Floriano Paes, Martin, Julio, de Figueiredo, Regina Célia Bressan Queiroz, Leite, Ana Cristina Lima
Published in Bioorganic & medicinal chemistry (15.04.2016)
Published in Bioorganic & medicinal chemistry (15.04.2016)
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Dual Parasiticidal Activities of Phthalimides: Synthesis and Biological Profile againstTrypanosoma cruziandPlasmodium falciparum
de Moraes Gomes, Paulo Andre Teixeira, de Oliveira Cardoso, Marcos Verissimo, dos Santos, Ignes Regina, de Sousa, Fabiano Amaro, da Conceicao, Juliana Maria, de Melo Silva, Vanessa Gouveia, Duarte, Denise, Pereira, Raquel, Oliveira, Rafael, Nogueira, Fatima, Alves, Luiz Carlos, Brayner, Fabio Andre, da Silva Santos, Aline Caroline, Alves Pereira, Valeria Rego, Lima Leite, Ana Cristina
Published in ChemMedChem (18.11.2020)
Published in ChemMedChem (18.11.2020)
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Synthesis, ADMET Prediction, and Antitumor Profile of Phenoxyhydrazine- 1,3-thiazoles Derivatives
de Siqueira, Lucianna Rabelo Pessoa, de Lima Ferreira, Larissa Pelágia, de Oliveira Filho, Gevanio Bezerra, de Oliveira, Marcos Victor Gregório, Pinto, Aline Ferreira, de Melo Silva, Vanessa Gouveia, de Moraes Gomes, Paulo André Teixeira, de Oliveira Cardoso, Marcos Veríssimo, de Nazaré Correia Soeiro, Maria, Dos Santos, Flaviana Alves, da Rocha Pitta, Maíra Galdino, Nunes, Janine Siqueira, de Melo Rego, Moacyr Jesus Barreto, Leite, Ana Cristina Lima
Published in Current topics in medicinal chemistry (2023)
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Published in Current topics in medicinal chemistry (2023)
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Synthesis and In Vitro and Silico Anti-inflammatory Activity of New Thiazolidinedione-quinoline Derivatives
Barbosa da Silva, Sandra Elizabeth, da Silva Moura, José Arion, Branco Júnior, Jeann Fabiann, Teixeira de Moraes Gomes, Paulo André, Silva de Paula, Simão Kalebe, Francisco Viana, Douglas Carvalho, Vasconcelos de Freitas Ramalho, Eduardo Augusto, Gomes, João Victor de Melo, Pereira, Michelly Cristiny, Pitta, Maira Galdino da Rocha, Pitta, Ivan da Rocha, Pitta, Marina Galdino da Rocha
Published in Current topics in medicinal chemistry (21.03.2024)
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Published in Current topics in medicinal chemistry (21.03.2024)
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