Search Results - "TAVERNE THIERRY" :: K.UTB vyhledávací portál | TBU Library Retrieval Portal

A novel DYRK1A (Dual specificity tyrosine phosphorylation‐regulated kinase 1A) inhibitor for the treatment of Alzheimer's disease: effect on Tau and amyloid pathologies in vitro

A novel DYRK1A (Dual specificity tyrosine phosphorylation‐regulated kinase 1A) inhibitor for the treatment of Alzheimer's disease: effect on Tau and amyloid pathologies in vitro

by Coutadeur, Séverine, Benyamine, Hélène, Delalonde, Laurence, Oliveira, Catherine, Leblond, Bertrand, Foucourt, Alicia, Besson, Thierry, Casagrande, Anne‐Sophie, Taverne, Thierry, Girard, Angélique, Pando, Matthew P., Désiré, Laurent
Published in Journal of neurochemistry (01.05.2015)

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Design and synthesis of thiazolo[5,4-f]quinazolines as DYRK1A inhibitors, part II

Design and synthesis of thiazolo[5,4-f]quinazolines as DYRK1A inhibitors, part II

by Foucourt, Alicia, Hédou, Damien, Dubouilh-Benard, Carole, Girard, Angélique, Taverne, Thierry, Casagrande, Anne-Sophie, Désiré, Laurent, Leblond, Bertrand, Besson, Thierry
Published in Molecules (Basel, Switzerland) (26.09.2014)

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New COX-2/5-LOX Inhibitors: Apoptosis-Inducing Agents Potentially Useful in Prostate Cancer Chemotherapy

New COX-2/5-LOX Inhibitors: Apoptosis-Inducing Agents Potentially Useful in Prostate Cancer Chemotherapy

by Pommery, Nicole, Taverne, Thierry, Telliez, Aurélie, Goossens, Laurence, Charlier, Caroline, Pommery, Jean, Goossens, Jean-François, Houssin, Raymond, Durant, François, Hénichart, Jean-Pierre
Published in Journal of medicinal chemistry (02.12.2004)

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Synthesis and Activity of a New Methoxytetrahydropyran Derivative as Dual Cyclooxygenase-2/5-Lipoxygenase Inhibitor

Synthesis and Activity of a New Methoxytetrahydropyran Derivative as Dual Cyclooxygenase-2/5-Lipoxygenase Inhibitor

by Barbey, Sabine, Goossens, Laurence, Taverne, Thierry, Cornet, Joséphine, Choesmel, Valérie, Rouaud, Céline, Gimeno, Gilles, Yannic-Arnoult, Sylvie, Michaux, Catherine, Charlier, Caroline, Houssin, Raymond, Hénichart, Jean-Pierre
Published in Bioorganic & medicinal chemistry letters (11.03.2002)

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RAC1 Inhibition Targets Amyloid Precursor Protein Processing by γ-Secretase and Decreases Aβ Production in Vitro and in Vivo

RAC1 Inhibition Targets Amyloid Precursor Protein Processing by γ-Secretase and Decreases Aβ Production in Vitro and in Vivo

by Désiré, Laurent, Bourdin, Jérôme, Loiseau, Nadia, Peillon, Hélène, Picard, Virginie, De Oliveira, Catherine, Bachelot, Florence, Leblond, Bertrand, Taverne, Thierry, Beausoleil, Eric, Lacombe, Sandrine, Drouin, Dominique, Schweighoffer, Fabien
Published in The Journal of biological chemistry (11.11.2005)

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Abstract 2794: Cytotoxic and vascular disrupting activity of EHT 6706, a novel tubulin polymerization inhibitor

Abstract 2794: Cytotoxic and vascular disrupting activity of EHT 6706, a novel tubulin polymerization inhibitor

by Casagrande, Anne-Sophie, Bachelot, Florence, Oliveira, Catherine De, Coutadeur, Séverine, Carton, Rachel, Chauvignac, Cédric, Pognante, Laure, Petibon, Angélique, Taverne, Thierry, Beausoleil, Eric, Leblond, Bertrand, Pando, Matt, Desire, Laurent
Published in Cancer research (Chicago, Ill.) (15.04.2012)

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Abstract C89: Rac1 splicing variant Rac1b: Towards isoform selective inhibitors for the treatment of cancer

