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Published in The Journal of biological chemistry (27.05.2011)
Published in The Journal of biological chemistry (27.05.2011)
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Published in The Journal of chemical physics (21.08.2018)
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Two-dimensional replica-exchange method for predicting protein-ligand binding structures
Kokubo, Hironori, Tanaka, Toshimasa, Okamoto, Yuko
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Published in Journal of computational chemistry (15.11.2013)
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Design and Synthesis of Novel Human Epidermal Growth Factor Receptor 2 (HER2)/Epidermal Growth Factor Receptor (EGFR) Dual Inhibitors Bearing a Pyrrolo[3,2-d]pyrimidine Scaffold
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Published in Journal of medicinal chemistry (08.12.2011)
Published in Journal of medicinal chemistry (08.12.2011)
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Discovery of TAK-875: A Potent, Selective, and Orally Bioavailable GPR40 Agonist
Negoro, Nobuyuki, Sasaki, Shinobu, Mikami, Satoshi, Ito, Masahiro, Suzuki, Masami, Tsujihata, Yoshiyuki, Ito, Ryo, Harada, Ayako, Takeuchi, Koji, Suzuki, Nobuhiro, Miyazaki, Junichi, Santou, Takashi, Odani, Tomoyuki, Kanzaki, Naoyuki, Funami, Miyuki, Tanaka, Toshimasa, Kogame, Akifumi, Matsunaga, Shinichiro, Yasuma, Tsuneo, Momose, Yu
Published in ACS medicinal chemistry letters (09.09.2010)
Published in ACS medicinal chemistry letters (09.09.2010)
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Published in Journal of medicinal chemistry (22.12.2011)
Published in Journal of medicinal chemistry (22.12.2011)
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Design, Synthesis, and Biological Activity of Potent and Orally Available G Protein-Coupled Receptor 40 Agonists
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Published in Journal of medicinal chemistry (10.03.2011)
Published in Journal of medicinal chemistry (10.03.2011)
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Conformational switch of angiotensin II type 1 receptor underlying mechanical stress-induced activation
Yasuda, Noritaka, Miura, Shin-ichiro, Akazawa, Hiroshi, Tanaka, Toshimasa, Qin, Yingjie, Kiya, Yoshihiro, Imaizumi, Satoshi, Fujino, Masahiro, Ito, Kaoru, Zou, Yunzeng, Fukuhara, Shigetomo, Kunimoto, Satoshi, Fukuzaki, Koichi, Sato, Toshiaki, Ge, Junbo, Mochizuki, Naoki, Nakaya, Haruaki, Saku, Keijiro, Komuro, Issei
Published in EMBO reports (01.02.2008)
Published in EMBO reports (01.02.2008)
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Novel approach of fragment-based lead discovery applied to renin inhibitors
Tawada, Michiko, Suzuki, Shinkichi, Imaeda, Yasuhiro, Oki, Hideyuki, Snell, Gyorgy, Behnke, Craig A., Kondo, Mitsuyo, Tarui, Naoki, Tanaka, Toshimasa, Kuroita, Takanobu, Tomimoto, Masaki
Published in Bioorganic & medicinal chemistry (15.11.2016)
Published in Bioorganic & medicinal chemistry (15.11.2016)
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Discovery, synthesis and biological evaluation of isoquinolones as novel and highly selective JNK inhibitors ( 2)
Asano, Yasutomi, Kitamura, Shuji, Ohra, Taiichi, Itoh, Fumio, Kajino, Masahiro, Tamura, Tomoko, Kaneko, Manami, Ikeda, Shota, Igata, Hideki, Kawamoto, Tomohiro, Sogabe, Satoshi, Matsumoto, Shin-ichi, Tanaka, Toshimasa, Yamaguchi, Masashi, Kimura, Hiroyuki, Fukumoto, Shoji
Published in Bioorganic & medicinal chemistry (15.04.2008)
Published in Bioorganic & medicinal chemistry (15.04.2008)
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Evaluation of line-tracing controller of intelligently controllable walker
Kikuchi, Takehito, Tanaka, Toshimasa, Anzai, Kenichi, Kawakami, Sensi, Hosaka, Masayuki, Niino, Kazumi
Published in Advanced robotics (01.05.2013)
Published in Advanced robotics (01.05.2013)
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Discovery of Imidazo[1,5-c]imidazol-3-ones: Weakly Basic, Orally Active Factor Xa Inhibitors
Imaeda, Yasuhiro, Kuroita, Takanobu, Sakamoto, Hiroki, Kawamoto, Tetsuji, Tobisu, Mamoru, Konishi, Noriko, Hiroe, Katsuhiko, Kawamura, Masaki, Tanaka, Toshimasa, Kubo, Keiji
Published in Journal of medicinal chemistry (26.06.2008)
Published in Journal of medicinal chemistry (26.06.2008)
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