Novel Uncomplexed and Complexed Structures of Plasmepsin II, an Aspartic Protease from Plasmodium falciparum
Asojo, Oluwatoyin A., Gulnik, Sergei V., Afonina, Elena, Yu, Betty, Ellman, Jonathan A., Haque, Tasir S., Silva, Abelardo M.
Published in Journal of molecular biology (14.03.2003)
Published in Journal of molecular biology (14.03.2003)
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Journal Article
Identification of potent 11mer Glucagon-Like Peptide-1 Receptor agonist peptides with novel C-terminal amino acids: Homohomophenylalanine analogs
Haque, Tasir S., Lee, Ving G., Riexinger, Douglas, Lei, Ming, Malmstrom, Sarah, Xin, Li, Han, Songping, Mapelli, Claudio, Cooper, Christopher B., Zhang, Ge, Ewing, William R., Krupinski, John
Published in Peptides (New York, N.Y. : 1980) (01.05.2010)
Published in Peptides (New York, N.Y. : 1980) (01.05.2010)
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Liquid-liquid extraction coupled with LC/MS/MS for monitoring of malonyl-CoA in rat brain tissue
Onorato, Joelle M, Chen, Luping, Shipkova, Petia, Ma, Zhengping, Azzara, Anthony V, Devenny, James J, Liang, Ningning, Haque, Tasir S, Cheng, Dong
Published in Analytical and bioanalytical chemistry (01.08.2010)
Published in Analytical and bioanalytical chemistry (01.08.2010)
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Journal Article
Potent, Low-Molecular-Weight Non-Peptide Inhibitors of Malarial Aspartyl Protease Plasmepsin II
Haque, Tasir S, Skillman, A. Geoffrey, Lee, Christina E, Habashita, Hiromu, Gluzman, Ilya Y, Ewing, Todd J. A, Goldberg, Daniel E, Kuntz, Irwin D, Ellman, Jonathan A
Published in Journal of medicinal chemistry (22.04.1999)
Published in Journal of medicinal chemistry (22.04.1999)
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Journal Article
Parallel Synthesis of Potent, Pyrazole-Based Inhibitors of Helicobacter pylori Dihydroorotate Dehydrogenase
HAQUE, Tasir S., TADESSE, Seifu, MARCINKEVICIENE, Jovita, ROGERS, M. John, SIZEMORE, Christine, KOPCHO, Lisa M., AMSLER, Karen, ECRET, Lisa D., ZHAN, Dong Liang, HOBBS, Frank, SLEE, Andrew, TRAINOR, George L., STERN, Andrew M., COPELAND, Robert A., COMBS, Andrew P.
Published in Journal of medicinal chemistry (10.10.2002)
Published in Journal of medicinal chemistry (10.10.2002)
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Journal Article
Exploration of structure–activity relationships at the two C-terminal residues of potent 11mer Glucagon-Like Peptide-1 receptor agonist peptides via parallel synthesis
Haque, Tasir S., Martinez, Rogelio L., Lee, Ving G., Riexinger, Douglas G., Lei, Ming, Feng, Ming, Koplowitz, Barry, Mapelli, Claudio, Cooper, Christopher B., Zhang, Ge, Huang, Christine, Ewing, William R., Krupinski, John
Published in Peptides (New York, N.Y. : 1980) (01.07.2010)
Published in Peptides (New York, N.Y. : 1980) (01.07.2010)
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Journal Article
Potent biphenyl- and 3-phenyl pyridine-based inhibitors of acetyl-CoA carboxylase
Haque, Tasir S., Liang, Ningning, Golla, Rajasree, Seethala, Ramakrishna, Ma, Zhengping, Ewing, William R., Cooper, Christopher B., Pelleymounter, Mary Ann, Poss, Michael A., Cheng, Dong
Published in Bioorganic & medicinal chemistry letters (15.10.2009)
Published in Bioorganic & medicinal chemistry letters (15.10.2009)
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Journal Article
Searching for Minimum Increments of Hydrophobic Collapse: Flexible Dinaphthyl Carboxylates
Newcomb, Lisa F, Haque, Tasir S, Gellman, Samuel H
Published in Journal of the American Chemical Society (01.06.1995)
Published in Journal of the American Chemical Society (01.06.1995)
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Journal Article
Selective inhibition of bacterial dihydroorotate dehydrogenases by thiadiazolidinediones