Abstract C89: Rac1 splicing variant Rac1b: Towards isoform selective inhibitors for the treatment of cancer

by Laurent, Desire, Casagrande, Anne-Sophie, Leblond, Bertrand, Beausoleil, Eric, Taverne, Thierry, Chauvignac, Cedric, Pando, Matt
Published in Molecular cancer therapeutics (10.12.2009)

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Structure–activity relationship of isoform selective inhibitors of Rac1/1b GTPase nucleotide binding

Structure–activity relationship of isoform selective inhibitors of Rac1/1b GTPase nucleotide binding

by Beausoleil, Eric, Chauvignac, Cédric, Taverne, Thierry, Lacombe, Sandrine, Pognante, Laure, Leblond, Bertrand, Pallares, Diego, Oliveira, Catherine De, Bachelot, Florence, Carton, Rachel, Peillon, Hélène, Coutadeur, Séverine, Picard, Virginie, Lambeng, Nathalie, Désiré, Laurent, Schweighoffer, Fabien
Published in Bioorganic & medicinal chemistry letters (01.10.2009)

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Vascular disrupting activity and the mechanism of action of EHT 6706, a novel anticancer tubulin polymerization inhibitor

Vascular disrupting activity and the mechanism of action of EHT 6706, a novel anticancer tubulin polymerization inhibitor

by Belzacq-Casagrande, Anne-Sophie, Bachelot, Florence, De Oliveira, Catherine, Coutadeur, Séverine, Maurier-Mahé, Florence, Throo, Emeline, Chauvignac, Cédric, Pognante, Laure, Petibon, Angélique, Taverne, Thierry, Beausoleil, Eric, Leblond, Bertrand, Pando, Matthew P., Désiré, Laurent
Published in Investigational new drugs (01.04.2013)

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SUBSTITUTED 6,7-DIALKOXY-3-ISOQUINOLINOL DERIVATIVES AS INHIBITORS OF PHOSPHODIESTERASE 10 (PDE10A)

SUBSTITUTED 6,7-DIALKOXY-3-ISOQUINOLINOL DERIVATIVES AS INHIBITORS OF PHOSPHODIESTERASE 10 (PDE10A)

by DESIRE LAURENT J.R, LEBLOND BERTRAND, CASAGRANDE ANNE SOPHIE, TAVERNE THIERRY, DONELLO JOHN E, BEAUSOLEIL ERIC, CHAUVIGNAC CEDRIC, PANDO MATTHEW P, YANG RONG
Year of Publication 22.01.2014

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Patent

3-(4-FLUOROPHENYL)-3-HYDROXY-2-AMINO-PROPIONIC ACID AMIDES AND RELATED COMPOUNDS HAVING ANALGESIC ACTIVITY

3-(4-FLUOROPHENYL)-3-HYDROXY-2-AMINO-PROPIONIC ACID AMIDES AND RELATED COMPOUNDS HAVING ANALGESIC ACTIVITY

by LEBLOND BERTRAND, TAVERNE THIERRY, BEAUSOLEIL ERIC, DONELLO JOHN E, CHAUVIGNAC CEDRIC, YANG RONG
Year of Publication 01.12.2010

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Patent

RAC1 inhibition targets amyloid precursor protein processing by gamma-secretase and decreases Abeta production in vitro and in vivo

RAC1 inhibition targets amyloid precursor protein processing by gamma-secretase and decreases Abeta production in vitro and in vivo

by Désiré, Laurent, Bourdin, Jérôme, Loiseau, Nadia, Peillon, Hélène, Picard, Virginie, De Oliveira, Catherine, Bachelot, Florence, Leblond, Bertrand, Taverne, Thierry, Beausoleil, Eric, Lacombe, Sandrine, Drouin, Dominique, Schweighoffer, Fabien
Published in The Journal of biological chemistry (11.11.2005)

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Journal Article

P2-339: Development of a screening platform for the identification of new Rac1/Rac1b inhibitors active in the prevention of amyloid-beta production

P2-339: Development of a screening platform for the identification of new Rac1/Rac1b inhibitors active in the prevention of amyloid-beta production

by Lambeng, Nathalie, Coutadeur, Séverine, Peillon, Hélène, Loiseau, Nadia, Bachelot, Florence, De Oliveira, Catherine, Carton, Rachel, Leblond, Bertr, Beausoleil, Eric, Chauvignac, Cédric, Taverne, Thierry, Schweighoffer, Fabien, Desire, Laurent
Published in Alzheimer's & dementia (01.07.2008)

