Towards the synthesis of a Yersinia pestis cell wall polysaccharide: enantioselective synthesis of an L-glycero-D-manno-heptose building block
Ohara, Takafumi, Adibekian, Alexander, Esposito, Davide, Stallforth, Pierre, Seeberger, Peter H.
Published in Chemical communications (Cambridge, England) (01.01.2010)
Published in Chemical communications (Cambridge, England) (01.01.2010)
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Development of a Manufacturing Process toward the Convergent Synthesis of the COVID-19 Antiviral Ensitrelvir
Kawajiri, Takahiro, Kijima, Akihito, Iimuro, Atsuhiro, Ohashi, Eisaku, Yamakawa, Katsuya, Agura, Kazushi, Masuda, Kengo, Kouki, Kensuke, Kasamatsu, Koji, Yanagisawa, Shuichi, Nakashima, Sho, Shibahara, Setsuya, Toyota, Takashi, Higuchi, Takafumi, Suto, Takahiro, Oohara, Tadashi, Maki, Toshikatsu, Sahara, Naoto, Fukui, Nobuaki, Wakamori, Hisayuki, Ikemoto, Hidaka, Murakami, Hiroaki, Ando, Hiroyasu, Hosoya, Masahiro, Sato, Mizuki, Suzuki, Yusuke, Nakagawa, Yuta, Unoh, Yuto, Hirano, Yoichi, Nagasawa, Yoshitomo, Goda, Satoshi, Ohara, Takafumi, Tsuritani, Takayuki
Published in ACS central science (26.04.2023)
Published in ACS central science (26.04.2023)
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Journal Article
Synthesis and evaluation of novel pyrimidine-based dual EGFR/Her-2 inhibitors
Suzuki, Naoyuki, Shiota, Takeshi, Watanabe, Fumihiko, Haga, Norihiro, Murashi, Takami, Ohara, Takafumi, Matsuo, Kenji, Oomori, Naoki, Yari, Hiroshi, Dohi, Keiji, Inoue, Makiko, Iguchi, Motofumi, Sentou, Jyunko, Wada, Tooru
Published in Bioorganic & medicinal chemistry letters (15.03.2011)
Published in Bioorganic & medicinal chemistry letters (15.03.2011)
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Highly Screw-Sense Selective Polymerization of 1,2-Diisocyano-3,6-di-p-tolylbenzene Initiated by Optically Active Binaphthylpalladium(II) Complexes
Ito, Yoshihiko, Ohara, Takafumi, Shima, Ryoto, Suginome, Michinori
Published in Journal of the American Chemical Society (25.09.1996)
Published in Journal of the American Chemical Society (25.09.1996)
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Journal Article
Catalytic Activity of Triphenylphosphine for Electrophilic Aromatic Bromination Using N‑Bromosuccinimide and Process Safety Evaluation
Hosoya, Masahiro, Ishibashi, Kenichi, Ohara, Takafumi, Mori, Atsunori, Okano, Kentaro
Published in Organic process research & development (18.10.2024)
Published in Organic process research & development (18.10.2024)
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Stereoselective Synthesis of Baloxavir Marboxil Using Diastereoselective Cyclization and Photoredox Decarboxylation of l‑Serine
Okamoto, Kazuya, Ueno, Tatsuhiko, Hato, Yoshio, Kawaguchi, Yasunori, Hakogi, Toshikazu, Majima, Shohei, Ohara, Takafumi, Hagihara, Motoyuki, Tanimoto, Norihiko, Tsuritani, Takayuki
Published in Journal of organic chemistry (19.07.2024)
Published in Journal of organic chemistry (19.07.2024)
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Practical Manufacturing Process for Baloxavir Marboxil: Effective Selection and Replacement of Protective Group toward Enhancement of Crystallization-Induced Diastereomer Transformation
Fukui, Nobuaki, Shibahara, Setsuya, Maki, Toshikatsu, Ueno, Tatsuhiko, Yanagisawa, Shuichi, Okamoto, Kazuya, Tanimoto, Emi, Ohara, Takafumi, Yasukata, Tatsuro, Tsuritani, Takayuki
Published in Organic process research & development (21.06.2024)
Published in Organic process research & development (21.06.2024)
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Journal Article
Design, Synthesis, and Anti-Inflammatory Evaluation of a Novel PPARδ Agonist with a 4‑(1-Pyrrolidinyl)piperidine Structure
Kato, Terukazu, Fukao, Keita, Ohara, Takafumi, Naya, Noriyuki, Tokuyama, Ryukou, Muto, Susumu, Fukasawa, Hiroshi, Itai, Akiko, Matsumura, Ken-ichi
Published in Journal of medicinal chemistry (24.08.2023)
Published in Journal of medicinal chemistry (24.08.2023)
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Journal Article
Discovery and structure-based design of a new series of potent and selective PPAR6 agonists utilizing a virtual screening method
