Diversity-oriented synthesis as a tool for identifying new modulators of mitosis
Ibbeson, Brett M., Laraia, Luca, Alza, Esther, O' Connor, Cornelius J., Tan, Yaw Sing, Davies, Huw M.L., McKenzie, Grahame, Venkitaraman, Ashok R., Spring, David R.
Published in Nature communications (01.01.2014)
Published in Nature communications (01.01.2014)
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Journal Article
Macrocyclization of an all-d linear alpha-helical peptide imparts cellular permeability
Kannan, Srinivasaraghavan, Aronica, Pietro G. A., Ng, Simon, Lian, Dawn Thean Gek, Frosi, Yuri, Chee, Sharon, Jiang, Shimin, Yuen, Tsz Ying, Sadruddin, Ahmad, Kaan, Hung Yi Kristal, Chandramohan, Arun, Wong, Jin Huei, Tan, Yaw Sing, Chang, Zi Wei, Ferrer-Gago, Fernando J., Arumugam, Prakash, Han, Yi, Chen, Shiying, Renia, Laurent, Brown, Christopher J., Johannes, Charles W., Henry, Brian, Lane, David P., Sawyer, Tomi K., Verma, Chandra S., Partridge, Anthony W.
Published in Chemical science (Cambridge) (07.06.2020)
Published in Chemical science (Cambridge) (07.06.2020)
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Journal Article
Kinetic and thermodynamic effects of phosphorylation on p53 binding to MDM2
Yadahalli, Shilpa, Neira, José L., Johnson, Christopher M., Tan, Yaw Sing, Rowling, Pamela J. E., Chattopadhyay, Anasuya, Verma, Chandra S., Itzhaki, Laura S.
Published in Scientific reports (24.01.2019)
Published in Scientific reports (24.01.2019)
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Journal Article
Stapled peptides as a new technology to investigate protein-protein interactions in human platelets
Iegre, Jessica, Ahmed, Niaz S., Gaynord, Josephine S., Wu, Yuteng, Herlihy, Kara M., Tan, Yaw Sing, Lopes-Pires, Maria E., Jha, Rupam, Lau, Yu Heng, Sore, Hannah F., Verma, Chandra, O'Donovan, Daniel H., Pugh, Nicholas, Spring, David R.
Published in Chemical science (Cambridge) (28.05.2018)
Published in Chemical science (Cambridge) (28.05.2018)
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Journal Article
An intramolecular tryptophan-condensation approach for peptide staplingElectronic supplementary information (ESI) available. See DOI: 10.1039/c7ob02667f
Hui, Eunice Y.-L, Rout, Bhimsen, Tan, Yaw Sing, Verma, Chandra S, Chan, Kok-Ping, Johannes, Charles W
Year of Publication 17.01.2018
Year of Publication 17.01.2018
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Journal Article
Efficient development of stable and highly functionalised peptides targeting the CK2α/CK2β protein–protein interaction† †Electronic supplementary information (ESI) available. See DOI: 10.1039/c9sc00798a
Iegre, Jessica, Brear, Paul, Baker, David J., Tan, Yaw Sing, Atkinson, Eleanor L., Sore, Hannah F., O' Donovan, Daniel H., Verma, Chandra S., Hyvönen, Marko, Spring, David R.
Published in Chemical science (Cambridge) (12.04.2019)
Published in Chemical science (Cambridge) (12.04.2019)
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Journal Article
Benzene Probes in Molecular Dynamics Simulations Reveal Novel Binding Sites for Ligand Design
Tan, Yaw Sing, Reeks, Judith, Brown, Christopher J, Thean, Dawn, Ferrer Gago, Fernando Jose, Yuen, Tsz Ying, Goh, Eunice Tze Leng, Lee, Xue Er Cheryl, Jennings, Claire E, Joseph, Thomas L, Lakshminarayanan, Rajamani, Lane, David P, Noble, Martin E. M, Verma, Chandra S
Published in The journal of physical chemistry letters (01.09.2016)
Published in The journal of physical chemistry letters (01.09.2016)
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Journal Article
The p53-Mdm2 interaction and the E3 ligase activity of Mdm2/Mdm4 are conserved from lampreys to humans
Coffill, Cynthia R, Lee, Alison P, Siau, Jia Wei, Chee, Sharon M, Joseph, Thomas L, Tan, Yaw Sing, Madhumalar, Arumugam, Tay, Boon-Hui, Brenner, Sydney, Verma, Chandra S, Ghadessy, Farid J, Venkatesh, Byrappa, Lane, David P
Published in Genes & development (01.02.2016)
Published in Genes & development (01.02.2016)
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Discovery of a small-molecule binder of the oncoprotein gankyrin that modulates gankyrin activity in the cell
Chattopadhyay, Anasuya, O’Connor, Cornelius J., Zhang, Fengzhi, Galvagnion, Celine, Galloway, Warren R. J. D., Tan, Yaw Sing, Stokes, Jamie E., Rahman, Taufiq, Verma, Chandra, Spring, David R., Itzhaki, Laura S.
