1378 Discovery and characterization of PM-4321, a selective inhibitor of the aryl hydrocarbon receptor (AHR) with anti-tumor immunomodulatory effects
Ramani, Kritika, Wrocklage, Christopher, Bai, Ming, Bosco, Anna Nicole, Carter, Benjamin, Pruteanu-Malinici, Iulian, Perales, Lizeth, Dworakowski, Wojciech, Eustace, Brenda K, Yi, Kun Don, Sinclair, Charles, Kumar, Seema, Abbinanti, Matthew, Bartolozzi, Alessandra, Proudfoot, John Robert, Briggs, Timothy, Taylor, John Steven, Salter-Cid, Luisa, Ranganath, Sheila
Published in Journal for immunotherapy of cancer (01.11.2023)
Published in Journal for immunotherapy of cancer (01.11.2023)
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Journal Article
AHR 길항제로서의 피리도피리미디논 유도체
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Year of Publication 29.08.2022
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Year of Publication 29.08.2022
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모노메틸 푸마르산염-담체 접합체 및 그 사용 방법
BERRY DAVID ARTHUR, CASEY JOHN PATRICK JR, ALEXANDER JESSICA ELIZABETH, YASUDA KOJI, GUNASEKERA DINARA SHASHANKA, BRIGGS TIMOTHY, LIANG ANNA, PECK SPENCER CORY, NUDEL KATHLEEN, KAMALI SARVESTANI AFRAND, TAYLOR STEVEN JOHN, ROSS CHERI, BUCKBINDER LEONARD, LANTER BERNARD, KIM MI JEONG
Year of Publication 13.08.2021
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Year of Publication 13.08.2021
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대사 장애 및 비알코올성 지방 간 질환의 치료를 위한 활성제 및 그 사용 방법
BERRY DAVID ARTHUR, ALEXANDER JESSICA, CASEY JOHN PATRICK JR, BRIGGS TIMOTHY F, YASUDA KOJI, SNEDEKER CHERI, GUNASEKERA DINARA, LIANG ANNA, PECK SPENCER CORY, PROUDFOOT JOHN ROBERT, NUDEL KATHLEEN, KAMALI SARVESTANI AFRAND, TAYLOR STEVEN JOHN, BUCKBINDER LEONARD, MASSARI FERDINAND EDWARD, LANTER BERNARD, KIM MI JEONG, LE DIANA
Year of Publication 15.02.2021
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Year of Publication 15.02.2021
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ASPARAGINE DERIVATIVES AND METHODS OF USING SAME
MCELROY, William, LIU, Jenny, BRIGGS, Timothy F, PROUDFOOT, John Robert, MYERS, Robert Walter, TAYLOR, Steven John, PECK, Spencer Cory
Year of Publication 27.07.2023
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Year of Publication 27.07.2023
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Fused Imidazole Derivatives as AHR Antagonists
Blois, Anna, Ly, Vu Linh, Proudfoot, John Robert, Buckbinder, Leonard, Bartolozzi, Alessandra, Mancuso, John, Lanter, Bernard, Taylor, Steven John, Bos, Maxence, Briggs, Timothy
Year of Publication 19.10.2023
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Year of Publication 19.10.2023
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Fused Azole Heterocycles as AHR Antagonists
Blois, Anna, Ly, Vu Linh, Proudfoot, John Robert, Buckbinder, Leonard, Bartolozzi, Alessandra, Guo, Tianlin, Mancuso, John, Lanter, Bernard, Taylor, Steven John, Bos, Maxence, Briggs, Timothy
Year of Publication 27.07.2023
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Year of Publication 27.07.2023
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Conjugates and methods of using the same
Im, Joo Hyun, Proudfoot, John Robert, Ross, Cheri, Bogart, Elijah Lane, Isaac, Dervla Tamara, Peck, Spencer Cory, Massari, Ferdinand Edward, Myers, Robert Walter, Casey, Jr., John Patrick, Taylor, Steven John, Liu, Jenny, Doud, Devin Forest Reed, Berry, David Arthur
Year of Publication 04.06.2024
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Year of Publication 04.06.2024
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ASPARAGINE DERIVATIVES AND METHODS OF USING SAME
MCELROY, William, LIU, Jenny, BRIGGS, Timothy F, PROUDFOOT, John Robert, MYERS, Robert Walter, TAYLOR, Steven John, PECK, Spencer Cory
Year of Publication 16.12.2021
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Year of Publication 16.12.2021
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PYRIDOPYRIMIDINONE DERIVATIVES AS AHR ANTAGONISTS
