Modulation of adenosine receptor affinity and intrinsic efficacy in adenine nucleosides substituted at the 2-position
Ohno, Michihiro, Gao, Zhan-Guo, Van Rompaey, Philippe, Tchilibon, Susanna, Kim, Soo-Kyung, Harris, Brian A, Gross, Ariel S, Duong, Heng T, Van Calenbergh, Serge, Jacobson, Kenneth A
Published in Bioorganic & medicinal chemistry (01.06.2004)
Published in Bioorganic & medicinal chemistry (01.06.2004)
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(N)-Methanocarba 2,N6-Disubstituted Adenine Nucleosides as Highly Potent and Selective A3 Adenosine Receptor Agonists
TCHILIBON, Susanna, JOSHI, Bhalchandra V., KIM, Soo-Kyung, DUONG, Heng T., GAO, Zhan-Guo, JACOBSON, Kenneth A.
Published in Journal of medicinal chemistry (24.03.2005)
Published in Journal of medicinal chemistry (24.03.2005)
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Journal Article
Antiaggregatory activity in human platelets of potent antagonists of the P2Y1 receptor
CATTANEO, Marco, LECCHI, Anna, OHNO, Michihiro, JOSHI, Bhalchandra V, BESADA, Pedro, TCHILIBON, Susanna, LOMBARDI, Rossana, BISCHOFBERGER, Norbert, HARDEN, T. Kendall, JACOBSON, Kenneth A
Published in Biochemical pharmacology (01.11.2004)
Published in Biochemical pharmacology (01.11.2004)
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Journal Article
Exploring distal regions of the A3 adenosine receptor binding site: sterically constrained N6-(2-phenylethyl)adenosine derivatives as potent ligands
TCHILIBON, Susanna, KIM, Soo-Kyung, GAO, Zhan-Guo, HARRIS, Brian A, BLAUSTEIN, Joshua B, GROSS, Ariel S, DUONG, Heng T, MELMAN, Neli, JACOBSON, Kenneth A
Published in Bioorganic & medicinal chemistry (01.05.2004)
Published in Bioorganic & medicinal chemistry (01.05.2004)
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Journal Article
Molecular targets for cannabidiol and its synthetic analogues: effect on vanilloid VR1 receptors and on the cellular uptake and enzymatic hydrolysis of anandamide
Bisogno, Tiziana, Hanuš, Lumír, De Petrocellis, Luciano, Tchilibon, Susanna, Ponde, Datta E, Brandi, Ines, Moriello, Aniello Schiano, Davis, John B, Mechoulam, Raphael, Di Marzo, Vincenzo
Published in British journal of pharmacology (01.10.2001)
Published in British journal of pharmacology (01.10.2001)
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Journal Article
Antiaggregatory activity in human platelets of potent antagonists of the P2Y 1 receptor
Cattaneo, Marco, Lecchi, Anna, Ohno, Michihiro, Joshi, Bhalchandra V., Besada, Pedro, Tchilibon, Susanna, Lombardi, Rossana, Bischofberger, Norbert, Harden, T. Kendall, Jacobson, Kenneth A.