Published in Scientific reports (05.04.2016)
Published in Scientific reports (05.04.2016)
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Journal Article
Functional characterization of p53 pathway components in the ancient metazoan Trichoplax adhaerens
Siau, Jia Wei, Coffill, Cynthia R., Zhang, Weiyun Villien, Tan, Yaw Sing, Hundt, Juliane, Lane, David, Verma, Chandra, Ghadessy, Farid
Published in Scientific reports (28.09.2016)
Published in Scientific reports (28.09.2016)
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Journal Article
Stereoisomerism of stapled peptide inhibitors of the p53-Mdm2 interaction: an assessment of synthetic strategies and activity profiles† †Electronic supplementary information (ESI) available. See DOI: 10.1039/c9sc01456j
Yuen, Tsz Ying, Brown, Christopher J., Xue, Yuezhen, Tan, Yaw Sing, Ferrer Gago, Fernando J., Lee, Xue Er, Neo, Jin Yong, Thean, Dawn, Kaan, Hung Yi Kristal, Partridge, Anthony W., Verma, Chandra S., Lane, David P., Johannes, Charles W.
Published in Chemical science (Cambridge) (30.05.2019)
Published in Chemical science (Cambridge) (30.05.2019)
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Journal Article
Macrocyclization of an all-d linear α-helical peptide imparts cellular permeability† †Electronic supplementary information (ESI) available. See DOI: 10.1039/c9sc06383h
Kannan, Srinivasaraghavan, Aronica, Pietro G. A., Ng, Simon, Gek Lian, Dawn Thean, Frosi, Yuri, Chee, Sharon, Shimin, Jiang, Yuen, Tsz Ying, Sadruddin, Ahmad, Kaan, Hung Yi Kristal, Chandramohan, Arun, Wong, Jin Huei, Tan, Yaw Sing, Chang, Zi Wei, Ferrer-Gago, Fernando J., Arumugam, Prakash, Han, Yi, Chen, Shiying, Rénia, Laurent, Brown, Christopher J., Johannes, Charles W., Henry, Brian, Lane, David P., Sawyer, Tomi K., Verma, Chandra S., Partridge, Anthony W.
Published in Chemical science (Cambridge) (11.05.2020)
Published in Chemical science (Cambridge) (11.05.2020)
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Journal Article
Stapled peptides as a new technology to investigate protein-protein interactions in human plateletsElectronic supplementary information (ESI) available. See DOI: 10.1039/c8sc00284c
Iegre, Jessica, Ahmed, Niaz S, Gaynord, Josephine S, Wu, Yuteng, Herlihy, Kara M, Tan, Yaw Sing, Lopes-Pires, Maria E, Jha, Rupam, Lau, Yu Heng, Sore, Hannah F, Verma, Chandra, O' Donovan, Daniel H, Pugh, Nicholas, Spring, David R
Year of Publication 23.05.2018
Year of Publication 23.05.2018
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Journal Article
Stapled peptides as a new technology to investigate protein–protein interactions in human platelets† †Electronic supplementary information (ESI) available. See DOI: 10.1039/c8sc00284c
Iegre, Jessica, Ahmed, Niaz S., Gaynord, Josephine S., Wu, Yuteng, Herlihy, Kara M., Tan, Yaw Sing, Lopes-Pires, Maria E., Jha, Rupam, Lau, Yu Heng, Sore, Hannah F., Verma, Chandra, O' Donovan, Daniel H., Pugh, Nicholas, Spring, David R.
Published in Chemical science (Cambridge) (25.04.2018)
Published in Chemical science (Cambridge) (25.04.2018)
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Journal Article
Role of the N-terminal lid in regulating the interaction of phosphorylated MDMX with p53
Chan, Jane Vin, Ping Koh, Dawn Xin, Liu, Yun, Joseph, Thomas L, Lane, David P, Verma, Chandra S, Tan, Yaw Sing
Published in Oncotarget (22.12.2017)
Published in Oncotarget (22.12.2017)
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Journal Article
Synthesis and biological profiling of tellimagrandin I and analogues reveals that the medium ring can significantly modulate biological activity
Zheng, Shaojun, Laraia, Luca, Connor, Cornelius J. O', Sorrell, David, Tan, Yaw Sing, Xu, Zhaochao, Venkitaraman, Ashok R., Wu, Wenjun, Spring, David R.
Published in Organic & biomolecular chemistry (07.04.2012)
Published in Organic & biomolecular chemistry (07.04.2012)
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