Atropisomeric 4‑Phenyl‑4H‑1,2,4-triazoles as Selective Glycine Transporter 1 Inhibitors
Sugane, Takashi, Tobe, Takahiko, Hamaguchi, Wataru, Shimada, Itsuro, Maeno, Kyoichi, Miyata, Junji, Suzuki, Takeshi, Kimizuka, Tetsuya, Sakamoto, Shuichi, Tsukamoto, Shin-ichi
Published in Journal of medicinal chemistry (25.07.2013)
Published in Journal of medicinal chemistry (25.07.2013)
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Journal Article
Consequence of Hapten Stereochemistry: An Efficacious Methamphetamine Vaccine
Olson, Margaret E, Sugane, Takashi, Zhou, Bin, Janda, Kim D
Published in Journal of the American Chemical Society (11.09.2019)
Published in Journal of the American Chemical Society (11.09.2019)
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Journal Article
Catch and Anchor Approach To Combat Both Toxicity and Longevity of Botulinum Toxin A
Lin, Lucy, Olson, Margaret E, Sugane, Takashi, Turner, Lewis D, Tararina, Margarita A, Nielsen, Alexander L, Kurbanov, Elbek K, Pellett, Sabine, Johnson, Eric A, Cohen, Seth M, Allen, Karen N, Janda, Kim D
Published in Journal of medicinal chemistry (08.10.2020)
Published in Journal of medicinal chemistry (08.10.2020)
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Journal Article
Covalent inhibition of botulinum neurotoxin A – Exploration of warhead reactivity and function using a bifunctional approach
Turner, Lewis D., Nielsen, Alexander L., Lin, Lucy, Pellett, Sabine, Sugane, Takashi, Olson, Margaret E., Janda, Kim D.
Published in Toxicon (Oxford) (01.01.2021)
Published in Toxicon (Oxford) (01.01.2021)
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Journal Article
Atropisomeric 4-Phenyl-4 H -1,2,4-triazoles as Selective Glycine Transporter 1 Inhibitors
Sugane, Takashi, Tobe, Takahiko, Hamaguchi, Wataru, Shimada, Itsuro, Maeno, Kyoichi, Miyata, Junji, Suzuki, Takeshi, Kimizuka, Tetsuya, Sakamoto, Shuichi, Tsukamoto, Shin-ichi
Published in Journal of medicinal chemistry (25.07.2013)
Published in Journal of medicinal chemistry (25.07.2013)
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Journal Article
Irreversible inhibition of BoNT/A protease: proximity-driven reactivity contingent upon a bifunctional approach
Turner, Lewis D, Nielsen, Alexander L, Lin, Lucy, Pellett, Sabine, Sugane, Takashi, Olson, Margaret E, Johnson, Eric A, Janda, Kim D
Published in MedChemComm (23.06.2021)
Published in MedChemComm (23.06.2021)
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Journal Article
Synthesis and Biological Evaluation of 3-Biphenyl-4-yl-4-phenyl-4 H -1,2,4-triazoles as Novel Glycine Transporter 1 Inhibitors
Sugane, Takashi, Tobe, Takahiko, Hamaguchi, Wataru, Shimada, Itsuro, Maeno, Kyoichi, Miyata, Junji, Suzuki, Takeshi, Kimizuka, Tetsuya, Kohara, Atsuyuki, Morita, Takuma, Doihara, Hitoshi, Saita, Kyouko, Aota, Masaki, Furutani, Masako, Shimada, Yoshiaki, Hamada, Noritaka, Sakamoto, Shuichi, Tsukamoto, Shin-ichi
Published in Journal of medicinal chemistry (13.01.2011)
Published in Journal of medicinal chemistry (13.01.2011)
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Journal Article
Synthesis and Biological Evaluation of 3-Biphenyl-4-yl-4-phenyl-4H-1,2,4-triazoles as Novel Glycine Transporter 1 Inhibitors
Sugane, Takashi, Tobe, Takahiko, Hamaguchi, Wataru, Shimada, Itsuro, Maeno, Kyoichi, Miyata, Junji, Suzuki, Takeshi, Kimizuka, Tetsuya, Kohara, Atsuyuki, Morita, Takuma, Doihara, Hitoshi, Saita, Kyouko, Aota, Masaki, Furutani, Masako, Shimada, Yoshiaki, Hamada, Noritaka, Sakamoto, Shuichi, Tsukamoto, Shin-ichi
Published in Journal of medicinal chemistry (13.01.2011)
Published in Journal of medicinal chemistry (13.01.2011)
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Journal Article
A versatile and efficient method for the synthesis of benz[a]azulenic enones starting from readily available o-(2-furyl)cycloheptatrienylbenzenes
Sasabe, M, Houda, Y, Takagi, H, Sugane, T, Bo, Yamamura, K
Published in Perkin 1 : an international journal of organic and bio-organic chemistry (01.01.2000)
Published in Perkin 1 : an international journal of organic and bio-organic chemistry (01.01.2000)
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Journal Article
Practical and efficient synthesis of the (R)-atropisomer of a 4-phenyl 1,2,4-triazole derivative as a selective GlyT1 inhibitor
Sugane, Takashi, Hamada, Noritaka, Tobe, Takahiko, Hamaguchi, Wataru, Shimada, Itsuro, Maeno, Kyoichi, Miyata, Junji, Suzuki, Takeshi, Kimizuka, Tetsuya, Sakamoto, Shuichi, Tsukamoto, Shin-ichi
Published in Tetrahedron: asymmetry (15.12.2012)
Published in Tetrahedron: asymmetry (15.12.2012)
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Journal Article
Synthesis and biological evaluation of (4H-1,2,4-triazol-4-yl)isoquinoline derivatives as selective glycine transporter 1 inhibitors
Sugane, Takashi, Tobe, Takahiko, Hamaguchi, Wataru, Shimada, Itsuro, Maeno, Kyoichi, Miyata, Junji, Suzuki, Takeshi, Kimizuka, Tetsuya, Morita, Takuma, Sakamoto, Shuichi, Tsukamoto, Shin-ichi
Published in Bioorganic & medicinal chemistry (01.01.2012)
Published in Bioorganic & medicinal chemistry (01.01.2012)
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Journal Article
Piperazine derivative
Moritomo, Hiroyuki, Sugane, Takashi, Yamashita, Daisuke, Asai, Norio, Hosogai, Naomi
Year of Publication 14.07.2020
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Year of Publication 14.07.2020
Patent
PIPERAZINE DERIVATIVE
MORITOMO, Hiroyuki, SUGANE, Takashi, YAMASHITA, Daisuke, HOSOGAI, Naomi, ASAI, Norio
Year of Publication 04.03.2020
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Year of Publication 04.03.2020
Patent
PIPERAZINE DERIVATIVE
MORITOMO, Hiroyuki, SUGANE, Takashi, YAMASHITA, Daisuke, HOSOGAI, Naomi, ASAI, Norio
Year of Publication 04.07.2019
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Year of Publication 04.07.2019
Patent
PIPERAZINE DERIVATIVE
MORITOMO, Hiroyuki, SUGANE, Takashi, YAMASHITA, Daisuke, HOSOGAI, Naomi, ASAI, Norio
Year of Publication 29.05.2019
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Year of Publication 29.05.2019
Patent