Published in Biochemical pharmacology (15.11.2004)
Published in Biochemical pharmacology (15.11.2004)
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Journal Article
Enantiomeric cannabidiol derivatives: synthesis and binding to cannabinoid receptors
Hanus, LO, Tchilibon, S, Ponde, DE, Breuer, A, Fride, E, Mechoulam, R
Published in Organic & biomolecular chemistry (21.03.2005)
Published in Organic & biomolecular chemistry (21.03.2005)
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A neoceptor approach to unraveling microscopic interactions between the human A2A adenosine receptor and its agonists
Jacobson, Kenneth A, Ohno, Michihiro, Duong, Heng T, Kim, Soo-Kyung, Tchilibon, Susanna, Cesnek, Michal, Holý, Antonín, Gao, Zhan-Guo
Published in Chemistry & biology (01.02.2005)
Published in Chemistry & biology (01.02.2005)
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Journal Article
Semirational Design of (North)-Methanocarba Nucleosides as Dual Acting A1 and A3 Adenosine Receptor Agonists: Novel Prototypes for Cardioprotection
Jacobson, Kenneth A, Gao, Zhan-Guo, Tchilibon, Susanna, Duong, Heng T, Joshi, Bhalchandra V, Sonin, Dmitry, Liang, Bruce T
Published in Journal of medicinal chemistry (29.12.2005)
Published in Journal of medicinal chemistry (29.12.2005)
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Amphiphilic pyridinium salts block TNFα/NFκB signaling and constitutive hypersecretion of interleukin-8 (IL-8) from cystic fibrosis lung epithelial cells
Tchilibon, Susanna, Zhang, Jian, Yang, QingFeng, Eidelman, Ofer, Kim, Haksung, Caohuy, Hung, Jacobson, Kenneth A., Pollard, Bette S., Pollard, Harvey B.
Published in Biochemical pharmacology (01.08.2005)
Published in Biochemical pharmacology (01.08.2005)
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Journal Article
Semi-rational design of (north)-methanocarba nucleosides as dual acting A(1) and A(3) adenosine receptor agonists: novel prototypes for cardioprotection
Jacobson, Kenneth A, Gao, Zhan-Guo, Tchilibon, Susanna, Duong, Heng T, Joshi, Bhalchandra V, Sonin, Dmitry, Liang, Bruce T
Published in Journal of medicinal chemistry (29.12.2005)
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Published in Journal of medicinal chemistry (29.12.2005)
Journal Article
Semi-Rational Design of (N)-Methanocarba Nucleosides as Dual Acting A1 and A3Adenosine Receptor Agonists: Novel Prototypes for Cardioprotection
Jacobson, Kenneth A., Gao, Zhan-Guo, Tchilibon, Susanna, Duong, Heng T., Joshi, Bhalchandra V., Sonin, Dmitry, Liang, Bruce T.
Published in Journal of medicinal chemistry (29.12.2005)
Published in Journal of medicinal chemistry (29.12.2005)
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Journal Article
Semirational Design of (North)-Methanocarba Nucleosides as Dual Acting A 1 and A 3 Adenosine Receptor Agonists: Novel Prototypes for Cardioprotection
Jacobson, Kenneth A., Gao, Zhan-Guo, Tchilibon, Susanna, Duong, Heng T., Joshi, Bhalchandra V., Sonin, Dmitry, Liang, Bruce T.
Published in Journal of medicinal chemistry (01.12.2005)
Published in Journal of medicinal chemistry (01.12.2005)
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Structure activity and molecular modeling analyses of ribose- and base-modified uridine 5′-triphosphate analogues at the human P2Y 2 and P2Y 4 receptors
Jacobson, Kenneth A., Costanzi, Stefano, Ivanov, Andrei A., Tchilibon, Susanna, Besada, Pedro, Gao, Zhan-Guo, Maddileti, Savitri, Harden, T. Kendall
Published in Biochemical pharmacology (2006)
Published in Biochemical pharmacology (2006)
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Journal Article
( N )-Methanocarba 2, N 6 -Disubstituted Adenine Nucleosides as Highly Potent and Selective A 3 Adenosine Receptor Agonists
Tchilibon, Susanna, Joshi, Bhalchandra V., Kim, Soo-Kyung, Duong, Heng T., Gao, Zhan-Guo, Jacobson, Kenneth A.
Published in Journal of medicinal chemistry (01.03.2005)
Published in Journal of medicinal chemistry (01.03.2005)
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Journal Article
(N)-Methanocarba 2,N6-disubstituted adenine nucleosides as highly potent and selective as adenosine receptor agonists
TCHILIBON, Susanna, JOSHI, Bhalchandra V, KIM, Soo-Kyung, DUONG, Heng T, GAO, Zhan-Guo, JACOBSON, Kenneth A
Published in Journal of medicinal chemistry (2005)
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Published in Journal of medicinal chemistry (2005)
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