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RAC1 Inhibition Targets Amyloid Precursor Protein Processing by Î³-Secretase and Decreases AÎ² Production in Vitro and in Vivo

RAC1 Inhibition Targets Amyloid Precursor Protein Processing by Î³-Secretase and Decreases AÎ² Production in Vitro and in Vivo

by Laurent DÃ©sirÃ, JÃ©rÃ´me Bourdin, Nadia Loiseau, HÃ©lÃ¨ne Peillon, Virginie Picard, Catherine De Oliveira, Florence Bachelot, Bertrand Leblond, Thierry Taverne, Eric Beausoleil, Sandrine Lacombe, Dominique Drouin, Fabien Schweighoffer
Published in The Journal of biological chemistry (11.11.2005)

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Journal Article

New COOX-2/5-LOX inhibitors: Apoptosis-inducing agents potentially useful in prostate cancer chemotherapy

New COOX-2/5-LOX inhibitors: Apoptosis-inducing agents potentially useful in prostate cancer chemotherapy

by POMMERY, Nicole, TAVERNE, Thierry, TELLIEZ, Aurélie, GOOSSENS, Laurence, CHARLIER, Caroline, POMMERY, Jean, GOOSSENS, Jean-Francois, HOUSSIN, Raymond, DURANT, Francois, HENICHART, Jean-Pierre
Published in Journal of medicinal chemistry (2004)

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3-aryl-3-hydroxy-2-amino-propionic acid amides, 3-heteroaryl-3-hydroxy-2-amino-propionic acid amides and related compounds having analgesic and/or immunostimulant activity

3-aryl-3-hydroxy-2-amino-propionic acid amides, 3-heteroaryl-3-hydroxy-2-amino-propionic acid amides and related compounds having analgesic and/or immunostimulant activity

by Donello, John E, Beausoleil, Eric, Taverne, Thierry, Leblond, Bertrand
Year of Publication 18.07.2019

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Patent

3-aryl-3-hydroxy-2-amino-propionic acid amides, 3-heteroaryl-3-hydroxy-2-amino-propionic acid amides and related compounds having analgesic and/or immunostimulant activity

3-aryl-3-hydroxy-2-amino-propionic acid amides, 3-heteroaryl-3-hydroxy-2-amino-propionic acid amides and related compounds having analgesic and/or immunostimulant activity

by Donello, John E, Beausoleil, Eric, Taverne, Thierry, Leblond, Bertrand
Year of Publication 17.05.2018

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Patent

3-aryl-3-hydroxy-2-amino-propionic acid amides, 3-heteroaryl-3-hydroxy-2-amino-propionic acid amides and related compounds having analgesic and/or immunostimulant activity

3-aryl-3-hydroxy-2-amino-propionic acid amides, 3-heteroaryl-3-hydroxy-2-amino-propionic acid amides and related compounds having analgesic and/or immunostimulant activity

by Donello, John E, Beausoleil, Eric, Taverne, Thierry, Leblond, Bertrand
Year of Publication 01.02.2018

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Patent

1-aryl-1-hydroxy-2,3-diamino-propyl amines, 1-heteroaryl-1-hydroxy-2,3-diamino-propyl amines and related compounds having analgesic and/or immuno stimulant activity

1-aryl-1-hydroxy-2,3-diamino-propyl amines, 1-heteroaryl-1-hydroxy-2,3-diamino-propyl amines and related compounds having analgesic and/or immuno stimulant activity

by Donello John E, Taverne Thierry, Leblond Bertrand, Beusoleil Eric
Year of Publication 28.11.2017

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Patent

Amidas de ácido 3-aril-3-hidróxi-2-amino-propiônico, 3-heteroaril-3-hidróxi-2-amino-propiônico e compostos relacionados tendo atividade analgésica e/ou imunoestimulante

Amidas de ácido 3-aril-3-hidróxi-2-amino-propiônico, 3-heteroaril-3-hidróxi-2-amino-propiônico e compostos relacionados tendo atividade analgésica e/ou imunoestimulante

by LEBLOND BERTRAND, TAVERNE THIERRY, BEAUSOLEIL ERIC, JOHN E. DONELLO
Year of Publication 08.02.2022

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Patent

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