GUO, Tianlin, BUREAU, Patrick, BOS, Maxence, BLOIS, Anna, BRIGGS, Timothy, BONEPALLY, Karunakar Reddy, BARONE, Francesca, BARTOLOZZI, Alessandra, BUCKBINDER, Leonard, PROUDFOOT, John Robert, MANCUSO, John, LANTER, Bernard, TAYLOR, Steven John
Year of Publication 21.09.2023
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Year of Publication 21.09.2023
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ACTIVE AGENTS AND METHODS OF THEIR USE FOR THE TREATMENT OF METABOLIC DISORDERS AND NONALCOHOLIC FATTY LIVER DISEASE
MASSARI, Ferdinand Edward, GUNASEKERA, Dinara, NUDEL, Kathleen, YASUDA, Koji, PECK, Spencer Cory, LE, Diana, ALEXANDER, Jessica, SNEDEKER, Cheri, LIANG, Anna, KIM, Mi-Jeong, KAMALI SARVESTANI, Afrand, BUCKBINDER, Leonard, BRIGGS, Timothy F, PROUDFOOT, John Robert, LANTER, Bernard, TAYLOR, Steven John, BERRY, David Arthur, CASEY, JR., John Patrick
Year of Publication 06.06.2024
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Year of Publication 06.06.2024
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MONOMETHYL FUMARATE-CARRIER CONJUGATES AND METHODS OF THEIR USE
BERRY, David, Arthur, PECK, Spencer, Cory, TAYLOR, Steven, John, GUNASEKERA, Dinara, Shashanka, BRIGGS, Timothy, NUDEL, Kathleen, YASUDA, Koji, LIANG, Anna, KIM, Mi-Jeong, BUCKBINDER, Leonard, KAMALI SARVESTANI, Afrand, CASEY, John, Patrick, Jr, ALEXANDER, Jessica, Elizabeth, LANTER, Bernard, ROSS, Cheri
Year of Publication 28.12.2022
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Year of Publication 28.12.2022
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Active agents and methods of their use for the treatment of metabolic disorders and nonalcoholic fatty liver disease
Proudfoot, John Robert, Briggs, Timothy F, Snedeker, Cheri, Kamali Sarvestani, Afrand, Peck, Spencer Cory, Liang, Anna, Massari, Ferdinand Edward, Alexander, Jessica, Gunasekera, Dinara, Nudel, Kathleen, Buckbinder, Leonard, Lanter, Bernard, Casey, Jr., John Patrick, Taylor, Steven John, Le, Diana, Kim, Mi-Jeong, Yasuda, Koji, Berry, David Arthur
Year of Publication 14.11.2023
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Year of Publication 14.11.2023
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FUSED AZOLE HETEROCYCLES AS AHR ANTAGONISTS
BARTOLOZZI, Alessandra, GUO, Tianlin, LY, Vu Linh, BUCKBINDER, Leonard, PROUDFOOT, John Robert, MANCUSO, John, BOS, Maxence, BLOIS, Anna, LANTER, Bernard, TAYLOR, Steven John, BRIGGS, Timothy
Year of Publication 02.12.2021
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Year of Publication 02.12.2021
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FUSED IMIDAZOLE DERIVATIVES AS AHR ANTAGONISTS
BARTOLOZZI, Alessandra, LY, Vu Linh, BUCKBINDER, Leonard, PROUDFOOT, John Robert, MANCUSO, John, BOS, Maxence, BLOIS, Anna, LANTER, Bernard, TAYLOR, Steven John, BRIGGS, Timothy
Year of Publication 25.11.2021
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Year of Publication 25.11.2021
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PYRIDOPYRIMIDINONE DERIVATIVES AS AHR ANTAGONISTS
GUO, Tianlin, BUREAU, Patrick, BOS, Maxence, BLOIS, Anna, BRIGGS, Timothy, BONEPALLY, Karunakar Reddy, BARONE, Francesca, BARTOLOZZI, Alessandra, BUCKBINDER, Leonard, PROUDFOOT, John Robert, MANCUSO, John, LANTER, Bernard, TAYLOR, Steven John
Year of Publication 28.09.2022
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Year of Publication 28.09.2022
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ACYLATED CATECHIN POLYPHENOLS AND METHODS OF THEIR USE FOR THE TREATMENT OF CANCER
BERRY, David, Arthur, CASEY, John Patrick, Jr, KIM, Mi-Jeong, TAYLOR, Steven, John, BUCKBINDER, Leonard, PECK, Spencer, Cory, PROUDFOOT, John, Robert, BRIGGS, Timothy, F, MOAREFI, Amir, MASSARI, Ferdinand, Edward, YASUDA, Koji
Year of Publication 10.08.2022
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Year of Publication 10.08.2022
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