Kato, Terukazu, Ohara, Takafumi, Suzuki, Naoyuki, Muto, Susumu, Tokuyama, Ryukou, Mizutani, Miho, Fukasawa, Hiroshi, Matsumura, Ken-ichi, Itai, Akiko
Published in Bioorganic & medicinal chemistry letters (01.03.2022)
Published in Bioorganic & medicinal chemistry letters (01.03.2022)
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Journal Article
Discovery and structure-activity relationship study of 2-piperazinyl-benzo- thiazole derivatives as potent and selective PPAR delta; agonists
Kato, Terukazu, Ohara, Takafumi, Suzuki, Naoyuki, Naya, Noriyuki, Fukao, Keita, Tokuyama, Ryukou, Muto, Susumu, Fukasawa, Hiroshi, Itai, Akiko, Matsumura, Ken-ichi
Published in Bioorganic & medicinal chemistry (15.03.2023)
Published in Bioorganic & medicinal chemistry (15.03.2023)
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Journal Article
Discovery and structure-activity relationship study of 2-piperazinyl-benzothiazole derivatives as potent and selective PPARδ agonists
Kato, Terukazu, Ohara, Takafumi, Suzuki, Naoyuki, Naya, Noriyuki, Fukao, Keita, Tokuyama, Ryukou, Muto, Susumu, Fukasawa, Hiroshi, Itai, Akiko, Matsumura, Ken-ichi
Published in Bioorganic & medicinal chemistry (15.03.2023)
Published in Bioorganic & medicinal chemistry (15.03.2023)
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Journal Article
Discovery and structure-based design of a new series of potent and selective PPARδ agonists utilizing a virtual screening method
Kato, Terukazu, Ohara, Takafumi, Suzuki, Naoyuki, Muto, Susumu, Tokuyama, Ryukou, Mizutani, Miho, Fukasawa, Hiroshi, Matsumura, Ken-ichi, Itai, Akiko
Published in Bioorganic & medicinal chemistry letters (01.03.2022)
Published in Bioorganic & medicinal chemistry letters (01.03.2022)
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Journal Article
Discovery of novel 5-alkynyl-4-anilinopyrimidines as potent, orally active dual inhibitors of EGFR and Her-2 tyrosine kinases
Suzuki, Naoyuki, Shiota, Takeshi, Watanabe, Fumihiko, Haga, Norihiro, Murashi, Takami, Ohara, Takafumi, Matsuo, Kenji, Omori, Naoki, Yari, Hiroshi, Dohi, Keiji, Inoue, Makiko, Iguchi, Motofumi, Sentou, Jyunko, Wada, Tooru
Published in Bioorganic & medicinal chemistry letters (01.01.2012)
Published in Bioorganic & medicinal chemistry letters (01.01.2012)
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Journal Article
Towards the synthesis of a Yersinia pestis cell wall polysaccharide: enantioselective synthesis of an l-glycero-d-manno-heptose building blockElectronic supplementary information (ESI) available: General information and procedures (S1-S12) and copies of NMR spectra (S13-S49). See DOI: 10.1039/c000784f
Ohara, Takafumi, Adibekian, Alexander, Esposito, Davide, Stallforth, Pierre, Seeberger, Peter H
Year of Publication 02.06.2010
Year of Publication 02.06.2010
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Journal Article
Asymmetric Synthesis of Helical Poly(quinoxaline-2,3-diyl)s by Palladium-Mediated Polymerization of 1,2-Diisocyanobenzenes: Effective Control of the Screw-Sense by a Binaphthyl Group at the Chain-End
Ito, Yoshihiko, Miyake, Toshiyuki, Hatano, Seiji, Shima, Ryoto, Ohara, Takafumi, Suginome, Michinori
Published in Journal of the American Chemical Society (25.11.1998)
Published in Journal of the American Chemical Society (25.11.1998)
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Journal Article
Long-term follow-up of primary anterior chamber intraocular lens implantation
Sawada, Tatsu, Kimura, Wataru, Kimura, Tohru, Suga, Hideki, Ohte, Akitoshi, Yamanishi, Shigeki, Ohara, Takafumi
Published in Journal of cataract and refractive surgery (01.11.1998)
Published in Journal of cataract and refractive surgery (01.11.1998)
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Journal Article
Conference Proceeding
Novel Antibacterial Macrolides: Synthesis of 15-Membered Diolides
Ohara, Takafumi, Kume, Masaharu, Narukawa, Yukitoshi, Motokawa, Kiyoshi, Uotani, Kouichi, Nakai, Hiroshi
Published in Journal of organic chemistry (27.12.2002)
Published in Journal of organic chemistry (27.12.2002)
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