Structure-based design and optimization of 2-aminothiazole-4-carboxamide as a new class of CHK1 inhibitors
Huang, Xiaohua, Cheng, Cliff C., Fischmann, Thierry O., Duca, José S., Richards, Matthew, Tadikonda, Praveen K., Reddy, Panduranga Adulla, Zhao, Lianyun, Arshad Siddiqui, M., Parry, David, Davis, Nicole, Seghezzi, Wolfgang, Wiswell, Derek, Shipps, Gerald W.
Published in Bioorganic & medicinal chemistry letters (01.05.2013)
Published in Bioorganic & medicinal chemistry letters (01.05.2013)
Get full text
Journal Article
Identification of a Small Molecule Nonpeptide Active Site β-Secretase Inhibitor That Displays a Nontraditional Binding Mode for Aspartyl Proteases
Coburn, Craig A, Stachel, Shawn J, Li, Yue-Ming, Rush, Diane M, Steele, Thomas G, Chen-Dodson, Elizabeth, Holloway, M. Katharine, Xu, Min, Huang, Qian, Lai, Ming-Tain, DiMuzio, Jillian, Crouthamel, Ming-Chih, Shi, Xiao-Ping, Sardana, Vinod, Chen, Zhongguo, Munshi, Sanjeev, Kuo, Lawrence, Makara, Gergely M, Annis, D. Allen, Tadikonda, Praveen K, Nash, Huw M, Vacca, Joseph P, Wang, Tong
Published in Journal of medicinal chemistry (02.12.2004)
Published in Journal of medicinal chemistry (02.12.2004)
Get full text
Journal Article
HETEROCYCLIC AMIDE COMPOUNDS AS PROTEIN KINASE INHIBITORS
TORRES LUIS E, TADIKONDA PRAVEEN K, GUZI TIMOTHY J, SIDDIQUI M. ARSHAD, REDDY PANDURANGA ADULLA P, WONG TZU TSHIN, TANG SHUYI, ZHAO LIANYUN, CAUBLE DAVID F. JR
Year of Publication 03.05.2010
Get full text
Year of Publication 03.05.2010
Patent
2-AMIN0THIAZ0LE-4-CARB0XYLIC AMIDES AS PROTEIN KINASE INHIBITORS
FISCHMANN THIERRY O, TADIKONDA PRAVEEN K, GUZI TIMOTHY J, ZENG HONGBO, REDDY PANDURANGA A, TANG SHUYI, ZHAO LIANYUN, HUANG XIAOHUA, TORRES LUIS E, DWYER MICHAEL P, DUCA JOSE S, SUN BINYUAN, CHENG CLIFF C, SIDDIQUI M. ARSHAD, RICHARDS MATTHEW, SHIPPS GERALD W. JR, KEERTIKAR KARTIK M, WONG TZU T
Year of Publication 30.07.2009
Get full text
Year of Publication 30.07.2009
Patent
ANILINOPIPERAZINE DERIVATIVES AND METHODS OF USE THEREOF
FISCHMANN THIERRY O, TADIKONDA PRAVEEN K, GUZI TIMOTHY J, ZENG HONGBO, REDDY PANDURANGA A, LABROLI MARC M, HUANG XIAOHUA, DUCA JOSE S, SUN BINYUAN, POKER CORY, CHENG CLIFF C, SIDDIQUI M. ARSHAD, RICHARDS MATTHEW, SHIPPS GERALD W. JR, WONG TZU T
Year of Publication 09.07.2009
Get full text
Year of Publication 09.07.2009
Patent
ANILINOPIPERAZINE DERIVATIVES AND METHODS OF USE THEREOF
