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Published in Archives of biochemistry and biophysics (15.01.2008)
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Published in Bioorganic & medicinal chemistry letters (01.11.2007)
Published in Bioorganic & medicinal chemistry letters (01.11.2007)
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Kinesin spindle protein (KSP) inhibitors. Part 7: Design and synthesis of 3,3-disubstituted dihydropyrazolobenzoxazines as potent inhibitors of the mitotic kinesin KSP
Garbaccio, Robert M., Tasber, Edward S., Neilson, Lou Anne, Coleman, Paul J., Fraley, Mark E., Olson, Christy, Bergman, Jeff, Torrent, Maricel, Buser, Carolyn A., Rickert, Keith, Walsh, Eileen S., Hamilton, Kelly, Lobell, Robert B., Tao, Weikang, South, Vicki J., Diehl, Ronald E., Davide, Joseph P., Yan, Youwei, Kuo, Lawrence C., Li, Chunze, Prueksaritanont, Thomayant, Fernandez-Metzler, Carmen, Mahan, Elizabeth A., Slaughter, Donald E., Salata, Joseph J., Kohl, Nancy E., Huber, Hans E., Hartman, George D.
Published in Bioorganic & medicinal chemistry letters (15.10.2007)
Published in Bioorganic & medicinal chemistry letters (15.10.2007)
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Kinesin spindle protein (KSP) inhibitors. Part 2: The design, synthesis, and characterization of 2,4-diaryl-2,5-dihydropyrrole inhibitors of the mitotic kinesin KSP
Fraley, Mark E., Garbaccio, Robert M., Arrington, Kenneth L., Hoffman, William F., Tasber, Edward S., Coleman, Paul J., Buser, Carolyn A., Walsh, Eileen S., Hamilton, Kelly, Fernandes, Christine, Schaber, Michael D., Lobell, Robert B., Tao, Weikang, South, Victoria J., Yan, Youwei, Kuo, Lawrence C., Prueksaritanont, Thomayant, Shu, Cathy, Torrent, Maricel, Heimbrook, David C., Kohl, Nancy E., Huber, Hans E., Hartman, George D.
Published in Bioorganic & medicinal chemistry letters (01.04.2006)
Published in Bioorganic & medicinal chemistry letters (01.04.2006)
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Stereospecific reduction of a potent kinesin spindle protein (KSP) inhibitor in human tissues
Li, Chunze, Lu, Bing, Garbaccio, Robert M., Tasber, Edward S., Fraley, Mark E., Hartman, George D., Ye, Jingjing, Harrelson, Jane C., Prueksaritanont, Thomayant
Published in Biochemical pharmacology (15.05.2010)
Published in Biochemical pharmacology (15.05.2010)
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Synthesis and evaluation of substituted benzoisoquinolinones as potent inhibitors of Chk1 kinase
Garbaccio, Robert M., Huang, Shaei, Tasber, Edward S., Fraley, Mark E., Yan, Youwei, Munshi, Sanjeev, Ikuta, Mari, Kuo, Lawrence, Kreatsoulas, Constanine, Stirdivant, Steve, Drakas, Bob, Rickert, Keith, Walsh, Eileen S., Hamilton, Kelly A., Buser, Carolyn A., Hardwick, James, Mao, Xianzhi, Beck, Stephen C., Abrams, Marc T., Tao, Weikang, Lobell, Rob, Sepp-Lorenzino, Laura, Hartman, George D.
Published in Bioorganic & medicinal chemistry (15.11.2007)
Published in Bioorganic & medicinal chemistry (15.11.2007)
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Kinesin spindle protein (KSP) inhibitors. Part 3: Synthesis and evaluation of phenolic 2,4-diaryl-2,5-dihydropyrroles with reduced hERG binding and employment of a phosphate prodrug strategy for aqueous solubility
Garbaccio, Robert M., Fraley, Mark E., Tasber, Edward S., Olson, Christy M., Hoffman, William F., Arrington, Kenneth L., Torrent, Maricel, Buser, Carolyn A., Walsh, Eileen S., Hamilton, Kelly, Schaber, Michael D., Fernandes, Christine, Lobell, Robert B., Tao, Weikang, South, Vicki J., Yan, Youwei, Kuo, Lawrence C., Prueksaritanont, Thomayant, Slaughter, Donald E., Shu, Cathy, Heimbrook, David C., Kohl, Nancy E., Huber, Hans E., Hartman, George D.
Published in Bioorganic & medicinal chemistry letters (01.04.2006)
Published in Bioorganic & medicinal chemistry letters (01.04.2006)
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Design and synthesis of 3,7-diarylimidazopyridines as inhibitors of the VEGF-receptor KDR
ZHICAI WU, FRALEY, Mark E, BIN SHI, SEPP-LORENZINO, Laura, THOMAS, Kenneth A, BILODEAU, Mark T, KAUFMAN, Mildred L, TASBER, Edward S, BALITZA, Adrienne E, HARTMAN, George D, COLL, Kathleen E, RICKERT, Keith, SHIPMAN, Jennifer
Published in Bioorganic & medicinal chemistry letters (23.02.2004)
Published in Bioorganic & medicinal chemistry letters (23.02.2004)
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ALKOXY PYRAZOLES AS SOLUBLE GUANYLATE CYCLASE ACTIVATORS
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Year of Publication 07.05.2015
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Year of Publication 07.05.2015
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Optimization of a pyrazoloquinolinone class of Chkl kinase inhibitors
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Published in Bioorganic & medicinal chemistry letters (2007)
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Published in Bioorganic & medicinal chemistry letters (2007)
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ALKOXY PYRAZOLES AS SOLUBLE GUANYLATE CYCLASE ACTIVATORS
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ALKOXY PYRAZOLES AS SOLUBLE GUANYLATE CYCLASE ACTIVATORS
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Year of Publication 28.04.2020
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Year of Publication 27.12.2019
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Year of Publication 29.11.2019
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Year of Publication 29.11.2019
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Year of Publication 05.11.2019
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Year of Publication 14.10.2019
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