Marcinkeviciene, Jovita, Rogers, M.John, Kopcho, Lisa, Jiang, Wenjun, Wang, Kathy, Murphy, Dennis J, Lippy, Jonathan, Link, Steven, Chung, Thomas D.Y, Hobbs, Frank, Haque, Tasir, Trainor, George L, Slee, Andrew, Stern, Andrew M, Copeland, Robert A
Published in Biochemical pharmacology (01.08.2000)
Published in Biochemical pharmacology (01.08.2000)
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Journal Article
I09 A Huntington’s disease embryonic stem cell phenotypic hts to identify small molecule modulators of mutant huntingtin
Todd, Daniel, Stebbeds, Marta, Thatcher, Emma, Barnard, Amy, Anton, Jeremy, Sienerth, Arnold, Visser, Mijke, Mitchell, Philip, Breccia, Perla, Smith, David, McAllister, George, Haque, Tasir, Liu, Longbin, Dominguez, Celia, Munoz-Sanjuan, Ignacio
Published in Journal of neurology, neurosurgery and psychiatry (12.09.2022)
Published in Journal of neurology, neurosurgery and psychiatry (12.09.2022)
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Journal Article
Novel Cathepsin D Inhibitors Block the Formation of Hyperphosphorylated Tau Fragments in Hippocampus
Bi, Xiaoning, Haque, Tasir S., Zhou, Jun, Skillman, A. Geoffrey, Lin, Bin, Lee, Christine E., Kuntz, Irwin D., Ellman, Jonathan A., Lynch, Gary
Published in Journal of neurochemistry (01.04.2000)
Published in Journal of neurochemistry (01.04.2000)
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Journal Article
Structural Characterization of Thiocyclophanes That Promote Edge-to-Face Aromatic-Aromatic Geometries
Schladetzky, Kurt D, Haque, Tasir S, Gellman, Samuel H
Published in Journal of organic chemistry (01.06.1995)
Published in Journal of organic chemistry (01.06.1995)
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Journal Article
Parallel Synthesis of Potent, Pyrazole-Based Inhibitors of Helicobacter p ylori Dihydroorotate Dehydrogenase
Haque, Tasir S, Tadesse, Seifu, Marcinkeviciene, Jovita, Rogers, M. John, Sizemore, Christine, Kopcho, Lisa M, Amsler, Karen, Ecret, Lisa D, Zhan, Dong Liang, Hobbs, Frank, Slee, Andrew, Trainor, George L, Stern, Andrew M, Copeland, Robert A, Combs, Andrew P
Published in Journal of medicinal chemistry (10.10.2002)
Published in Journal of medicinal chemistry (10.10.2002)
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Journal Article
Helicobacter pylori-selective Antibacterials Based on Inhibition of Pyrimidine Biosynthesis
Copeland, Robert A., Marcinkeviciene, Jovita, Haque, Tasir S., Kopcho, Lisa M., Jiang, Wenjun, Wang, Kathy, Ecret, Lisa D., Sizemore, Christine, Amsler, Karen A., Foster, Lori, Tadesse, Seifu, Combs, Andrew P., Stern, Andrew M., Trainor, George L., Slee, Andrew, Rogers, M. John, Hobbs, Frank
Published in The Journal of biological chemistry (27.10.2000)
Published in The Journal of biological chemistry (27.10.2000)
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Journal Article
N-Arylation of Primary and Secondary Aliphatic Amines on Solid Supports
Combs, Andrew P, Tadesse, Seifu, Rafalski, Maria, Haque, Tasir S, Lam, Patrick Y. S
Published in Journal of combinatorial chemistry (01.03.2002)
Published in Journal of combinatorial chemistry (01.03.2002)
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Journal Article
Differential activation of recombinant human acetyl-CoA carboxylases 1 and 2 by citrate
Locke, Gregory A., Cheng, Dong, Witmer, Mark R., Tamura, James K., Haque, Tasir, Carney, Robert F., Rendina, Alan R., Marcinkeviciene, Jovita
Published in Archives of biochemistry and biophysics (01.07.2008)
Published in Archives of biochemistry and biophysics (01.07.2008)
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Journal Article
"Mirror image" reverse turns promote .beta.-hairpin formation
Haque, Tasir S, Little, Jennifer C, Gellman, Samuel H
Published in Journal of the American Chemical Society (01.05.1994)
Published in Journal of the American Chemical Society (01.05.1994)
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