Formulating Amorphous Solid Dispersions: Impact of Inorganic Salts on Drug Release from Tablets Containing Itraconazole-HPMC Extrudate
Takano, Ryusuke, Maurer, Reto, Jacob, Laurence, Stowasser, Frank, Stillhart, Cordula, Page, Susanne
Published in Molecular pharmaceutics (03.08.2020)
Published in Molecular pharmaceutics (03.08.2020)
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Journal Article
Validation of a New Methodology to Create Oral Drugs beyond the Rule of 5 for Intracellular Tough Targets
Ohta, Atsushi, Tanada, Mikimasa, Shinohara, Shojiro, Morita, Yuya, Nakano, Kazuhiko, Yamagishi, Yusuke, Takano, Ryusuke, Kariyuki, Shiori, Iida, Takeo, Matsuo, Atsushi, Ozeki, Kazuhisa, Emura, Takashi, Sakurai, Yuuji, Takano, Koji, Higashida, Atsuko, Kojima, Miki, Muraoka, Terushige, Takeyama, Ryuuichi, Kato, Tatsuya, Kimura, Kaori, Ogawa, Kotaro, Ohara, Kazuhiro, Tanaka, Shota, Kikuchi, Yasufumi, Hisada, Nozomi, Hayashi, Ryuji, Nishimura, Yoshikazu, Nomura, Kenichi, Tachibana, Tatsuhiko, Irie, Machiko, Kawada, Hatsuo, Torizawa, Takuya, Murao, Naoaki, Kotake, Tomoya, Tanaka, Masahiko, Ishikawa, Shiho, Miyake, Taiji, Tamiya, Minoru, Arai, Masako, Chiyoda, Aya, Akai, Sho, Sase, Hitoshi, Kuramoto, Shino, Ito, Toshiya, Shiraishi, Takuya, Kojima, Tetsuo, Iikura, Hitoshi
Published in Journal of the American Chemical Society (08.11.2023)
Published in Journal of the American Chemical Society (08.11.2023)
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Journal Article
Oral absorption of poorly water-soluble drugs: computer simulation of fraction absorbed in humans from a miniscale dissolution test
Takano, Ryusuke, Sugano, Kiyohiko, Higashida, Atsuko, Hayashi, Yoshiki, Machida, Minoru, Aso, Yoshinori, Yamashita, Shinji
Published in Pharmaceutical research (01.06.2006)
Published in Pharmaceutical research (01.06.2006)
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Journal Article
Rate-Limiting Steps of Oral Absorption for Poorly Water-Soluble Drugs in Dogs; Prediction from a Miniscale Dissolution Test and a Physiologically-Based Computer Simulation
Takano, Ryusuke, Furumoto, Kentaro, Shiraki, Koji, Takata, Noriyuki, Hayashi, Yoshiki, Aso, Yoshinori, Yamashita, Shinji
Published in Pharmaceutical research (01.10.2008)
Published in Pharmaceutical research (01.10.2008)
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Journal Article
Cocrystal Screening of Stanolone and Mestanolone Using Slurry Crystallization
Takata, Noriyuki, Shiraki, Koji, Takano, Ryusuke, Hayashi, Yoshiki, Terada, Katsuhide
Published in Crystal growth & design (01.08.2008)
Published in Crystal growth & design (01.08.2008)
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Journal Article
Quantitative Analysis of the Effect of Supersaturation on in Vivo Drug Absorption
Takano, Ryusuke, Takata, Noriyuki, Saito, Ryoichi, Furumoto, Kentaro, Higo, Shoichi, Hayashi, Yoshiki, Machida, Minoru, Aso, Yoshinori, Yamashita, Shinji
Published in Molecular pharmaceutics (04.10.2010)
Published in Molecular pharmaceutics (04.10.2010)
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Journal Article
Effects of spray drying process parameters on the solubility behavior and physical stability of solid dispersions prepared using a laboratory-scale spray dryer
Kojima, Yuki, Ohta, Tomoaki, Shiraki, Kouji, Takano, Ryusuke, Maeda, Hiroyuki, Ogawa, Yutaka
Published in Drug development and industrial pharmacy (01.09.2013)
Published in Drug development and industrial pharmacy (01.09.2013)
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Journal Article
2-Phenylquinoline-Carbohydrate Hybrids: Molecular Design, Chemical Synthesis, and Evaluation of a New Family of Light-Activatable DNA-Cleaving Agents
Toshima, Kazunobu, Takano, Ryusuke, Maeda, Yutaka, Suzuki, Masataka, Asai, Akira, Matsumura, Shuichi
Published in Angewandte Chemie (International ed.) (16.12.1999)
Published in Angewandte Chemie (International ed.) (16.12.1999)
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Journal Article
Chemical Synthesis and DNA Photocleavage of the Intercalator-Carbohydrate Hybrid Moiety of the Neocarzinostatin Chromophore
Toshima, Kazunobu, Takai, Shigeki, Maeda, Yutaka, Takano, Ryusuke, Matsumura, Shuichi
Published in Angewandte Chemie (International ed.) (16.10.2000)
Published in Angewandte Chemie (International ed.) (16.10.2000)
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Journal Article
Integrating drug permeability with dissolution profile to develop IVIVC
Takano, Ryusuke, Kataoka, Makoto, Yamashita, Shinji
Published in Biopharmaceutics & drug disposition (01.10.2012)
Published in Biopharmaceutics & drug disposition (01.10.2012)
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Journal Article