Structural basis for allosteric PARP-1 retention on DNA breaks
Zandarashvili, Levani, Langelier, Marie-France, Velagapudi, Uday Kiran, Hancock, Mark A, Steffen, Jamin D, Billur, Ramya, Hannan, Zain M, Wicks, Andrew J, Krastev, Dragomir B, Pettitt, Stephen J, Lord, Christopher J, Talele, Tanaji T, Pascal, John M, Black, Ben E
Published in Science (American Association for the Advancement of Science) (03.04.2020)
Published in Science (American Association for the Advancement of Science) (03.04.2020)
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The ubiquitin-dependent ATPase p97 removes cytotoxic trapped PARP1 from chromatin
Krastev, Dragomir B, Li, Shudong, Sun, Yilun, Wicks, Andrew J, Hoslett, Gwendoline, Weekes, Daniel, Badder, Luned M, Knight, Eleanor G, Marlow, Rebecca, Pardo, Mercedes Calvo, Yu, Lu, Talele, Tanaji T, Bartek, Jiri, Choudhary, Jyoti S, Pommier, Yves, Pettitt, Stephen J, Tutt, Andrew N J, Ramadan, Kristijan, Lord, Christopher J
Published in Nature cell biology (01.01.2022)
Published in Nature cell biology (01.01.2022)
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Characterization of Solid Dispersion of Itraconazole Prepared by Solubilization in Concentrated Aqueous Solutions of Weak Organic Acids and Drying
Parikh, Tapan, Sandhu, Harpreet K., Talele, Tanaji T., Serajuddin, Abu T. M.
Published in Pharmaceutical research (01.06.2016)
Published in Pharmaceutical research (01.06.2016)
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Nek2 Kinase Signaling in Malaria, Bone, Immune and Kidney Disorders to Metastatic Cancers and Drug Resistance: Progress on Nek2 Inhibitor Development
Dana, Dibyendu, Das, Tuhin, Choi, Athena, Bhuiyan, Ashif I, Das, Tirtha K, Talele, Tanaji T, Pathak, Sanjai K
Published in Molecules (Basel, Switzerland) (06.01.2022)
Published in Molecules (Basel, Switzerland) (06.01.2022)
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Sildenafil Reverses ABCB1- and ABCG2-Mediated Chemotherapeutic Drug Resistance
ZHI SHI, TIWARI, Amit K, TALELE, Tanaji T, FU, Li-Wu, CHEN, Zhe-Sheng, SHUKLA, Suneet, ROBEY, Robert W, SINGH, Satyakam, KIM, In-Wha, BATES, Susan E, XINGXIANG PENG, ABRAHAM, Loana, AMBUDKAR, Suresh V
Published in Cancer research (Chicago, Ill.) (15.04.2011)
Published in Cancer research (Chicago, Ill.) (15.04.2011)
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Bafetinib (INNO-406) reverses multidrug resistance by inhibiting the efflux function of ABCB1 and ABCG2 transporters
Zhang, Yun-Kai, Zhang, Guan-Nan, Wang, Yi-Jun, Patel, Bhargav A, Talele, Tanaji T, Yang, Dong-Hua, Chen, Zhe-Sheng
Published in Scientific reports (09.05.2016)
Published in Scientific reports (09.05.2016)
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Nilotinib potentiates anticancer drug sensitivity in murine ABCB1-, ABCG2-, and ABCC10-multidrug resistance xenograft models
Tiwari, Amit K, Sodani, Kamlesh, Dai, Chun-ling, Abuznait, Alaa H, Singh, Satyakam, Xiao, Zhi-Jie, Patel, Atish, Talele, Tanaji T, Fu, Liwu, Kaddoumi, Amal, Gallo, James M, Chen, Zhe-Sheng
Published in Cancer letters (28.01.2013)
Published in Cancer letters (28.01.2013)
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Recent development in the discovery of PARP inhibitors as anticancer agents: a patent update (2016-2020)
Velagapudi, Uday Kiran, Patel, Bhargav A, Shao, Xuwei, Pathak, Sanjai Kumar, Ferraris, Dana V, Talele, Tanaji T