SIDDIQUI, M., Arshad, POKER, Cory, CHENG, Cliff, C, RICHARDS, Matthew, FISCHMANN, Thierry, O, SHIPPS, Gerald, W., Jr, REDDY, Panduranga, A, LABROLI, Marc, M, HUANG, Xiaohua, GUZI, Timothy, J, ZENG, Hongbo, SUN, Binyuan, DUCA, Jose, S, WONG, Tzu, T, TADIKONDA, Praveen, K
Year of Publication 08.03.2017
Get full text
Year of Publication 08.03.2017
Patent
JNK INHIBITORS
SIDDIQUI, M. ARSHAD, BELANGER, DAVID, B, SHIPPS, GERALD W., JR, MANSOOR, UMAR, FARUK, CURRAN, PATRICK J, TADIKONDA, PRAVEEN, K, REDDY, PANDURANGA, ADULLA, P, HAMANN, BLAKE, ZHAO, LIANYUN
Year of Publication 19.08.2015
Get full text
Year of Publication 19.08.2015
Patent
Compostos de amida heterocíclica como inibidores de proteína cinase
LIANYUN ZHAO, SHUYI TANG, LUIS E. TORRES, TZU TSHIN WONG, DAVID F. CAUBLE, TIMOTHY J. GUZI, M. ARSHAD SIDDIQUI, JR, PANDURANGA ADULLA P. REDDY, PRAVEEN K. TADIKONDA
Year of Publication 14.07.2015
Get full text
Year of Publication 14.07.2015
Patent
Heterocyclic Urea and Thiourea Derivatives and Methods of Use Thereof
TADIKONDA PRAVEEN K, GUZI TIMOTHY J, SIDDIQUI M. ARSHAD, CAUBLE DAVID F
Year of Publication 02.06.2011
Get full text
Year of Publication 02.06.2011
Patent
Anilinopiperazine derivatives and methods of use thereof
FISCHMANN THIERRY O, TADIKONDA PRAVEEN K, REDDY PANDURANGA ADULLA, GUZI TIMOTHY J, ZENG HONGBO, HUANG XIAOHUA, DUCA JOSE S, SUN BINYUAN, SHIPPS, JR. GERALD W, CHENG CLIFF C, SIDDIQUI M. ARSHAD, RICHARDS MATTHEW, LABROLI MARC A, POKER CORY S, WONG TZU T
Year of Publication 08.12.2015
Get full text
Year of Publication 08.12.2015
Patent
HETEROCYCLIC UREA AND THIOUREA DERIVATIVES AND METHODS OF USE THEREOF
SIDDIQUI, ARSHAD, M, TADIKONDA, PRAVEEN, K, GUZI, TIMOTHY, J, CAUBLE, DAVID, F., JR
Year of Publication 28.07.2010
Get full text
Year of Publication 28.07.2010
Patent
Imidazopyrazines as protein kinase inhibitors
TADIKONDA, PRAVEEN K, SIDDIQUI, M. ARSHAD, PARUCH, KAMIL, DWYER, MICHAEL P, REDDY, PANDURANGA A, BELANGER, DAVID B, CURRAN, PATRICK J, GUZI, TIMOTHY. J, HAMANN, BLAKE, ZHAO, LIANYUN
Year of Publication 04.10.2012
Get full text
Year of Publication 04.10.2012
Patent
2-AMINOTHIAZOLE-4-CARBOXYLIC AMIDES AS PROTEIN KINASE INHIBITORS
REDDY, PANDURANGA, A, WONG, TZU, T, DWYER, MICHAEL, P, RICHARDS, MATTHEW, SHIPPS, GERALD, W., JR, KEERTIKAR, KARTIK, M, ZENG, HONGBO, TADIKONDA, PRAVEEN, K, SUN, BINYUAN, GUZI, TIMOTHY, J, ZHAO, LIANYUN, FISCHMANN, THIERRY, O, CHENG, CLIFF, C, HUANG, XIAOHUA, DUCA, JOSE, S, TORRES, LUIS, E, TANG, SHUYI, SIDDIQUI, M., ARSHAD
Year of Publication 25.02.2015
Get full text
Year of Publication 25.02.2015
Patent