Published in Expert opinion on therapeutic patents (03.07.2021)
Published in Expert opinion on therapeutic patents (03.07.2021)
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Design and Synthesis of Human ABCB1 (P-Glycoprotein) Inhibitors by Peptide Coupling of Diverse Chemical Scaffolds on Carboxyl and Amino Termini of (S)‑Valine-Derived Thiazole Amino Acid
Singh, Satyakam, Prasad, Nagarajan Rajendra, Chufan, Eduardo E, Patel, Bhargav A, Wang, Yi-Jun, Chen, Zhe-Sheng, Ambudkar, Suresh V, Talele, Tanaji T
Published in Journal of medicinal chemistry (22.05.2014)
Published in Journal of medicinal chemistry (22.05.2014)
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2-O, 3-O desulfated heparin (ODSH) increases bacterial clearance and attenuates lung injury in cystic fibrosis by restoring HMGB1-compromised macrophage function
Wang, Mao, Gauthier, Alex G, Kennedy, Thomas P, Wang, Haichao, Velagapudi, Uday Kiran, Talele, Tanaji T, Lin, Mosi, Wu, Jiaqi, Daley, LeeAnne, Yang, Xiaojing, Patel, Vivek, Mun, Sung Soo, Ashby, Jr, Charles R, Mantell, Lin L
Published in Molecular medicine (Cambridge, Mass.) (16.07.2021)
Published in Molecular medicine (Cambridge, Mass.) (16.07.2021)
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Lamellarin O, a pyrrole alkaloid from an Australian marine sponge, Ianthella sp., reverses BCRP mediated drug resistance in cancer cells
Huang, Xiao-Cong, Xiao, Xue, Zhang, Yun-Kai, Talele, Tanaji T, Salim, Angela A, Chen, Zhe-Sheng, Capon, Robert J
Published in Marine drugs (27.06.2014)
Published in Marine drugs (27.06.2014)
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In Vitro Antibacterial Activity of Rhodanine Derivatives against Pathogenic Clinical Isolates
AbdelKhalek, Ahmed, Ashby, Jr, Charles R, Patel, Bhargav A, Talele, Tanaji T, Seleem, Mohamed N
Published in PloS one (06.10.2016)
Published in PloS one (06.10.2016)
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GW583340 and GW2974, human EGFR and HER-2 inhibitors, reverse ABCG2- and ABCB1-mediated drug resistance
Sodani, Kamlesh, Tiwari, Amit K., Singh, Satyakam, Patel, Atish, Xiao, Zhi-Jie, Chen, Jun-Jiang, Sun, Yue-Li, Talele, Tanaji T., Chen, Zhe-Sheng
Published in Biochemical pharmacology (15.06.2012)
Published in Biochemical pharmacology (15.06.2012)
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2-Heteroarylimino-5-arylidene-4-thiazolidinones as a new class of non-nucleoside inhibitors of HCV NS5B polymerase
Küçükgüzel, İlkay, Satılmış, Gökhan, Gurukumar, K.R., Basu, Amartya, Tatar, Esra, Nichols, Daniel B., Talele, Tanaji T., Kaushik-Basu, Neerja
Published in European journal of medicinal chemistry (01.11.2013)
Published in European journal of medicinal chemistry (01.11.2013)
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Discovery and Structure–Activity Relationship of Novel 2,3-Dihydrobenzofuran-7-carboxamide and 2,3-Dihydrobenzofuran-3(2H)‑one-7-carboxamide Derivatives as Poly(ADP-ribose)polymerase‑1 Inhibitors
Patel, Maulik R, Bhatt, Aaditya, Steffen, Jamin D, Chergui, Adel, Murai, Junko, Pommier, Yves, Pascal, John M, Trombetta, Louis D, Fronczek, Frank R, Talele, Tanaji T
Published in Journal of medicinal chemistry (10.07.2014)
Published in Journal of medicinal chemistry (10.07.2014)
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